JP2011520977A5 - - Google Patents

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Publication number
JP2011520977A5
JP2011520977A5 JP2011510691A JP2011510691A JP2011520977A5 JP 2011520977 A5 JP2011520977 A5 JP 2011520977A5 JP 2011510691 A JP2011510691 A JP 2011510691A JP 2011510691 A JP2011510691 A JP 2011510691A JP 2011520977 A5 JP2011520977 A5 JP 2011520977A5
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JP
Japan
Prior art keywords
composition
pharmaceutically acceptable
solvate
compound
acceptable salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2011510691A
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English (en)
Japanese (ja)
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JP2011520977A (ja
JP5757864B2 (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2009/044743 external-priority patent/WO2009143295A1/en
Publication of JP2011520977A publication Critical patent/JP2011520977A/ja
Publication of JP2011520977A5 publication Critical patent/JP2011520977A5/ja
Application granted granted Critical
Publication of JP5757864B2 publication Critical patent/JP5757864B2/ja
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2011510691A 2008-05-20 2009-05-20 水溶性アセトアミノフェン類似体 Expired - Fee Related JP5757864B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5477408P 2008-05-20 2008-05-20
US61/054,774 2008-05-20
PCT/US2009/044743 WO2009143295A1 (en) 2008-05-20 2009-05-20 Water-soluble acetaminophen analogs

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014049672A Division JP2014111658A (ja) 2008-05-20 2014-03-13 水溶性アセトアミノフェン類似体

Publications (3)

Publication Number Publication Date
JP2011520977A JP2011520977A (ja) 2011-07-21
JP2011520977A5 true JP2011520977A5 (enExample) 2012-07-05
JP5757864B2 JP5757864B2 (ja) 2015-08-05

Family

ID=41340538

Family Applications (6)

Application Number Title Priority Date Filing Date
JP2011510691A Expired - Fee Related JP5757864B2 (ja) 2008-05-20 2009-05-20 水溶性アセトアミノフェン類似体
JP2014049672A Withdrawn JP2014111658A (ja) 2008-05-20 2014-03-13 水溶性アセトアミノフェン類似体
JP2016016971A Expired - Fee Related JP6063072B2 (ja) 2008-05-20 2016-02-01 水溶性アセトアミノフェン類似体
JP2016242968A Withdrawn JP2017057217A (ja) 2008-05-20 2016-12-15 水溶性アセトアミノフェン類似体
JP2018098716A Withdrawn JP2018135392A (ja) 2008-05-20 2018-05-23 水溶性アセトアミノフェン類似体
JP2020074690A Withdrawn JP2020114876A (ja) 2008-05-20 2020-04-20 水溶性アセトアミノフェン類似体

Family Applications After (5)

Application Number Title Priority Date Filing Date
JP2014049672A Withdrawn JP2014111658A (ja) 2008-05-20 2014-03-13 水溶性アセトアミノフェン類似体
JP2016016971A Expired - Fee Related JP6063072B2 (ja) 2008-05-20 2016-02-01 水溶性アセトアミノフェン類似体
JP2016242968A Withdrawn JP2017057217A (ja) 2008-05-20 2016-12-15 水溶性アセトアミノフェン類似体
JP2018098716A Withdrawn JP2018135392A (ja) 2008-05-20 2018-05-23 水溶性アセトアミノフェン類似体
JP2020074690A Withdrawn JP2020114876A (ja) 2008-05-20 2020-04-20 水溶性アセトアミノフェン類似体

Country Status (12)

Country Link
US (4) US20110212926A1 (enExample)
EP (1) EP2291348A4 (enExample)
JP (6) JP5757864B2 (enExample)
KR (1) KR101698028B1 (enExample)
CN (2) CN105254662A (enExample)
AU (1) AU2009249067A1 (enExample)
BR (1) BRPI0912326A2 (enExample)
CA (1) CA2724877C (enExample)
IL (1) IL209382A0 (enExample)
MX (1) MX2010012648A (enExample)
RU (1) RU2010151952A (enExample)
WO (1) WO2009143295A1 (enExample)

