JP2014507445A5 - - Google Patents

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Publication number
JP2014507445A5
JP2014507445A5 JP2013555599A JP2013555599A JP2014507445A5 JP 2014507445 A5 JP2014507445 A5 JP 2014507445A5 JP 2013555599 A JP2013555599 A JP 2013555599A JP 2013555599 A JP2013555599 A JP 2013555599A JP 2014507445 A5 JP2014507445 A5 JP 2014507445A5
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JP
Japan
Prior art keywords
compound
alkyl
aryl
heteroaryl
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2013555599A
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English (en)
Japanese (ja)
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JP2014507445A (ja
JP6043733B2 (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2012/026517 external-priority patent/WO2012116279A1/en
Publication of JP2014507445A publication Critical patent/JP2014507445A/ja
Publication of JP2014507445A5 publication Critical patent/JP2014507445A5/ja
Application granted granted Critical
Publication of JP6043733B2 publication Critical patent/JP6043733B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2013555599A 2011-02-25 2012-02-24 カンナビノイド受容体モジュレーター Expired - Fee Related JP6043733B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161446729P 2011-02-25 2011-02-25
US61/446,729 2011-02-25
PCT/US2012/026517 WO2012116279A1 (en) 2011-02-25 2012-02-24 Cannabinoid receptor modulators

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016221615A Division JP2017039773A (ja) 2011-02-25 2016-11-14 カンナビノイド受容体モジュレーター

Publications (3)

Publication Number Publication Date
JP2014507445A JP2014507445A (ja) 2014-03-27
JP2014507445A5 true JP2014507445A5 (enExample) 2015-04-09
JP6043733B2 JP6043733B2 (ja) 2016-12-14

Family

ID=46000314

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2013555599A Expired - Fee Related JP6043733B2 (ja) 2011-02-25 2012-02-24 カンナビノイド受容体モジュレーター
JP2016221615A Withdrawn JP2017039773A (ja) 2011-02-25 2016-11-14 カンナビノイド受容体モジュレーター
JP2018106019A Withdrawn JP2018162260A (ja) 2011-02-25 2018-06-01 カンナビノイド受容体モジュレーター
JP2020028389A Withdrawn JP2020079302A (ja) 2011-02-25 2020-02-21 カンナビノイド受容体モジュレーター
JP2022029449A Pending JP2022066289A (ja) 2011-02-25 2022-02-28 カンナビノイド受容体モジュレーター

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2016221615A Withdrawn JP2017039773A (ja) 2011-02-25 2016-11-14 カンナビノイド受容体モジュレーター
JP2018106019A Withdrawn JP2018162260A (ja) 2011-02-25 2018-06-01 カンナビノイド受容体モジュレーター
JP2020028389A Withdrawn JP2020079302A (ja) 2011-02-25 2020-02-21 カンナビノイド受容体モジュレーター
JP2022029449A Pending JP2022066289A (ja) 2011-02-25 2022-02-28 カンナビノイド受容体モジュレーター

Country Status (11)

Country Link
US (6) US20140206649A1 (enExample)
EP (2) EP2678318A1 (enExample)
JP (5) JP6043733B2 (enExample)
CN (2) CN103492369B (enExample)
AU (1) AU2012222149B2 (enExample)
DK (1) DK3385252T3 (enExample)
ES (1) ES2929977T3 (enExample)
IL (2) IL227779A0 (enExample)
MX (2) MX346644B (enExample)
PT (1) PT3385252T (enExample)
WO (1) WO2012116279A1 (enExample)

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CN102596913B (zh) * 2009-08-28 2016-11-09 艾尼纳制药公司 大麻素受体调节剂
EA035989B1 (ru) 2011-02-25 2020-09-09 Арена Фармасьютикалз, Инк. Кристаллические формы и способы получения модуляторов каннабиноидного рецептора
JP6043733B2 (ja) 2011-02-25 2016-12-14 アリーナ ファーマシューティカルズ， インコーポレイテッド カンナビノイド受容体モジュレーター
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US10172797B2 (en) 2013-12-17 2019-01-08 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
US9492444B2 (en) 2013-12-17 2016-11-15 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
DK3169315T3 (da) 2014-07-17 2020-08-10 Pharmaceutical Manufacturing Res Services In Væskefyldt doseringsform til forhindring af misbrug med øjeblikkelig frigivelse
EP3209282A4 (en) 2014-10-20 2018-05-23 Pharmaceutical Manufacturing Research Services, Inc. Extended release abuse deterrent liquid fill dosage form
EA201892280A1 (ru) * 2016-04-10 2019-04-30 Арена Фармасьютикалз, Инк. Способы лечения селективными агонистами cb-рецептора
MX2019013311A (es) 2017-05-08 2020-08-03 Arena Pharm Inc Compuestos y metodos para el tratamiento del dolor visceral.
TWI768464B (zh) * 2019-09-12 2022-06-21 大陸商四川海思科製藥有限公司 三環吡唑衍生物及其製備
WO2021047581A1 (zh) * 2019-09-12 2021-03-18 四川海思科制药有限公司 一种六氢化苯并吡唑衍生物及其制备
CN112055360B (zh) * 2020-09-07 2024-09-17 中兴通讯股份有限公司 资源确定、配置方法、装置、通信节点及存储介质
WO2023081857A1 (en) 2021-11-04 2023-05-11 Skyhawk Therapeutics, Inc. Condensed pyridazine amine derivatives treating sca3
WO2023212239A1 (en) 2022-04-27 2023-11-02 Skyhawk Therapeutics, Inc. Compositions useful for modulating splicing
WO2023220435A1 (en) 2022-05-12 2023-11-16 Skyhawk Therapeutics, Inc. Compositions useful for modulating splicing

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WO2012116277A1 (en) 2011-02-25 2012-08-30 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
JP6043733B2 (ja) 2011-02-25 2016-12-14 アリーナ ファーマシューティカルズ， インコーポレイテッド カンナビノイド受容体モジュレーター
WO2012116278A1 (en) 2011-02-25 2012-08-30 Arena Pharmaceuticals, Inc. Cannabinoid receptor modulators
EA035989B1 (ru) * 2011-02-25 2020-09-09 Арена Фармасьютикалз, Инк. Кристаллические формы и способы получения модуляторов каннабиноидного рецептора

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