CN103492369B - 大麻素受体调节剂 - Google Patents

大麻素受体调节剂 Download PDF

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Publication number
CN103492369B
CN103492369B CN201280020334.4A CN201280020334A CN103492369B CN 103492369 B CN103492369 B CN 103492369B CN 201280020334 A CN201280020334 A CN 201280020334A CN 103492369 B CN103492369 B CN 103492369B
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compound
dimethyl
tetrahydro
diaza
amide
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Expired - Fee Related
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CN201280020334.4A
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Chinese (zh)
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CN103492369A (zh
Inventor
J.萨特
A.C.布莱克本
韩相敦
R.M.琼斯
郑宰奎
安东尼奥·加利多·蒙塔尔班
B.B.帕尔
J.K.鲁特
S.斯特拉-普莱内特
L.索雷森
熊意风
岳大伟
朱秀文
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Arena Pharmaceuticals Inc
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Arena Pharmaceuticals Inc
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    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
    • A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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    • A61K31/33—Heterocyclic compounds
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/66—Phosphorus compounds
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

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  • Urology & Nephrology (AREA)
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CN201280020334.4A 2011-02-25 2012-02-24 大麻素受体调节剂 Expired - Fee Related CN103492369B (zh)

Priority Applications (1)

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CN201910180370.0A CN109970708B (zh) 2011-02-25 2012-02-24 大麻素受体调节剂

Applications Claiming Priority (3)

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US201161446729P 2011-02-25 2011-02-25
US61/446,729 2011-02-25
PCT/US2012/026517 WO2012116279A1 (en) 2011-02-25 2012-02-24 Cannabinoid receptor modulators

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CN103492369A CN103492369A (zh) 2014-01-01
CN103492369B true CN103492369B (zh) 2019-03-29

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US (6) US20140206649A1 (enExample)
EP (2) EP2678318A1 (enExample)
JP (5) JP6043733B2 (enExample)
CN (2) CN103492369B (enExample)
AU (1) AU2012222149B2 (enExample)
DK (1) DK3385252T3 (enExample)
ES (1) ES2929977T3 (enExample)
IL (2) IL227779A0 (enExample)
MX (2) MX346644B (enExample)
PT (1) PT3385252T (enExample)
WO (1) WO2012116279A1 (enExample)

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