CN103347523A - 向具有肾损伤的个体给药氯卡色林 - Google Patents
向具有肾损伤的个体给药氯卡色林 Download PDFInfo
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- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10T—TECHNICAL SUBJECTS COVERED BY FORMER US CLASSIFICATION
- Y10T436/00—Chemistry: analytical and immunological testing
- Y10T436/14—Heterocyclic carbon compound [i.e., O, S, N, Se, Te, as only ring hetero atom]
- Y10T436/145555—Hetero-N
- Y10T436/147777—Plural nitrogen in the same ring [e.g., barbituates, creatinine, etc.]
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| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US40262810P | 2010-09-01 | 2010-09-01 | |
| US61/402,628 | 2010-09-01 | ||
| US40314910P | 2010-09-10 | 2010-09-10 | |
| US61/403,149 | 2010-09-10 | ||
| PCT/US2011/049936 WO2012030939A1 (en) | 2010-09-01 | 2011-08-31 | Administration of lorcaserin to individuals with renal impairment |
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| CN2011800528271A Pending CN103347523A (zh) | 2010-09-01 | 2011-08-31 | 向具有肾损伤的个体给药氯卡色林 |
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| US (3) | US8999970B2 (https=) |
| EP (2) | EP2939677A1 (https=) |
| JP (4) | JP2013540719A (https=) |
| KR (2) | KR20180094131A (https=) |
| CN (1) | CN103347523A (https=) |
| AU (3) | AU2011296015B2 (https=) |
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| MX (1) | MX2013002418A (https=) |
| NZ (2) | NZ630494A (https=) |
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| EP2288585A1 (en) * | 2008-03-04 | 2011-03-02 | Arena Pharmaceuticals, Inc. | Processes for the preparation of intermediates related to the 5-ht2c agonist (r)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1h-3-benzazepine |
| US9045431B2 (en) | 2010-06-02 | 2015-06-02 | Arena Pharmaceuticals, Inc. | Processes for the preparation of 5-HT2C receptor agonists |
| US20130267500A1 (en) * | 2010-09-01 | 2013-10-10 | Arena Pharmaceuticals, Inc. | 5-ht2c receptor agonists in the treatment of disorders ameliorated by reduction of norepinephrine level |
| JP2013536859A (ja) * | 2010-09-01 | 2013-09-26 | アリーナ ファーマシューティカルズ, インコーポレイテッド | 5−ht2cアゴニストの非吸湿性塩 |
| JP6272695B2 (ja) * | 2010-09-01 | 2018-01-31 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 体重管理のために有用な5−ht2cアゴニストの改変放出剤形 |
| AU2011296015B2 (en) | 2010-09-01 | 2015-11-12 | Arena Pharmaceuticals, Inc. | Administration of lorcaserin to individuals with renal impairment |
| KR20130138770A (ko) | 2010-09-01 | 2013-12-19 | 아레나 파마슈티칼스, 인크. | 광학적으로 활성 산을 갖는 로르카세린의 염 |
| JP2015534563A (ja) | 2012-10-09 | 2015-12-03 | アリーナ ファーマシューティカルズ, インコーポレイテッド | 体重管理の方法 |
| TW201618787A (zh) | 2014-10-30 | 2016-06-01 | 艾尼納製藥公司 | 組合物及方法 |
Citations (2)
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| CN101123955A (zh) * | 2004-12-23 | 2008-02-13 | 艾尼纳制药公司 | 5HT2c受体调节剂组合物和使用方法 |
| CN101547892A (zh) * | 2006-12-05 | 2009-09-30 | 艾尼纳制药公司 | 制备(r)-8-氯-1-甲基-2,3,4,5-四氢-1h-3-苯并氮杂卓的方法和其中间体 |
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- 2011-08-31 CN CN2011800528271A patent/CN103347523A/zh active Pending
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- 2011-08-31 JP JP2013527258A patent/JP2013540719A/ja active Pending
- 2011-08-31 KR KR1020187023062A patent/KR20180094131A/ko not_active Ceased
- 2011-08-31 BR BR112013004707A patent/BR112013004707A2/pt not_active Application Discontinuation
- 2011-08-31 SG SG2013015631A patent/SG188365A1/en unknown
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- 2011-08-31 KR KR1020137008393A patent/KR20140091458A/ko not_active Ceased
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- 2011-08-31 SG SG10201506896RA patent/SG10201506896RA/en unknown
- 2011-08-31 EA EA201390335A patent/EA201390335A1/ru unknown
- 2011-08-31 CA CA2808890A patent/CA2808890A1/en not_active Abandoned
- 2011-08-31 EP EP15169002.1A patent/EP2939677A1/en not_active Withdrawn
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2015
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2016
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|---|---|
| BR112013004707A2 (pt) | 2016-05-10 |
| NZ630494A (en) | 2016-05-27 |
| JP2013540719A (ja) | 2013-11-07 |
| AU2016200860A1 (en) | 2016-02-25 |
| US20120252787A1 (en) | 2012-10-04 |
| AU2016200860B2 (en) | 2017-10-12 |
| US8999970B2 (en) | 2015-04-07 |
| HK1210419A1 (en) | 2016-04-22 |
| AU2018200108A1 (en) | 2018-01-25 |
| US9770455B2 (en) | 2017-09-26 |
| NZ608266A (en) | 2015-09-25 |
| CA2808890A1 (en) | 2012-03-08 |
| SG188365A1 (en) | 2013-04-30 |
| JP2017132811A (ja) | 2017-08-03 |
| WO2012030939A1 (en) | 2012-03-08 |
| KR20180094131A (ko) | 2018-08-22 |
| EP2939677A1 (en) | 2015-11-04 |
| MX2013002418A (es) | 2013-08-01 |
| US20170216307A1 (en) | 2017-08-03 |
| AU2011296015A1 (en) | 2013-04-04 |
| JP2016106148A (ja) | 2016-06-16 |
| US20150196567A1 (en) | 2015-07-16 |
| KR20140091458A (ko) | 2014-07-21 |
| SG10201506896RA (en) | 2015-10-29 |
| EA201390335A1 (ru) | 2013-09-30 |
| JP2019031577A (ja) | 2019-02-28 |
| EP2611449A1 (en) | 2013-07-10 |
| AU2011296015B2 (en) | 2015-11-12 |
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