JP2013541567A5 - - Google Patents
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- JP2013541567A5 JP2013541567A5 JP2013537044A JP2013537044A JP2013541567A5 JP 2013541567 A5 JP2013541567 A5 JP 2013541567A5 JP 2013537044 A JP2013537044 A JP 2013537044A JP 2013537044 A JP2013537044 A JP 2013537044A JP 2013541567 A5 JP2013541567 A5 JP 2013541567A5
- Authority
- JP
- Japan
- Prior art keywords
- dose
- patient
- fentanyl
- composition
- composition according
- Prior art date
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Applications Claiming Priority (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP10014366.8 | 2010-11-08 | ||
| EP10014366 | 2010-11-08 | ||
| EP10014784 | 2010-11-19 | ||
| EP10014784.2 | 2010-11-19 | ||
| EP10014819 | 2010-11-22 | ||
| EP10014819.6 | 2010-11-22 | ||
| EP10014972.3 | 2010-11-25 | ||
| EP10014972A EP2450039A1 (en) | 2010-11-08 | 2010-11-25 | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
| PCT/EP2011/005581 WO2012062439A1 (en) | 2010-11-08 | 2011-11-07 | Dosing regimen for sedation with cns 7056 (remimazolam) |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013541567A JP2013541567A (ja) | 2013-11-14 |
| JP2013541567A5 true JP2013541567A5 (enExample) | 2014-11-06 |
| JP6084571B2 JP6084571B2 (ja) | 2017-02-22 |
Family
ID=44907114
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013537044A Active JP6084571B2 (ja) | 2010-11-08 | 2011-11-07 | Cns7056(レミマゾラム)を用いた鎮静のための投薬レジメン |
Country Status (17)
| Country | Link |
|---|---|
| US (10) | US9561236B2 (enExample) |
| EP (3) | EP2450039A1 (enExample) |
| JP (1) | JP6084571B2 (enExample) |
| KR (1) | KR102059399B1 (enExample) |
| CN (1) | CN103347519B (enExample) |
| AU (1) | AU2011328497B8 (enExample) |
| DK (1) | DK2637662T3 (enExample) |
| EA (1) | EA024926B1 (enExample) |
| ES (1) | ES2715179T3 (enExample) |
| HR (1) | HRP20190447T1 (enExample) |
| HU (1) | HUE044095T2 (enExample) |
| LT (1) | LT2637662T (enExample) |
| PL (1) | PL2637662T3 (enExample) |
| PT (1) | PT2637662T (enExample) |
| RS (1) | RS58577B1 (enExample) |
| SI (1) | SI2637662T1 (enExample) |
| WO (1) | WO2012062439A1 (enExample) |
Families Citing this family (68)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK2081921T3 (da) | 2006-07-10 | 2011-01-03 | Paion Uk Ltd | Korttidsvirkende benzodiazepinsalte og deres polymorfe former |
| EP2305647A1 (en) | 2009-09-18 | 2011-04-06 | PAION UK Limited | Process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4 H-imidazo[1,2-a][1,4]benzodiazepine-4-yl] propionic acid methyl ester or the benzene sulfonate salt thereof, and compounds useful in that process |
| EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
| WO2014037832A2 (en) | 2012-09-06 | 2014-03-13 | Mahesh Kandula | Compositions and methods for the treatment of epilepsy and neurological diseases |
| WO2013167990A1 (en) | 2012-05-07 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of depression |
| SG11201407300VA (en) | 2012-05-07 | 2014-12-30 | Cellix Bio Private Ltd | Compositions and methods for the treatment of neurological disorders |
| CA2873093A1 (en) | 2012-05-07 | 2013-11-14 | Cellixbio Private Limited | Compositions and methods for treatment of neuromuscular disorders and neurodegenerative disorders |
| US9434704B2 (en) | 2012-05-08 | 2016-09-06 | Cellix Bio Private Limited | Compositions and methods for the treatment of neurological degenerative disorders |
| WO2013168025A1 (en) | 2012-05-08 | 2013-11-14 | Mahesh Kandula | Compositions and methods for treatment of blood clotting disorders |
