JP2013537901A5 - - Google Patents
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- Publication number
- JP2013537901A5 JP2013537901A5 JP2013529758A JP2013529758A JP2013537901A5 JP 2013537901 A5 JP2013537901 A5 JP 2013537901A5 JP 2013529758 A JP2013529758 A JP 2013529758A JP 2013529758 A JP2013529758 A JP 2013529758A JP 2013537901 A5 JP2013537901 A5 JP 2013537901A5
- Authority
- JP
- Japan
- Prior art keywords
- aprepitant
- proline
- neuropsychiatric
- pruritus
- cancers
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38574410P | 2010-09-23 | 2010-09-23 | |
| US61/385,744 | 2010-09-23 | ||
| US201161439654P | 2011-02-04 | 2011-02-04 | |
| US61/439,654 | 2011-02-04 | ||
| US201161498214P | 2011-06-17 | 2011-06-17 | |
| US61/498,214 | 2011-06-17 | ||
| PCT/IB2011/054210 WO2012038937A1 (en) | 2010-09-23 | 2011-09-23 | Aprepitant l-proline composition and cocrystal |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2013537901A JP2013537901A (ja) | 2013-10-07 |
| JP2013537901A5 true JP2013537901A5 (enExample) | 2016-02-12 |
| JP5997162B2 JP5997162B2 (ja) | 2016-09-28 |
Family
ID=44907915
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013529758A Active JP5997162B2 (ja) | 2010-09-23 | 2011-09-23 | アプレピタントｌ−プロリン組成物および共結晶 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9029369B2 (enExample) |
| EP (1) | EP2618828B1 (enExample) |
| JP (1) | JP5997162B2 (enExample) |
| KR (1) | KR101833578B1 (enExample) |
| CN (1) | CN103221049B (enExample) |
| AR (1) | AR083095A1 (enExample) |
| AU (1) | AU2011306391B2 (enExample) |
| BR (1) | BR112013006651A2 (enExample) |
| CA (1) | CA2846460C (enExample) |
| ES (1) | ES2616752T3 (enExample) |
| IL (1) | IL225443A0 (enExample) |
| TW (1) | TWI540131B (enExample) |
| WO (1) | WO2012038937A1 (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103221049B (zh) | 2010-09-23 | 2015-11-25 | 诺弗米克斯有限公司 | 阿瑞匹坦l-脯氨酸组合物和共晶 |
| WO2013076659A1 (en) | 2011-11-25 | 2013-05-30 | Nuformix Limited | Aprepitant l-proline solvates - compositions and cocrystals |
| US10098859B2 (en) | 2012-09-05 | 2018-10-16 | Amri Ssci, Llc | Cocrystals of p-coumaric acid |
| US20160324881A1 (en) * | 2013-12-30 | 2016-11-10 | Oncoprevent Gmbh | Neurokinin-1 Receptor Antagonists For Use In A Method Of Prevention Of Cancer |
| SG11202007530XA (en) * | 2018-02-07 | 2020-09-29 | Reata Pharmaceuticals Inc | Co-crystal forms of a novobiocin analog and proline |
| CN116283947A (zh) * | 2023-02-07 | 2023-06-23 | 成都医学院 | 一种阿瑞匹坦共晶及其制备方法和用途 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5145684A (en) | 1991-01-25 | 1992-09-08 | Sterling Drug Inc. | Surface modified drug nanoparticles |
| US6048859A (en) | 1992-06-29 | 2000-04-11 | Merck & Co., Inc. | Morpholine and thiomorpholine tachykinin receptor antagonists |
| US5719147A (en) | 1992-06-29 | 1998-02-17 | Merck & Co., Inc. | Morpholine and thiomorpholine tachykinin receptor antagonists |
| IL111960A (en) | 1993-12-17 | 1999-12-22 | Merck & Co Inc | Morpholines and thiomorpholines their preparation and pharmaceutical compositions containing them |
| ZA985765B (en) | 1997-07-02 | 1999-08-04 | Merck & Co Inc | Polymorphic form of a tachykinin receptor antagonist. |
| CA2489984A1 (en) * | 2002-06-21 | 2003-12-31 | Transform Pharmaceuticals, Inc. | Pharmaceutical compositions with improved dissolution |
| JP4923182B2 (ja) * | 2003-02-28 | 2012-04-25 | マクニール−ピーピーシー・インコーポレーテツド | セレコキシブ及びニコチンアミド共結晶並びにこの共結晶を含む医薬組成物 |
| EP2034952A4 (en) * | 2006-06-16 | 2011-08-17 | Reddys Lab Ltd Dr | APREPITANT COMPOSITIONS |
| US20110009362A1 (en) * | 2008-02-27 | 2011-01-13 | Dr. Reddy's Laboratories Ltd. | Solubility-enhanced forms of aprepitant and pharmaceutical compositions thereof |
| CN103221049B (zh) | 2010-09-23 | 2015-11-25 | 诺弗米克斯有限公司 | 阿瑞匹坦l-脯氨酸组合物和共晶 |
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2011
- 2011-09-23 CN CN201180055997.5A patent/CN103221049B/zh active Active
- 2011-09-23 JP JP2013529758A patent/JP5997162B2/ja active Active
- 2011-09-23 KR KR1020137010228A patent/KR101833578B1/ko active Active
- 2011-09-23 US US13/825,380 patent/US9029369B2/en active Active
- 2011-09-23 ES ES11779217.6T patent/ES2616752T3/es active Active
- 2011-09-23 CA CA2846460A patent/CA2846460C/en active Active
- 2011-09-23 AR ARP110103486 patent/AR083095A1/es unknown
- 2011-09-23 AU AU2011306391A patent/AU2011306391B2/en active Active
- 2011-09-23 WO PCT/IB2011/054210 patent/WO2012038937A1/en not_active Ceased
- 2011-09-23 BR BR112013006651A patent/BR112013006651A2/pt not_active Application Discontinuation
- 2011-09-23 EP EP11779217.6A patent/EP2618828B1/en active Active
- 2011-09-23 TW TW100134362A patent/TWI540131B/zh active
-
2013
- 2013-03-21 IL IL225443A patent/IL225443A0/en active IP Right Grant