JP2013540719A - 腎欠陥を有する個体へのロルカセリンの投与 - Google Patents

腎欠陥を有する個体へのロルカセリンの投与 Download PDF

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JP2013540719A
JP2013540719A JP2013527258A JP2013527258A JP2013540719A JP 2013540719 A JP2013540719 A JP 2013540719A JP 2013527258 A JP2013527258 A JP 2013527258A JP 2013527258 A JP2013527258 A JP 2013527258A JP 2013540719 A JP2013540719 A JP 2013540719A
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individual
less
tetrahydro
chloro
benzazepine
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JP2013540719A5 (https=
Inventor
クリステン エム. アンダーソン,
ウィリアム アール. シャナハン,
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アリーナ ファーマシューティカルズ, インコーポレイテッド
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Application filed by アリーナ ファーマシューティカルズ, インコーポレイテッド filed Critical アリーナ ファーマシューティカルズ, インコーポレイテッド
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/70Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing involving creatine or creatinine
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10TTECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
    • Y10T436/00Chemistry: analytical and immunological testing
    • Y10T436/14Heterocyclic carbon compound [i.e., O, S, N, Se, Te, as only ring hetero atom]
    • Y10T436/145555Hetero-N
    • Y10T436/147777Plural nitrogen in the same ring [e.g., barbituates, creatinine, etc.]

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Physics & Mathematics (AREA)
  • General Physics & Mathematics (AREA)
  • Biotechnology (AREA)
  • Food Science & Technology (AREA)
  • Microbiology (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • Cell Biology (AREA)
  • Pathology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
JP2013527258A 2010-09-01 2011-08-31 腎欠陥を有する個体へのロルカセリンの投与 Pending JP2013540719A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US40262810P 2010-09-01 2010-09-01
US61/402,628 2010-09-01
US40314910P 2010-09-10 2010-09-10
US61/403,149 2010-09-10
PCT/US2011/049936 WO2012030939A1 (en) 2010-09-01 2011-08-31 Administration of lorcaserin to individuals with renal impairment

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016050724A Division JP2016106148A (ja) 2010-09-01 2016-03-15 腎欠陥を有する個体へのロルカセリンの投与

Publications (2)

Publication Number Publication Date
JP2013540719A true JP2013540719A (ja) 2013-11-07
JP2013540719A5 JP2013540719A5 (https=) 2014-10-16

Family

ID=44653552

Family Applications (4)

Application Number Title Priority Date Filing Date
JP2013527258A Pending JP2013540719A (ja) 2010-09-01 2011-08-31 腎欠陥を有する個体へのロルカセリンの投与
JP2016050724A Pending JP2016106148A (ja) 2010-09-01 2016-03-15 腎欠陥を有する個体へのロルカセリンの投与
JP2017093900A Withdrawn JP2017132811A (ja) 2010-09-01 2017-05-10 腎欠陥を有する個体へのロルカセリンの投与
JP2018226624A Pending JP2019031577A (ja) 2010-09-01 2018-12-03 腎欠陥を有する個体へのロルカセリンの投与

Family Applications After (3)

Application Number Title Priority Date Filing Date
JP2016050724A Pending JP2016106148A (ja) 2010-09-01 2016-03-15 腎欠陥を有する個体へのロルカセリンの投与
JP2017093900A Withdrawn JP2017132811A (ja) 2010-09-01 2017-05-10 腎欠陥を有する個体へのロルカセリンの投与
JP2018226624A Pending JP2019031577A (ja) 2010-09-01 2018-12-03 腎欠陥を有する個体へのロルカセリンの投与

Country Status (14)

Country Link
US (3) US8999970B2 (https=)
EP (2) EP2939677A1 (https=)
JP (4) JP2013540719A (https=)
KR (2) KR20180094131A (https=)
CN (1) CN103347523A (https=)
AU (3) AU2011296015B2 (https=)
BR (1) BR112013004707A2 (https=)
CA (1) CA2808890A1 (https=)
EA (1) EA201390335A1 (https=)
HK (1) HK1210419A1 (https=)
MX (1) MX2013002418A (https=)
NZ (2) NZ630494A (https=)
SG (2) SG188365A1 (https=)
WO (1) WO2012030939A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2288585A1 (en) * 2008-03-04 2011-03-02 Arena Pharmaceuticals, Inc. Processes for the preparation of intermediates related to the 5-ht2c agonist (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine
US9045431B2 (en) 2010-06-02 2015-06-02 Arena Pharmaceuticals, Inc. Processes for the preparation of 5-HT2C receptor agonists
US20130267500A1 (en) * 2010-09-01 2013-10-10 Arena Pharmaceuticals, Inc. 5-ht2c receptor agonists in the treatment of disorders ameliorated by reduction of norepinephrine level
JP2013536859A (ja) * 2010-09-01 2013-09-26 アリーナ ファーマシューティカルズ, インコーポレイテッド 5−ht2cアゴニストの非吸湿性塩
JP6272695B2 (ja) * 2010-09-01 2018-01-31 エーザイ・アール・アンド・ディー・マネジメント株式会社 体重管理のために有用な5−ht2cアゴニストの改変放出剤形
AU2011296015B2 (en) 2010-09-01 2015-11-12 Arena Pharmaceuticals, Inc. Administration of lorcaserin to individuals with renal impairment
KR20130138770A (ko) 2010-09-01 2013-12-19 아레나 파마슈티칼스, 인크. 광학적으로 활성 산을 갖는 로르카세린의 염
JP2015534563A (ja) 2012-10-09 2015-12-03 アリーナ ファーマシューティカルズ, インコーポレイテッド 体重管理の方法
TW201618787A (zh) 2014-10-30 2016-06-01 艾尼納製藥公司 組合物及方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2008525480A (ja) * 2004-12-23 2008-07-17 アリーナ ファーマシューティカルズ, インコーポレイテッド 5ht2cレセプターモジュレーターの組成物およびその使用方法

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