JP5714228B2 - 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形 - Google Patents

3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形 Download PDF

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JP5714228B2
JP5714228B2 JP2009529270A JP2009529270A JP5714228B2 JP 5714228 B2 JP5714228 B2 JP 5714228B2 JP 2009529270 A JP2009529270 A JP 2009529270A JP 2009529270 A JP2009529270 A JP 2009529270A JP 5714228 B2 JP5714228 B2 JP 5714228B2
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disease
cancer
fluorophenyl
benzoic acid
oxadiazol
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JP2010504340A (ja
JP2010504340A5 (enExample
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ジー.アルムステアド ネイル
ジー.アルムステアド ネイル
セオングウォオ フワング ペテル
セオングウォオ フワング ペテル
モオン ヨウング‐チョオン
モオン ヨウング‐チョオン
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PTC Therapeutics Inc
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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JP2009529270A 2006-09-25 2007-09-24 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形 Active JP5714228B2 (ja)

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US84732606P 2006-09-25 2006-09-25
US60/847,326 2006-09-25
PCT/US2007/020633 WO2008039431A2 (en) 2006-09-25 2007-09-24 Crystalline forms of 3-[5-(2-fhjorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid

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JP2015003265A Division JP6407733B2 (ja) 2006-09-25 2015-01-09 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形

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JP2010504340A JP2010504340A (ja) 2010-02-12
JP2010504340A5 JP2010504340A5 (enExample) 2010-11-11
JP5714228B2 true JP5714228B2 (ja) 2015-05-07

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JP2009529270A Active JP5714228B2 (ja) 2006-09-25 2007-09-24 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2015003265A Active JP6407733B2 (ja) 2006-09-25 2015-01-09 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2017106030A Active JP6495375B2 (ja) 2006-09-25 2017-05-29 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2019040137A Withdrawn JP2019104752A (ja) 2006-09-25 2019-03-06 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2021090763A Active JP7245868B2 (ja) 2006-09-25 2021-05-31 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形
JP2023038770A Pending JP2023078271A (ja) 2006-09-25 2023-03-13 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形

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JP2017106030A Active JP6495375B2 (ja) 2006-09-25 2017-05-29 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2019040137A Withdrawn JP2019104752A (ja) 2006-09-25 2019-03-06 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形
JP2021090763A Active JP7245868B2 (ja) 2006-09-25 2021-05-31 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形
JP2023038770A Pending JP2023078271A (ja) 2006-09-25 2023-03-13 3-[5-(2-フルオロフェニル)-[1,2,4]オキサジアゾール-3-イル]-安息香酸の結晶形

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US (10) US7863456B2 (enExample)
EP (2) EP2559689B1 (enExample)
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KR (1) KR101430144B1 (enExample)
CN (3) CN104341371A (enExample)
AR (2) AR062963A1 (enExample)
AU (1) AU2007300542B2 (enExample)
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NZ (1) NZ575795A (enExample)
PE (3) PE20081225A1 (enExample)
PL (2) PL2559689T3 (enExample)
PT (1) PT2076501E (enExample)
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2015110607A (ja) * 2006-09-25 2015-06-18 ピーティーシー セラピューティクス,インコーポレーテッド 3−[5−(2−フルオロフェニル)−[1,2,4]オキサジアゾール−3−イル]−安息香酸の結晶形

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EP2387995A1 (en) * 2006-03-30 2011-11-23 PTC Therapeutics, Inc. Methods for the production of functional protein from DNA having a nonsense mutation and the treatment of disorders associated therewith
KR20170100072A (ko) 2006-10-12 2017-09-01 피티씨 테라퓨틱스, 인크. 넌센스 돌연변이 억제 치료를 위한 경구 활성 1,2,4-옥사디아졸의 투여 방법
NZ601967A (en) 2010-03-12 2015-03-27 Omeros Corp Pde10 inhibitors and related compositions and methods
WO2014153643A1 (en) * 2013-03-26 2014-10-02 The University Of British Columbia Compositions and methods for use thereof in the treatment of aniridia
US9347014B2 (en) 2013-04-03 2016-05-24 Gfo Oil Llc Methods and systems for generating aldehydes from organic seed oils
RS57508B1 (sr) 2013-09-06 2018-10-31 Aurigene Discovery Tech Ltd 1,2,4-derivati oksadiazola kao imunomodulatori
WO2015134711A1 (en) * 2014-03-06 2015-09-11 Ptc Therapeutics, Inc. Pharmaceutical compositions and salts of a 1,2,4-oxadiazole benzoic acid
NZ716462A (en) 2014-04-28 2017-11-24 Omeros Corp Optically active pde10 inhibitor
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KR101703137B1 (ko) 2014-05-30 2017-02-07 선문대학교 산학협력단 당 부가 아미노글리코사이드 화합물, 이의 제조방법 및 이를 유효성분으로 함유하는 약학적 조성물
CN105461650B (zh) * 2014-09-12 2018-04-13 杭州普晒医药科技有限公司 一种噁二唑化合物的溶剂化物及其制备方法
KR102894264B1 (ko) 2015-03-10 2025-12-02 오리진 온콜로지 리미티드 면역조절제로서의 1,2,4-옥사다이아졸 및 티아다이아졸 화합물
CA2980801A1 (en) 2015-04-24 2016-10-27 Omeros Corporation Pde10 inhibitors and related compositions and methods
TW201729807A (zh) 2015-10-30 2017-09-01 Ptc治療公司 用於治療癲癇的方法
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US10960018B2 (en) * 2016-04-15 2021-03-30 The Uab Research Foundation Methods and compounds for stimulating read-through of premature termination codons
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WO2019061324A1 (en) 2017-09-29 2019-04-04 Curis Inc. CRYSTALLINE FORMS OF IMMUNOMODULATORS
AU2018348350B2 (en) 2017-10-11 2024-05-02 Aurigene Oncology Limited Crystalline forms of 3-substituted 1,2,4-oxadiazole
MX2020004531A (es) 2017-11-03 2020-08-03 Aurigene Discovery Tech Ltd Inhibidores dobles de tim-3 y las vias de pd-1.
EP3706798A1 (en) 2017-11-06 2020-09-16 Aurigene Discovery Technologies Limited Conjoint therapies for immunomodulation
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