JP2015110607A5 - - Google Patents

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Publication number
JP2015110607A5
JP2015110607A5 JP2015003265A JP2015003265A JP2015110607A5 JP 2015110607 A5 JP2015110607 A5 JP 2015110607A5 JP 2015003265 A JP2015003265 A JP 2015003265A JP 2015003265 A JP2015003265 A JP 2015003265A JP 2015110607 A5 JP2015110607 A5 JP 2015110607A5
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JP
Japan
Prior art keywords
oxadiazol
fluorophenyl
benzoic acid
water
crystallizing
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JP2015003265A
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English (en)
Japanese (ja)
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JP6407733B2 (ja
JP2015110607A (ja
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Publication of JP2015110607A5 publication Critical patent/JP2015110607A5/ja
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JP2015003265A 2006-09-25 2015-01-09 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形 Active JP6407733B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US84732606P 2006-09-25 2006-09-25
US60/847,326 2006-09-25

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2009529270A Division JP5714228B2 (ja) 2006-09-25 2007-09-24 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2017106030A Division JP6495375B2 (ja) 2006-09-25 2017-05-29 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形

Publications (3)

Publication Number Publication Date
JP2015110607A JP2015110607A (ja) 2015-06-18
JP2015110607A5 true JP2015110607A5 (enExample) 2017-07-27
JP6407733B2 JP6407733B2 (ja) 2018-10-17

Family

ID=39123850

Family Applications (6)

Application Number Title Priority Date Filing Date
JP2009529270A Active JP5714228B2 (ja) 2006-09-25 2007-09-24 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2015003265A Active JP6407733B2 (ja) 2006-09-25 2015-01-09 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2017106030A Active JP6495375B2 (ja) 2006-09-25 2017-05-29 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2019040137A Withdrawn JP2019104752A (ja) 2006-09-25 2019-03-06 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2021090763A Active JP7245868B2 (ja) 2006-09-25 2021-05-31 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形
JP2023038770A Pending JP2023078271A (ja) 2006-09-25 2023-03-13 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2009529270A Active JP5714228B2 (ja) 2006-09-25 2007-09-24 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2017106030A Active JP6495375B2 (ja) 2006-09-25 2017-05-29 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2019040137A Withdrawn JP2019104752A (ja) 2006-09-25 2019-03-06 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2021090763A Active JP7245868B2 (ja) 2006-09-25 2021-05-31 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形
JP2023038770A Pending JP2023078271A (ja) 2006-09-25 2023-03-13 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形

Country Status (29)

Country Link
US (10) US7863456B2 (enExample)
EP (2) EP2076501B8 (enExample)
JP (6) JP5714228B2 (enExample)
KR (1) KR101430144B1 (enExample)
CN (3) CN102382075B (enExample)
AR (2) AR062963A1 (enExample)
AU (1) AU2007300542B2 (enExample)
BR (1) BRPI0717107A2 (enExample)
CA (1) CA2663574C (enExample)
CL (1) CL2007002743A1 (enExample)
DK (1) DK2076501T3 (enExample)
ES (2) ES2655338T3 (enExample)
HK (1) HK1207070A1 (enExample)
HU (1) HUE028503T2 (enExample)
IL (1) IL197717A (enExample)
LT (1) LTC2076501I2 (enExample)
MX (2) MX344418B (enExample)
MY (1) MY191209A (enExample)
NO (1) NO341858B1 (enExample)
NZ (1) NZ575795A (enExample)
PE (3) PE20120768A1 (enExample)
PL (2) PL2076501T3 (enExample)
PT (1) PT2076501E (enExample)
SG (2) SG185979A1 (enExample)
SI (1) SI2076501T1 (enExample)
TW (2) TWI452038B (enExample)
UA (1) UA99600C2 (enExample)
WO (1) WO2008039431A2 (enExample)
ZA (1) ZA200901949B (enExample)

