JP2010540438A - 免疫障害を処置するためのｓ１ｐ受容体調節剤としての１−（４−ベンジルベンズアミド）−ベンジル）アゼチジン−３−カルボン酸誘導体および関連化合物 - Google Patents
免疫障害を処置するためのｓ１ｐ受容体調節剤としての１−（４−ベンジルベンズアミド）−ベンジル）アゼチジン−３−カルボン酸誘導体および関連化合物 Download PDFInfo
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- JP2010540438A JP2010540438A JP2010525834A JP2010525834A JP2010540438A JP 2010540438 A JP2010540438 A JP 2010540438A JP 2010525834 A JP2010525834 A JP 2010525834A JP 2010525834 A JP2010525834 A JP 2010525834A JP 2010540438 A JP2010540438 A JP 2010540438A
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Landscapes
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| US99481207P | 2007-09-20 | 2007-09-20 | |
| PCT/US2008/010887 WO2009038759A2 (en) | 2007-09-20 | 2008-09-19 | 1-(4-(benzylbenzamid0) -benzyl) azetidine-3-carboxylic acid derivatives and related compounds as slp receptor modulators for the treatment of immune disorders |
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| JP2010540438A true JP2010540438A (ja) | 2010-12-24 |
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| EP (1) | EP2188252B1 (enExample) |
| JP (1) | JP2010540438A (enExample) |
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| AU (1) | AU2008302746B2 (enExample) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015129859A1 (ja) * | 2014-02-28 | 2015-09-03 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
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| CA2630714C (en) | 2005-11-23 | 2014-01-14 | Epix Delaware, Inc. | S1p receptor modulating compounds and use thereof |
| US7919519B2 (en) | 2005-11-23 | 2011-04-05 | Epix Pharmaceuticals Inc. | S1P receptor modulating compounds and use thereof |
| WO2007109330A2 (en) | 2006-03-21 | 2007-09-27 | Epix Delaware, Inc. | S1p receptor modulating compounds |
| WO2009011850A2 (en) * | 2007-07-16 | 2009-01-22 | Abbott Laboratories | Novel therapeutic compounds |
| ATE505454T1 (de) | 2007-09-20 | 2011-04-15 | Amgen Inc | 1-(4-(4-benzylbenzamid)-benzyl)-azetidin-3- carboxylsäurederivate und entsprechende verbindungen als s1p-rezeptor-modulatoren zur behandlung von immunerkrankungen |
| TW201000099A (en) * | 2008-06-20 | 2010-01-01 | Amgen Inc | S1P1 receptor agonists and use thereof |
| US8791100B2 (en) * | 2010-02-02 | 2014-07-29 | Novartis Ag | Aryl benzylamine compounds |
| BR112013012836A2 (pt) | 2010-11-24 | 2019-09-24 | Allergan Inc | moduladores dos receptores s1p" |
| FR3017867A1 (fr) * | 2014-02-21 | 2015-08-28 | Inventiva | Nouveaux composes de type phenylazetidine carboxylate ou carboxamide |
| US9895324B2 (en) | 2014-03-26 | 2018-02-20 | University Of Kentucky Research Foundation | Halogenated diarylacetylenes and methods of treating cancer |
| US20170107216A1 (en) | 2015-10-19 | 2017-04-20 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| MD3377488T2 (ro) | 2015-11-19 | 2023-02-28 | Incyte Corp | Compuși heterociclici ca imunomodulatori |
| ES2916874T3 (es) | 2015-12-17 | 2022-07-06 | Incyte Corp | Derivados de N-fenil-piridina-2-carboxamida y su uso como moduladores de la interacción proteína/proteína PD-1/PD-L1 |
| CA3009474A1 (en) | 2015-12-22 | 2017-06-29 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| ES2906460T3 (es) | 2016-05-06 | 2022-04-18 | Incyte Corp | Compuestos heterocíclicos como inmunomoduladores |
| EP3464279B1 (en) | 2016-05-26 | 2021-11-24 | Incyte Corporation | Heterocyclic compounds as immunomodulators |
| SG11201811414TA (en) | 2016-06-20 | 2019-01-30 | Incyte Corp | Heterocyclic compounds as immunomodulators |
| MA45669A (fr) | 2016-07-14 | 2019-05-22 | Incyte Corp | Composés hétérocycliques utilisés comme immunomodulateurs |
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| WO2018119236A1 (en) | 2016-12-22 | 2018-06-28 | Incyte Corporation | Triazolo[1,5-a]pyridine derivatives as immunomodulators |
| SMT202300065T1 (it) | 2018-03-30 | 2023-05-12 | Incyte Corp | Composti eterociclici come immunomodulatori |
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Cited By (4)
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| WO2015129859A1 (ja) * | 2014-02-28 | 2015-09-03 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
| JPWO2015129859A1 (ja) * | 2014-02-28 | 2017-03-30 | キッセイ薬品工業株式会社 | 新規なアニリン誘導体、それを含有する医薬組成物およびそれらの用途 |
| US9718771B2 (en) | 2014-02-28 | 2017-08-01 | Kissei Pharmaceutical Co., Ltd. | Aniline derivative, pharmaceutical composition containing same, and use thereof |
| US9988350B2 (en) | 2014-02-28 | 2018-06-05 | Kissei Pharmaceutical Co., Ltd. | Aniline derivative, pharmaceutical composition containing same, and use thereof |
Also Published As
| Publication number | Publication date |
|---|---|
| US20090082331A1 (en) | 2009-03-26 |
| AU2008302746A1 (en) | 2009-03-26 |
| MX2010002885A (es) | 2010-04-01 |
| AU2008302746B2 (en) | 2014-07-03 |
| CA2699417A1 (en) | 2009-03-26 |
| ATE505454T1 (de) | 2011-04-15 |
| EP2188252A2 (en) | 2010-05-26 |
| US8080542B2 (en) | 2011-12-20 |
| DE602008006209D1 (de) | 2011-05-26 |
| US20120088749A1 (en) | 2012-04-12 |
| ES2360929T3 (es) | 2011-06-10 |
| WO2009038759A3 (en) | 2009-07-23 |
| WO2009038759A2 (en) | 2009-03-26 |
| EP2188252B1 (en) | 2011-04-13 |
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