| WO2013167991A1 (en) | 2012-05-08 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of metabolic disorders |
| US9403826B2 (en) | 2012-05-08 | 2016-08-02 | Cellix Bio Private Limited | Compositions and methods for the treatment of inflammatory disorders |
| US9266823B2 (en) | 2012-05-08 | 2016-02-23 | Cellix Bio Private Limited | Compositions and methods for the treatment of parkinson's disease |
| US9573927B2 (en) | 2012-05-10 | 2017-02-21 | Cellix Bio Private Limited | Compositions and methods for the treatment of severe pain |
| WO2013168001A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of moderate to severe pain |
| WO2013168033A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for treatment of neurologic diseases |
| US9346742B2 (en) | 2012-05-10 | 2016-05-24 | Cellix Bio Private Limited | Compositions and methods for the treatment of fibromyalgia pain |
| US9315478B2 (en) | 2012-05-10 | 2016-04-19 | Cellix Bio Private Limited | Compositions and methods for the treatment of metabolic syndrome |
| WO2013168002A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of neurological conditions |
| SG11201407318UA (en) | 2012-05-10 | 2014-12-30 | Cellix Bio Private Ltd | Compositions and methods for the treatment of metabolic syndrome |
| WO2013168015A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of asthma and allergy |
| US9339484B2 (en) | 2012-05-10 | 2016-05-17 | Cellix Bio Private Limited | Compositions and methods for the treatment of restless leg syndrome and fibromyalgia |
| WO2013168011A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of chronic pain |
| WO2013168014A1 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of familial amyloid polyneuropathy |
| WO2013167999A2 (en) | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for the treatment of neurologic diseases |
| US9242939B2 (en) | 2012-05-10 | 2016-01-26 | Cellix Bio Private Limited | Compositions and methods for the treatment of respiratory disorders |
| WO2013168010A1 (en) * | 2012-05-10 | 2013-11-14 | Mahesh Kandula | Compositions and methods for treatment of severe pain |
| PT2852389T (pt) * | 2012-05-22 | 2017-12-13 | Paion Uk Ltd | Composições que compreendem benzodiazepinas de ação rápida |
| US9227974B2 (en) | 2012-05-23 | 2016-01-05 | Cellex Bio Private Limited | Compositions and methods for the treatment of respiratory disorders |
| US9492409B2 (en) | 2012-05-23 | 2016-11-15 | Cellix Bio Private Limited | Compositions and methods for the treatment of local pain |
| AU2013264896A1 (en) | 2012-05-23 | 2014-11-27 | Cellixbio Private Limited | Compositions and methods for the treatment of multiple sclerosis |
| WO2013175357A2 (en) | 2012-05-23 | 2013-11-28 | Mahesh Kandula | Compositions and methods for the treatment of inflammatory bowel disease |
| US9434729B2 (en) | 2012-05-23 | 2016-09-06 | Cellix Bio Private Limited | Compositions and methods for the treatment of periodontitis and rheumatoid arthritis |
| AU2013264820A1 (en) | 2012-05-23 | 2014-11-27 | Cellixbio Private Limited | Compositions and methods for treatment of mucositis |
| US9108942B1 (en) | 2014-11-05 | 2015-08-18 | Mahesh Kandula | Compositions and methods for the treatment of moderate to severe pain |
| WO2014020480A2 (en) | 2012-08-03 | 2014-02-06 | Mahesh Kandula | Compositions and methods for the treatment migraine and neurologic diseases |
| BR112015004477A8 (pt) | 2012-08-31 | 2019-08-27 | Paion Uk Ltd | uso de composto na preparação de um sedativo e composição farmacêutica |