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ES2683359T3 (es) * 2005-04-08 2018-09-26 Ptc Therapeutics, Inc. Composiciones que comprenden un 1,2,4-oxadiazol y usos de las mismas para tratar enfermedades asociadas con un codón de parada prematura
RU2462246C2 (ru) * 2006-03-30 2012-09-27 ПиТиСи ТЕРАПЬЮТИКС, ИНК. Способы получения функционального белка из днк, имеющей нонсенс-мутацию, и лечения нарушений, ассоциированных с ней
PL2076501T3 (pl) * 2006-09-25 2016-06-30 Ptc Therapeutics Inc Postacie krystaliczne kwasu 3-[5-(2-fluorofenylo)[1,2,4]oksadiazol-3-ilo]-benzoesowego
ES2538359T3 (es) 2006-10-12 2015-06-19 Ptc Therapeutics, Inc. Métodos para administrar un 1,2,4-oxadiazol activo por vía oral para terapia de supresión de mutación sin sentido
KR101713453B1 (ko) 2010-03-12 2017-03-07 오메로스 코포레이션 Pde10 억제제 및 관련 조성물 및 방법
WO2014153643A1 (en) * 2013-03-26 2014-10-02 The University Of British Columbia Compositions and methods for use thereof in the treatment of aniridia
CN105324467B (zh) 2013-04-03 2018-03-20 Gfo油有限责任公司 从有机种子油产生乙醛的方法和系统
DK3363790T3 (da) 2013-09-06 2020-04-27 Aurigene Discovery Tech Ltd 1,2,4-oxadiazolderivater som immunmodulatorer
CA3174516A1 (en) 2014-03-06 2015-09-11 Ptc Therapeutics, Inc. Pharmaceutical compositions and salts of a 1,2,4-oxadiazole benzoic acid
NZ630810A (en) 2014-04-28 2016-03-31 Omeros Corp Processes and intermediates for the preparation of a pde10 inhibitor
NZ716462A (en) * 2014-04-28 2017-11-24 Omeros Corp Optically active pde10 inhibitor
KR101703137B1 (ko) 2014-05-30 2017-02-07 선문대학교 산학협력단 당 부가 아미노글리코사이드 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 약학적 조성물
CN105461650B (zh) * 2014-09-12 2018-04-13 杭州普晒医药科技有限公司 一种噁二唑化合物的溶剂化物及其制备方法
CU24509B1 (es) 2015-03-10 2021-05-12 Aurigene Discovery Tech Ltd Compuestos de 1,2,4-oxadiazol y tiadiazol como inmunomoduladores
CA2980801A1 (en) 2015-04-24 2016-10-27 Omeros Corporation Pde10 inhibitors and related compositions and methods
TW201729807A (zh) 2015-10-30 2017-09-01 Ptc治療公司 用於治療癲癇的方法
CA3003611C (en) 2015-11-04 2022-11-01 Omeros Corporation Solid state forms of a pde10 inhibitor
EP3442512A4 (en) * 2016-04-15 2020-07-22 The UAB Research Foundation METHODS AND COMPOUNDS FOR STIMULATING THE TRANSLECTURE OF PREMATURE TERMINATION CODONS
EP3512516A1 (en) * 2016-09-13 2019-07-24 Marco Cipolli Method of treatment of shwachman-diamond syndrome
WO2019061324A1 (en) 2017-09-29 2019-04-04 Curis Inc. CRYSTALLINE FORMS OF IMMUNOMODULATORS
KR20240151258A (ko) 2017-10-11 2024-10-17 오리진 온콜로지 리미티드 3-치환된 1,2,4-옥사다이아졸의 결정질 형태
EA202090746A1 (ru) 2017-11-03 2020-08-17 Ориджен Дискавери Текнолоджис Лимитед Двойные ингибиторы путей tim-3 и pd-1
CN111386128A (zh) 2017-11-06 2020-07-07 奥瑞基尼探索技术有限公司 用于免疫调节的联合疗法
MX2021012428A (es) 2019-04-10 2022-01-19 Ptc Therapeutics Inc Metodo para el tratamiento de distrofia muscular de duchenne mediada por mutacion sin sentido en pacientes pediatricos.
JP7339900B2 (ja) * 2020-02-26 2023-09-06 新 井上 視野異常診断方法、視野異常診断装置
KR102665711B1 (ko) * 2021-12-21 2024-05-14 재단법인 아산사회복지재단 Ras 활성도를 이용한 신경섬유종증 치료제에 대한 감수성 예측용 바이오마커 조성물 및 Ras 활성 억제제를 포함하는 신경섬유종증 예방 또는 치료용 약학적 조성물
WO2025110781A1 (ko) * 2023-11-24 2025-05-30 재단법인 아산사회복지재단 Ampd3를 포함하는 신경섬유종증 치료제에 대한 감수성 예측용 바이오마커 조성물 및 ampd3 저해제를 포함하는 신경섬유종증 예방 또는 치료용 약학 조성물
CN118178408A (zh) * 2024-03-22 2024-06-14 核工业总医院 Ptc124在制备治疗血小板无力症的药物中的应用

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PL2076501T3 (pl) * 2006-09-25 2016-06-30 Ptc Therapeutics Inc Postacie krystaliczne kwasu 3-[5-(2-fluorofenylo)[1,2,4]oksadiazol-3-ilo]-benzoesowego
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