SG10201609581TA - Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid - Google Patents

Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid

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Publication number
SG10201609581TA
SG10201609581TA SG10201609581TA SG10201609581TA SG10201609581TA SG 10201609581T A SG10201609581T A SG 10201609581TA SG 10201609581T A SG10201609581T A SG 10201609581TA SG 10201609581T A SG10201609581T A SG 10201609581TA SG 10201609581T A SG10201609581T A SG 10201609581TA
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Singapore
Prior art keywords
oxadiazol
fluorophenyl
benzoic acid
crystalline forms
crystalline
Prior art date
Application number
SG10201609581TA
Inventor
Neil G Almstead
Peter Seongwoo Hwang
Young-Choon Moon
Original Assignee
Ptc Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Ptc Therapeutics Inc filed Critical Ptc Therapeutics Inc
Publication of SG10201609581TA publication Critical patent/SG10201609581TA/en

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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D271/00Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/061,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
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SG10201609581TA 2006-09-25 2007-09-24 Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid SG10201609581TA (en)

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US84732606P 2006-09-25 2006-09-25

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SG10201609581TA true SG10201609581TA (en) 2016-12-29

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SG2012082715A SG185979A1 (en) 2006-09-25 2007-09-24 Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid
SG10201609581TA SG10201609581TA (en) 2006-09-25 2007-09-24 Crystalline forms of 3-[5-(2-fluorophenyl)-[1,2,4]oxadiazol-3-yl]-benzoic acid

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US (10) US7863456B2 (en)
EP (2) EP2559689B1 (en)
JP (6) JP5714228B2 (en)
KR (1) KR101430144B1 (en)
CN (3) CN102382075B (en)
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CN102382075B (en) 2015-10-28
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AR109300A2 (en) 2018-11-14
JP2021130697A (en) 2021-09-09
WO2008039431A3 (en) 2008-05-08
EP2076501B1 (en) 2015-12-02
HUE028503T2 (en) 2016-12-28
PE20081225A1 (en) 2008-09-04
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US20130158081A1 (en) 2013-06-20
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US20190231754A1 (en) 2019-08-01
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US20110040100A1 (en) 2011-02-17
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