JP2013518107A5 - - Google Patents
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- Publication number
- JP2013518107A5 JP2013518107A5 JP2012551213A JP2012551213A JP2013518107A5 JP 2013518107 A5 JP2013518107 A5 JP 2013518107A5 JP 2012551213 A JP2012551213 A JP 2012551213A JP 2012551213 A JP2012551213 A JP 2012551213A JP 2013518107 A5 JP2013518107 A5 JP 2013518107A5
- Authority
- JP
- Japan
- Prior art keywords
- acceptable salt
- pharmaceutically acceptable
- combination
- abacavir
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000003839 salts Chemical class 0.000 claims 10
- 229960004748 abacavir Drugs 0.000 claims 4
- MCGSCOLBFJQGHM-SCZZXKLOSA-N abacavir Chemical compound C=12N=CN([C@H]3C=C[C@@H](CO)C3)C2=NC(N)=NC=1NC1CC1 MCGSCOLBFJQGHM-SCZZXKLOSA-N 0.000 claims 4
- 150000001875 compounds Chemical class 0.000 claims 4
- 239000008194 pharmaceutical composition Substances 0.000 claims 4
- 229960001627 lamivudine Drugs 0.000 claims 2
- JTEGQNOMFQHVDC-NKWVEPMBSA-N lamivudine Chemical compound O=C1N=C(N)C=CN1[C@H]1O[C@@H](CO)SC1 JTEGQNOMFQHVDC-NKWVEPMBSA-N 0.000 claims 2
- 159000000000 sodium salts Chemical class 0.000 claims 2
- XPOQHMRABVBWPR-UHFFFAOYSA-N Efavirenz Natural products O1C(=O)NC2=CC=C(Cl)C=C2C1(C(F)(F)F)C#CC1CC1 XPOQHMRABVBWPR-UHFFFAOYSA-N 0.000 claims 1
- 208000031886 HIV Infections Diseases 0.000 claims 1
- 208000037357 HIV infectious disease Diseases 0.000 claims 1
- XPOQHMRABVBWPR-ZDUSSCGKSA-N efavirenz Chemical compound C([C@]1(C2=CC(Cl)=CC=C2NC(=O)O1)C(F)(F)F)#CC1CC1 XPOQHMRABVBWPR-ZDUSSCGKSA-N 0.000 claims 1
- 229960003804 efavirenz Drugs 0.000 claims 1
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 claims 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US29858910P | 2010-01-27 | 2010-01-27 | |
| US61/298,589 | 2010-01-27 | ||
| PCT/US2011/022219 WO2011094150A1 (en) | 2010-01-27 | 2011-01-24 | Antiviral therapy |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016015242A Division JP2016145204A (ja) | 2010-01-27 | 2016-01-29 | 抗ウイルス療法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2013518107A JP2013518107A (ja) | 2013-05-20 |
| JP2013518107A5 true JP2013518107A5 (https=) | 2014-03-13 |
Family
ID=44319704
Family Applications (9)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012551213A Pending JP2013518107A (ja) | 2010-01-27 | 2011-01-24 | 抗ウイルス療法 |
| JP2016015242A Pending JP2016145204A (ja) | 2010-01-27 | 2016-01-29 | 抗ウイルス療法 |
| JP2016161610A Active JP6268386B2 (ja) | 2010-01-27 | 2016-08-22 | 抗ウイルス療法 |
| JP2018072861A Pending JP2018127473A (ja) | 2010-01-27 | 2018-04-05 | 抗ウイルス療法 |
| JP2019106635A Pending JP2019167371A (ja) | 2010-01-27 | 2019-06-07 | 抗ウイルス療法 |
| JP2021030306A Active JP7724619B2 (ja) | 2010-01-27 | 2021-02-26 | 抗ウイルス療法 |
| JP2022032464A Pending JP2022071126A (ja) | 2010-01-27 | 2022-03-03 | 抗ウイルス療法 |
| JP2023060638A Pending JP2023085431A (ja) | 2010-01-27 | 2023-04-04 | 抗ウイルス療法 |
| JP2025091741A Pending JP2025131664A (ja) | 2010-01-27 | 2025-06-02 | 抗ウイルス療法 |
Family Applications After (8)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2016015242A Pending JP2016145204A (ja) | 2010-01-27 | 2016-01-29 | 抗ウイルス療法 |
| JP2016161610A Active JP6268386B2 (ja) | 2010-01-27 | 2016-08-22 | 抗ウイルス療法 |
| JP2018072861A Pending JP2018127473A (ja) | 2010-01-27 | 2018-04-05 | 抗ウイルス療法 |
| JP2019106635A Pending JP2019167371A (ja) | 2010-01-27 | 2019-06-07 | 抗ウイルス療法 |
| JP2021030306A Active JP7724619B2 (ja) | 2010-01-27 | 2021-02-26 | 抗ウイルス療法 |
| JP2022032464A Pending JP2022071126A (ja) | 2010-01-27 | 2022-03-03 | 抗ウイルス療法 |
| JP2023060638A Pending JP2023085431A (ja) | 2010-01-27 | 2023-04-04 | 抗ウイルス療法 |
| JP2025091741A Pending JP2025131664A (ja) | 2010-01-27 | 2025-06-02 | 抗ウイルス療法 |
Country Status (45)
Families Citing this family (32)
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| TWI677489B (zh) | 2014-06-20 | 2019-11-21 | 美商基利科學股份有限公司 | 多環型胺甲醯基吡啶酮化合物之合成 |
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| TWI695003B (zh) | 2014-12-23 | 2020-06-01 | 美商基利科學股份有限公司 | 多環胺甲醯基吡啶酮化合物及其醫藥用途 |
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| FI3694522T3 (fi) * | 2017-10-13 | 2026-02-05 | Viiv Healthcare Co | Kaksikerroksinen lääketablettiformulaatio |
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2011
- 2011-01-24 PE PE2012001082A patent/PE20121524A1/es active IP Right Grant
- 2011-01-24 CA CA2967453A patent/CA2967453C/en active Active
- 2011-01-24 ME MEP-2015-106A patent/ME02182B/me unknown
- 2011-01-24 PT PT117374843T patent/PT2531027E/pt unknown
- 2011-01-24 UA UAA201209253A patent/UA105556C2/uk unknown
- 2011-01-24 FI FIEP19151897.6T patent/FI3494972T3/fi active
- 2011-01-24 BR BR112012018670-1A patent/BR112012018670A2/pt not_active Application Discontinuation
- 2011-01-24 SG SG10201509476RA patent/SG10201509476RA/en unknown
- 2011-01-24 HU HUE19151897A patent/HUE065569T2/hu unknown
- 2011-01-24 CA CA3060290A patent/CA3060290C/en active Active
- 2011-01-24 SI SI201131593T patent/SI3127542T1/sl unknown
- 2011-01-24 CA CA2787691A patent/CA2787691C/en active Active
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