| US9624168B2 (en) | 2012-09-06 | 2017-04-18 | Cellix Bio Private Limited | Compositions and methods for the treatment inflammation and lipid disorders |
| CA2873029A1 (en) | 2012-09-08 | 2014-03-13 | Cellixbio Private Limited | Compositions and methods for the treatment of inflammation and lipid disorders |
| AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión |
| CN103232454A (zh) * | 2013-05-05 | 2013-08-07 | 王元青 | 治疗精神疾病的药物 |
| US9333187B1 (en) | 2013-05-15 | 2016-05-10 | Cellix Bio Private Limited | Compositions and methods for the treatment of inflammatory bowel disease |
| CA2914461A1 (en) | 2013-06-04 | 2014-12-11 | Cellixbio Private Limited | Compositions and methods for the treatment of diabetes and pre-diabetes |
| US9096537B1 (en) | 2014-12-31 | 2015-08-04 | Mahesh Kandula | Compositions and methods for the treatment of mucositis |
| PL3162804T3 (pl) * | 2014-07-23 | 2020-04-30 | Jiangsu Nhwaluokang Pharmaceutical Research And Development Co., Ltd. | Nowa pochodna benzodiazepiny i jej zastosowanie |
| EP3240779B1 (en) | 2014-09-26 | 2020-10-28 | Cellixbio Private Limited | Compositions and methods for the treatment of epilepsy and neurological disorders |
| CN107207403A (zh) | 2014-09-29 | 2017-09-26 | 塞尔利克斯生物私人有限公司 | 用于治疗多发性硬化的组合物和方法 |
| EP3212626B1 (en) | 2014-10-27 | 2018-11-07 | Cellix Bio Private Limited | Three component salts of fumaric acid monomethyl ester with piperazine or ethylene diamine for the treatment of multiple sclerosis |
| US9173877B1 (en) | 2014-11-05 | 2015-11-03 | Cellix Bio Private Limited | Compositions and methods for the treatment of local pain |
| US9150557B1 (en) | 2014-11-05 | 2015-10-06 | Cellix Bio Private Limited | Compositions and methods for the treatment of hyperglycemia |
| US9175008B1 (en) | 2014-11-05 | 2015-11-03 | Cellix Bio Private Limited | Prodrugs of anti-platelet agents |
| US9290486B1 (en) | 2014-11-05 | 2016-03-22 | Cellix Bio Private Limited | Compositions and methods for the treatment of epilepsy |
| US9284287B1 (en) | 2014-11-05 | 2016-03-15 | Cellix Bio Private Limited | Compositions and methods for the suppression of carbonic anhydrase activity |
| US9321716B1 (en) | 2014-11-05 | 2016-04-26 | Cellix Bio Private Limited | Compositions and methods for the treatment of metabolic syndrome |
| US10208014B2 (en) | 2014-11-05 | 2019-02-19 | Cellix Bio Private Limited | Compositions and methods for the treatment of neurological disorders |
| US9932294B2 (en) | 2014-12-01 | 2018-04-03 | Cellix Bio Private Limited | Compositions and methods for the treatment of multiple sclerosis |
| US9206111B1 (en) | 2014-12-17 | 2015-12-08 | Cellix Bio Private Limited | Compositions and methods for the treatment of neurological diseases |
| CN110845355A (zh) | 2015-01-06 | 2020-02-28 | 塞尔利克斯生物私人有限公司 | 用于治疗炎症和疼痛的组合物和方法 |
| US10925864B2 (en) | 2015-07-18 | 2021-02-23 | Neon Laboratories Limited | Stable liquid injectable solution of midazolam and pentazocine |
| EP3331567B1 (en) | 2015-07-24 | 2020-09-23 | Neon Laboratories Ltd. | Stabilized injectable emulsion of propofol and ketamine |
| WO2017178663A1 (en) * | 2016-04-14 | 2017-10-19 | Paion Uk Limited | Orally inhaled and nasal benzodiazepines |
| CN106407676A (zh) * | 2016-09-12 | 2017-02-15 | 广东省农业科学院动物科学研究所 | 一种基于蒙特卡罗模拟的抗菌药物药效计算方法 |
| CN108143733B (zh) * | 2017-12-15 | 2020-12-25 | 宜昌人福药业有限责任公司 | 一种麻醉镇痛药物组合物及其制备方法 |
| US11708368B2 (en) * | 2018-02-13 | 2023-07-25 | Jiangsu Nhwaluokang Pharmaceutical Research And Development Co., Ltd. | Crystal form of ethyl (S)-3-(8-bromo-1-methyl-6-(pyridin-2-yl)-4H-benzo[f]imidazo[1,2-a][1,4]diazepin-4-yl)propanoate hydrochloride |
