JP2014501780A - ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法 - Google Patents

ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法 Download PDF

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JP2014501780A
JP2014501780A JP2013548455A JP2013548455A JP2014501780A JP 2014501780 A JP2014501780 A JP 2014501780A JP 2013548455 A JP2013548455 A JP 2013548455A JP 2013548455 A JP2013548455 A JP 2013548455A JP 2014501780 A JP2014501780 A JP 2014501780A
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phenyl
chloro
tetrahydro
pyran
triol
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チンリン チェン
ナセル エヌ． ニャムウェヤ
ケネス ケー． エイチ． オン
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レクシコン ファーマシューティカルズ インコーポレイテッド
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JP2013548455A 2011-01-05 2012-01-03 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法 Pending JP2014501780A (ja)

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US201161430027P 2011-01-05 2011-01-05
US61/430,027 2011-01-05
PCT/US2012/020042 WO2012094293A1 (en) 2011-01-05 2012-01-03 Compositions comprising and methods of using inhibitors of sodium-glucose cotransporters 1 and 2

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JP2017019445A Division JP6682460B2 (ja) 2011-01-05 2017-02-06 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法

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JP2014501780A true JP2014501780A (ja) 2014-01-23
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JP2013548455A Pending JP2014501780A (ja) 2011-01-05 2012-01-03 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法
JP2017019445A Active JP6682460B2 (ja) 2011-01-05 2017-02-06 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法
JP2018218925A Pending JP2019048866A (ja) 2011-01-05 2018-11-22 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法

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JP2018218925A Pending JP2019048866A (ja) 2011-01-05 2018-11-22 ナトリウム−グルコース共輸送体１及びナトリウム−グルコース共輸送体２の阻害剤を含む組成物、並びに該阻害剤を使用する方法

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EP (1) EP2661256B1 (enExample)
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KR (1) KR102024204B1 (enExample)
CN (1) CN103458875A (enExample)
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WO2018231702A1 (en) 2017-06-13 2018-12-20 The Regents Of The University Of California Methods of improving cell-based therapy
CN107540685B (zh) * 2017-09-04 2020-05-05 杭州科巢生物科技有限公司 一种Sotagliflozin的制备方法及其中间体
EP3456320A1 (de) * 2017-09-15 2019-03-20 Stada Arzneimittel Ag Dpp-4-inhibitor-mono-zusammensetzung
EP3712147B8 (en) * 2018-01-05 2023-04-26 Shandong Danhong Pharmaceutical Co., Ltd. Sglts inhibitor and application thereof
CN110117304A (zh) * 2018-04-23 2019-08-13 中国科学院成都生物研究所 一种钠-葡萄糖协同转运蛋白1和2抑制剂的药物用途
CN110818722B (zh) * 2018-08-14 2022-12-02 苏州鹏旭医药科技有限公司 三种化合物及其制备方法和在合成索格列净中的用途
US20220324897A1 (en) 2019-07-05 2022-10-13 Shandong Danhong Pharmaceutical Co., Ltd. Crystal form of sglt inhibitor and application thereof
CA3145678C (en) * 2019-07-26 2022-08-23 Medshine Discovery Inc. Sglt2/dpp4 inhibitor and application thereof
MX2022001029A (es) 2019-07-26 2022-05-24 Dongbao Purple Star Hangzhou Biopharmaceutical Co Ltd Inhibidor de sglts/dpp4 y aplicación del mismo.
US20230000816A1 (en) * 2019-11-07 2023-01-05 Increvet, Inc. Sodium-glucose linked transporter inhibitors for the management of chronic kidney disease, hypertension, and heart failure in companion animals
US20240100013A1 (en) 2021-01-04 2024-03-28 Lexicon Pharmaceuticals, Inc. Sotagliflozin for improving left atrial function
WO2022155303A1 (en) 2021-01-14 2022-07-21 Lexicon Pharmaceuticals, Inc. Sotagliflozin for treating or preventing cardiovascular diseases
US20250108032A1 (en) 2023-09-28 2025-04-03 Lexicon Pharmaceuticals, Inc. Methods of treating type 1 diabetes and kidney disease
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