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EP2285419A4 (en) 2008-05-20 2012-05-02 Neurogesx Inc LUBRICANT MUTUAL PARACETAMOL PRODRUGS
KR101677126B1 (ko) 2008-05-20 2016-11-22 노이로제스엑스, 인코포레이티드 탄산염 프로드러그 및 그것의 사용 방법
CA2724877C (en) 2008-05-20 2016-09-13 Neurogesx, Inc. Water-soluble acetaminophen analogs
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JP6029670B2 (ja) 2011-09-22 2016-11-24 アコーダ セラピューティクス、インク． アセトアミノフェンコンジュゲートおよびその組成物ならびにその使用方法
CA3042642A1 (en) 2013-08-12 2015-02-19 Pharmaceutical Manufacturing Research Services, Inc. Extruded immediate release abuse deterrent pill
US9492444B2 (en) 2013-12-17 2016-11-15 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
US10172797B2 (en) 2013-12-17 2019-01-08 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
AU2015290098B2 (en) 2014-07-17 2018-11-01 Pharmaceutical Manufacturing Research Services, Inc. Immediate release abuse deterrent liquid fill dosage form
EP4578865A3 (en) 2014-08-12 2025-07-30 Monash University Lymph directing prodrugs
US20160106737A1 (en) 2014-10-20 2016-04-21 Pharmaceutical Manufacturing Research Services, Inc. Extended Release Abuse Deterrent Liquid Fill Dosage Form
RU2021103000A (ru) 2014-10-21 2021-03-01 Эббви Инк. Пролекарства карбидопа и l-dopa и их применение для лечения болезни паркинсона
WO2016141065A1 (en) * 2015-03-03 2016-09-09 Kindred Biosciences, Inc. Compositions and methods for treatment and prevention of pyrexia in horses
JP7118888B2 (ja) 2015-09-08 2022-08-16 モナッシュ ユニバーシティ リンパ指向性プロドラッグ
JP2019515908A (ja) * 2016-04-20 2019-06-13 アッヴィ・インコーポレイテッド カルビドパ及びｌ−ドパプロドラッグ並びに使用方法
EP3675838A4 (en) 2017-08-29 2021-04-21 PureTech LYT, Inc. LIPID PRODRUGS DIRECTED TO THE LYMPHATIC SYSTEM
US11883497B2 (en) 2017-08-29 2024-01-30 Puretech Lyt, Inc. Lymphatic system-directing lipid prodrugs
WO2019126378A1 (en) 2017-12-19 2019-06-27 Ariya Therapeutics, Inc. Lipid prodrugs of mycophenolic acid and uses thereof
US11608345B1 (en) 2017-12-19 2023-03-21 Puretech Lyt, Inc. Lipid prodrugs of rapamycin and its analogs and uses thereof
US11304954B2 (en) 2017-12-19 2022-04-19 Puretech Lyt, Inc. Lipid prodrugs of mycophenolic acid and uses thereof
WO2020051585A1 (en) 2018-09-07 2020-03-12 R.P. Scherer Technologies, Llc Solid or semisolid lipid based dosage form stabilization through curing and addition of low hlb surfactant(s)
EP3880210A1 (en) 2018-11-15 2021-09-22 Abbvie Inc. Pharmaceutical formulations for subcutaneous administration
US11389409B2 (en) * 2019-08-30 2022-07-19 Remedy Diagnostics LLC Transdermal device comprising acetaminophen prodrug
CA3166908A1 (en) 2020-02-05 2021-08-12 Daniel Kenneth BONNER Lipid prodrugs of neurosteroids

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CA2724877C (en) 2008-05-20 2016-09-13 Neurogesx, Inc. Water-soluble acetaminophen analogs
EP2285419A4 (en) 2008-05-20 2012-05-02 Neurogesx Inc LUBRICANT MUTUAL PARACETAMOL PRODRUGS
KR101677126B1 (ko) 2008-05-20 2016-11-22 노이로제스엑스, 인코포레이티드 탄산염 프로드러그 및 그것의 사용 방법
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JP6029670B2 (ja) 2011-09-22 2016-11-24 アコーダ セラピューティクス、インク． アセトアミノフェンコンジュゲートおよびその組成物ならびにその使用方法

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