| EP3714884A1 (en) * | 2019-03-27 | 2020-09-30 | Paion UK Limited | Medical uses for benzodiazepines with a particular eeg pattern |
| CN112462015B (zh) * | 2020-11-18 | 2022-07-12 | 海南倍特药业有限公司 | 一种氢溴酸瑞马唑仑细菌内毒素的检测方法 |
| CN112402428B (zh) * | 2020-11-26 | 2022-02-25 | 李依泽 | 瑞马唑仑在制备治疗阿片类药物诱发的术后痛觉过敏的药物中的应用 |
| CN114903904B (zh) * | 2021-02-08 | 2024-02-09 | 宜昌人福药业有限责任公司 | 瑞马唑仑药用盐和阿片样物质的注射用药物组合物 |
| CN116270659A (zh) * | 2023-01-13 | 2023-06-23 | 上海市胸科医院 | 瑞马唑仑在制备治疗、减缓或处理骨癌疼痛的产品中的用途 |
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| EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
| CN102964349A (zh) | 2011-08-31 | 2013-03-13 | 江苏恒瑞医药股份有限公司 | 苯并二氮杂*衍生物的托西酸盐及其多晶型、它们的制备方法和用途 |
| JP5585597B2 (ja) | 2012-01-27 | 2014-09-10 | 株式会社デンソー | 車輪位置検出装置およびそれを備えたタイヤ空気圧検出装置 |
| PT2852389T (pt) | 2012-05-22 | 2017-12-13 | Paion Uk Ltd | Composições que compreendem benzodiazepinas de ação rápida |
| BR112015004477A8 (pt) | 2012-08-31 | 2019-08-27 | Paion Uk Ltd | uso de composto na preparação de um sedativo e composição farmacêutica |
| CN107659350A (zh) | 2012-09-28 | 2018-02-02 | 华为技术有限公司 | 信道状态信息进程处理方法、网络设备和用户设备 |
| AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión |
-
2010
- 2010-11-25 EP EP10014972A patent/EP2450039A1/en not_active Withdrawn
-
2011
- 2011-11-07 AU AU2011328497A patent/AU2011328497B8/en active Active
- 2011-11-07 LT LTEP11794020.5T patent/LT2637662T/lt unknown
- 2011-11-07 WO PCT/EP2011/005581 patent/WO2012062439A1/en not_active Ceased
- 2011-11-07 US US13/883,935 patent/US9561236B2/en active Active
- 2011-11-07 ES ES11794020T patent/ES2715179T3/es active Active
- 2011-11-07 HR HRP20190447TT patent/HRP20190447T1/hr unknown
- 2011-11-07 KR KR1020137014559A patent/KR102059399B1/ko active Active
- 2011-11-07 CN CN201180063667.0A patent/CN103347519B/zh not_active Ceased
- 2011-11-07 DK DK11794020.5T patent/DK2637662T3/en active
- 2011-11-07 EP EP19150745.8A patent/EP3492080A1/en not_active Ceased
- 2011-11-07 PT PT11794020T patent/PT2637662T/pt unknown
- 2011-11-07 SI SI201131688T patent/SI2637662T1/sl unknown
- 2011-11-07 JP JP2013537044A patent/JP6084571B2/ja active Active
- 2011-11-07 HU HUE11794020A patent/HUE044095T2/hu unknown
- 2011-11-07 EA EA201390672A patent/EA024926B1/ru unknown
- 2011-11-07 EP EP11794020.5A patent/EP2637662B1/en active Active
- 2011-11-07 PL PL11794020T patent/PL2637662T3/pl unknown
- 2011-11-07 RS RS20190329A patent/RS58577B1/sr unknown
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2017
- 2017-01-06 US US15/400,117 patent/US9737547B2/en active Active
- 2017-07-11 US US15/647,143 patent/US9827251B1/en active Active
- 2017-10-24 US US15/792,636 patent/US10052334B2/en active Active
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2018
- 2018-07-18 US US16/039,198 patent/US10195210B2/en active Active
- 2018-12-07 US US16/213,879 patent/US10342800B2/en active Active
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2019
- 2019-06-28 US US16/457,387 patent/US10722522B2/en active Active
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2020
- 2020-06-18 US US16/905,547 patent/US20200316088A1/en not_active Abandoned
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2023
- 2023-07-10 US US18/219,783 patent/US12201637B2/en active Active
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2024
- 2024-12-20 US US18/989,996 patent/US20250360144A1/en active Pending
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