JP2010540438A - 免疫障害を処置するためのｓ１ｐ受容体調節剤としての１−（４−ベンジルベンズアミド）−ベンジル）アゼチジン−３−カルボン酸誘導体および関連化合物 - Google Patents
免疫障害を処置するためのｓ１ｐ受容体調節剤としての１−（４−ベンジルベンズアミド）−ベンジル）アゼチジン−３−カルボン酸誘導体および関連化合物 Download PDFInfo
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- JP2010540438A JP2010540438A JP2010525834A JP2010525834A JP2010540438A JP 2010540438 A JP2010540438 A JP 2010540438A JP 2010525834 A JP2010525834 A JP 2010525834A JP 2010525834 A JP2010525834 A JP 2010525834A JP 2010540438 A JP2010540438 A JP 2010540438A
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Landscapes
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| JP2010540438A true JP2010540438A (ja) | 2010-12-24 |
| JP2010540438A5 JP2010540438A5 (enExample) | 2011-10-20 |
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| JP (1) | JP2010540438A (enExample) |
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| AU (1) | AU2008302746B2 (enExample) |
| CA (1) | CA2699417A1 (enExample) |
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| ES (1) | ES2360929T3 (enExample) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015129859A1 (ja) * | 2014-02-28 | 2015-09-03 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
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| US7919519B2 (en) | 2005-11-23 | 2011-04-05 | Epix Pharmaceuticals Inc. | S1P receptor modulating compounds and use thereof |
| CA2630714C (en) | 2005-11-23 | 2014-01-14 | Epix Delaware, Inc. | S1p receptor modulating compounds and use thereof |
| US7790707B2 (en) | 2006-03-21 | 2010-09-07 | Epix Pharmaceuticals Inc. | S1P receptor modulating compounds and use thereof |
| US20090069288A1 (en) * | 2007-07-16 | 2009-03-12 | Breinlinger Eric C | Novel therapeutic compounds |
| US8080542B2 (en) | 2007-09-20 | 2011-12-20 | Amgen, Inc. | S1P receptor modulating compounds and use thereof |
| TW201000099A (en) * | 2008-06-20 | 2010-01-01 | Amgen Inc | S1P1 receptor agonists and use thereof |
| US8791100B2 (en) * | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
| EP2643303A1 (en) | 2010-11-24 | 2013-10-02 | Allergan, Inc. | Modulators of s1p receptors |
| FR3017867A1 (fr) * | 2014-02-21 | 2015-08-28 | Inventiva | Nouveaux composes de type phenylazetidine carboxylate ou carboxamide |
| US9895324B2 (en) | 2014-03-26 | 2018-02-20 | University Of Kentucky Research Foundation | Halogenated diarylacetylenes and methods of treating cancer |
| WO2017070089A1 (en) | 2015-10-19 | 2017-04-27 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| ES2928856T3 (es) | 2015-11-19 | 2022-11-23 | Incyte Corp | Compuestos heterocíclicos como inmunomoduladores |
| WO2017106634A1 (en) | 2015-12-17 | 2017-06-22 | Incyte Corporation | N-phenyl-pyridine-2-carboxamide derivatives and their use as pd-1/pd-l1 protein/protein interaction modulators |
| TWI850624B (zh) | 2015-12-22 | 2024-08-01 | 美商英塞特公司 | 作為免疫調節劑之雜環化合物 |
| ES2906460T3 (es) | 2016-05-06 | 2022-04-18 | Incyte Corp | Compuestos heterocíclicos como inmunomoduladores |
| TW201808902A (zh) | 2016-05-26 | 2018-03-16 | 美商英塞特公司 | 作為免疫調節劑之雜環化合物 |
| PT3472167T (pt) | 2016-06-20 | 2022-11-11 | Incyte Corp | Compostos heterocíclicos como imunomoduladores |
| US20180016260A1 (en) | 2016-07-14 | 2018-01-18 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| MA46045A (fr) | 2016-08-29 | 2021-04-28 | Incyte Corp | Composés hétérocycliques utilisés comme immunomodulateurs |
| EP3558973B1 (en) | 2016-12-22 | 2021-09-15 | Incyte Corporation | Pyridine derivatives as immunomodulators |
| RS63710B1 (sr) | 2016-12-22 | 2022-11-30 | Incyte Corp | Derivati tetrahidro imidazo[4,5-c] piridina kao induktori internalizacije pd-l1 |
| JP7101678B2 (ja) | 2016-12-22 | 2022-07-15 | インサイト・コーポレイション | 免疫調節剤としての複素環式化合物 |
| US20180179201A1 (en) | 2016-12-22 | 2018-06-28 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| TW201835049A (zh) | 2016-12-22 | 2018-10-01 | 美商英塞特公司 | 作為免疫調節劑之雜環化合物 |
| RS66699B1 (sr) | 2018-03-30 | 2025-05-30 | Incyte Corp | Heterociklična jedinjenja kao imunomodulatori |
| TW202425987A (zh) | 2018-05-11 | 2024-07-01 | 美商英塞特公司 | 作為免疫調節劑之雜環化合物 |
| TW202115059A (zh) | 2019-08-09 | 2021-04-16 | 美商英塞特公司 | Ｐｄ—１／ｐｄ—ｌ１抑制劑之鹽 |
| JP7559059B2 (ja) | 2019-09-30 | 2024-10-01 | インサイト・コーポレイション | 免疫調節剤としてのピリド［３，２－ｄ］ピリミジン化合物 |
| PH12022551136A1 (en) | 2019-11-11 | 2023-10-09 | Incyte Corp | Salts and crystalline forms of a pd-1/pd-l1 inhibitor |
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Cited By (4)
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| WO2015129859A1 (ja) * | 2014-02-28 | 2015-09-03 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
| JPWO2015129859A1 (ja) * | 2014-02-28 | 2017-03-30 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
| US9718771B2 (en) | 2014-02-28 | 2017-08-01 | Kissei Pharmaceutical Co., Ltd. | Aniline derivative, pharmaceutical composition containing same, and use thereof |
| US9988350B2 (en) | 2014-02-28 | 2018-06-05 | Kissei Pharmaceutical Co., Ltd. | Aniline derivative, pharmaceutical composition containing same, and use thereof |
Also Published As
| Publication number | Publication date |
|---|---|
| MX2010002885A (es) | 2010-04-01 |
| AU2008302746A1 (en) | 2009-03-26 |
| US8080542B2 (en) | 2011-12-20 |
| EP2188252B1 (en) | 2011-04-13 |
| AU2008302746B2 (en) | 2014-07-03 |
| EP2188252A2 (en) | 2010-05-26 |
| DE602008006209D1 (de) | 2011-05-26 |
| ATE505454T1 (de) | 2011-04-15 |
| US20120088749A1 (en) | 2012-04-12 |
| US20090082331A1 (en) | 2009-03-26 |
| CA2699417A1 (en) | 2009-03-26 |
| WO2009038759A3 (en) | 2009-07-23 |
| ES2360929T3 (es) | 2011-06-10 |
| WO2009038759A2 (en) | 2009-03-26 |
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