JP2010533714A - ピコプラチンのための経口製剤 - Google Patents
ピコプラチンのための経口製剤 Download PDFInfo
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- JP2010533714A JP2010533714A JP2010517010A JP2010517010A JP2010533714A JP 2010533714 A JP2010533714 A JP 2010533714A JP 2010517010 A JP2010517010 A JP 2010517010A JP 2010517010 A JP2010517010 A JP 2010517010A JP 2010533714 A JP2010533714 A JP 2010533714A
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- Prior art keywords
- picoplatin
- cancer
- formulation
- oil
- combination
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 229950005566 picoplatin Drugs 0.000 title claims abstract description 368
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- 206010028980 Neoplasm Diseases 0.000 claims description 49
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- IIZPXYDJLKNOIY-JXPKJXOSSA-N 1-palmitoyl-2-arachidonoyl-sn-glycero-3-phosphocholine Chemical compound CCCCCCCCCCCCCCCC(=O)OC[C@H](COP([O-])(=O)OCC[N+](C)(C)C)OC(=O)CCC\C=C/C\C=C/C\C=C/C\C=C/CCCCC IIZPXYDJLKNOIY-JXPKJXOSSA-N 0.000 claims description 43
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| WO2018211847A1 (ja) * | 2017-05-18 | 2018-11-22 | キユーピー株式会社 | 自己乳化性を有する組成物、及びその製造方法、並びにナノエマルション、及びその製造方法 |
| JP2019500344A (ja) * | 2015-12-08 | 2019-01-10 | 広州藍亮医薬科技有限公司Ｂｌｕｅｌｉｇｈｔ Ｐｈａｒｍａｔｅｃｈ Ｃｏ．，Ｌｔｄ． | デコキネート固体分散体、その調製方法及び使用 |
| JP2024531060A (ja) * | 2022-07-06 | 2024-08-29 | アバンサール センディリアン ベルハッド | 親油性化合物の改善された経口バイオアベイラビリティを有する自己乳化薬物送達配合物 |
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| US8168662B1 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8178564B2 (en) | 2006-11-06 | 2012-05-15 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8168661B2 (en) | 2006-11-06 | 2012-05-01 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| US8173686B2 (en) * | 2006-11-06 | 2012-05-08 | Poniard Pharmaceuticals, Inc. | Use of picoplatin to treat colorectal cancer |
| WO2008097658A1 (en) * | 2007-02-09 | 2008-08-14 | Poniard Pharmaceuticals, Inc. | Encapsulated picoplatin |
| TW200916094A (en) * | 2007-06-27 | 2009-04-16 | Poniard Pharmaceuticals Inc | Stabilized picoplatin dosage form |
| AU2009210654A1 (en) * | 2008-02-08 | 2009-08-13 | Poniard Pharmaceuticals, Inc. | Use of picoplatin and bevacizumab to treat colorectal cancer |
| US20120148661A1 (en) * | 2009-04-15 | 2012-06-14 | Poniard Pharmaceuticals, Inc. | High bioavailability oral picoplatin anti-cancer therapy |
| MX348668B (es) * | 2009-09-21 | 2017-06-23 | J W Pharmaceutical Corp * | Nanopartículas de oxaliplatin y método para prepararlas. |
| AU2011260615B2 (en) * | 2010-06-02 | 2016-11-17 | Pharma& Schweiz Gmbh | Oral dosage forms of bendamustine |
| CN101926757B (zh) | 2010-09-01 | 2013-01-02 | 北京大学 | 一种难溶性药物的液体组合物及其制备方法 |
| EP2773323A4 (en) | 2011-10-31 | 2015-04-22 | Merck Sharp & Dohme | NANO-SUSPENSION METHOD |
| CN104427977B (zh) | 2012-05-10 | 2018-02-02 | 佩因拉佛姆有限公司 | 局部麻醉剂的储库制剂及其制备方法 |
| KR101612257B1 (ko) * | 2015-07-30 | 2016-04-20 | 대화제약 주식회사 | 고농도의 탁산을 포함하는 경구 투여용 약학 조성물 |
| WO2017018635A1 (ko) * | 2015-07-30 | 2017-02-02 | 대화제약 주식회사 | 고농도의 탁산을 포함하는 경구 투여용 약학 조성물 |
| KR101612260B1 (ko) | 2015-07-30 | 2016-04-20 | 대화제약 주식회사 | 고농도의 탁산을 포함하는 경구 투여용 약학 조성물 |
| GB2541387A (en) * | 2015-08-14 | 2017-02-22 | Res Center Pharmaceutical Eng Gmbh | Self-emulsifying Nanosuspensions as Drug Delivery Systems (SENDDS) |
| CN108066771A (zh) * | 2017-12-15 | 2018-05-25 | 北京思如诺科技有限公司 | 一种具有高载药量环境响应型抗肿瘤纳米药物、载体以及制备方法 |
| PL247245B1 (pl) * | 2019-01-31 | 2025-06-02 | Gdanski Univ Medyczny | Samoemulgująca kompozycja farmaceutyczna w postaci ciekłej zawierająca jako substancję aktywną substancję leczniczą nietrwałą w środowisku wodnym |
| CN119699569B (zh) * | 2024-12-23 | 2025-10-17 | 晨光生物科技集团股份有限公司 | 一种叶黄素酯油悬液及其制备方法与应用 |
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-
2008
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- 2008-07-16 CN CN200880103323A patent/CN101809024A/zh active Pending
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|---|---|---|---|---|
| JP2019500344A (ja) * | 2015-12-08 | 2019-01-10 | 広州藍亮医薬科技有限公司Ｂｌｕｅｌｉｇｈｔ Ｐｈａｒｍａｔｅｃｈ Ｃｏ．，Ｌｔｄ． | デコキネート固体分散体、その調製方法及び使用 |
| WO2018211847A1 (ja) * | 2017-05-18 | 2018-11-22 | キユーピー株式会社 | 自己乳化性を有する組成物、及びその製造方法、並びにナノエマルション、及びその製造方法 |
| JPWO2018211847A1 (ja) * | 2017-05-18 | 2020-02-27 | キユーピー株式会社 | 自己乳化性を有する組成物、及びその製造方法、並びにナノエマルション、及びその製造方法 |
| US11571385B2 (en) | 2017-05-18 | 2023-02-07 | Kewpie Corporation | Self-emulsifiable composition, production method therefor, nanoemulsion, and production method therefor |
| JP2024531060A (ja) * | 2022-07-06 | 2024-08-29 | アバンサール センディリアン ベルハッド | 親油性化合物の改善された経口バイオアベイラビリティを有する自己乳化薬物送達配合物 |
| JP7752233B2 (ja) | 2022-07-06 | 2025-10-09 | アバンサール センディリアン ベルハッド | 親油性化合物の改善された経口バイオアベイラビリティを有する自己乳化薬物送達配合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20100310661A1 (en) | 2010-12-09 |
| TW200920347A (en) | 2009-05-16 |
| WO2009011861A1 (en) | 2009-01-22 |
| EP2178893A4 (en) | 2012-09-19 |
| CA2693057A1 (en) | 2009-01-22 |
| EP2178893A1 (en) | 2010-04-28 |
| CN101809024A (zh) | 2010-08-18 |
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