JP2010528009A5 - - Google Patents

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JP2010528009A5
JP2010528009A5 JP2010509367A JP2010509367A JP2010528009A5 JP 2010528009 A5 JP2010528009 A5 JP 2010528009A5 JP 2010509367 A JP2010509367 A JP 2010509367A JP 2010509367 A JP2010509367 A JP 2010509367A JP 2010528009 A5 JP2010528009 A5 JP 2010528009A5
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Japan
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substituted
aryl
heteroaryl
heterocyclic
alkyl
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JP2010509367A
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Japanese (ja)
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JP5378362B2 (ja
JP2010528009A (ja
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Priority claimed from PCT/US2008/006475 external-priority patent/WO2008144062A1/en
Publication of JP2010528009A publication Critical patent/JP2010528009A/ja
Publication of JP2010528009A5 publication Critical patent/JP2010528009A5/ja
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Publication of JP5378362B2 publication Critical patent/JP5378362B2/ja
Expired - Fee Related legal-status Critical Current
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JP2010509367A 2007-05-21 2008-05-20 Ｃｓｆ−１ｒ阻害剤、組成物および使用方法 Expired - Fee Related JP5378362B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US93930307P 2007-05-21 2007-05-21
US60/939,303 2007-05-21
PCT/US2008/006475 WO2008144062A1 (en) 2007-05-21 2008-05-20 Csf-1r inhibitors, compositions, and methods of use

Publications (3)

Publication Number Publication Date
JP2010528009A JP2010528009A (ja) 2010-08-19
JP2010528009A5 true JP2010528009A5 (enExample) 2011-07-07
JP5378362B2 JP5378362B2 (ja) 2013-12-25

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JP2010509367A Expired - Fee Related JP5378362B2 (ja) 2007-05-21 2008-05-20 Ｃｓｆ−１ｒ阻害剤、組成物および使用方法

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Country Link
US (1) US8293769B2 (enExample)
EP (1) EP2152700B1 (enExample)
JP (1) JP5378362B2 (enExample)
KR (1) KR20100017866A (enExample)
CN (1) CN101754965B (enExample)
AU (1) AU2008254425A1 (enExample)
BR (1) BRPI0812159A2 (enExample)
CA (1) CA2685967A1 (enExample)
EA (1) EA200901548A1 (enExample)
ES (1) ES2452349T3 (enExample)
MX (1) MX2009012679A (enExample)
WO (1) WO2008144062A1 (enExample)

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EP3876930A4 (en) 2018-11-07 2022-07-20 Dana-Farber Cancer Institute, Inc. BENZIMIDAZOLE DERIVATIVES AND AZA-BENZIMIDAZOLE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF
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KR102913995B1 (ko) * 2019-04-12 2026-01-16 내셔날 헬스 리서치 인스티튜트 치료 용도를 위한 키나제 억제제로서의 헤테로사이클릭 화합물
US20220401461A1 (en) * 2019-10-24 2022-12-22 Kyoto University Pharmaceutical Composition for Protecting Cartilage
BR112022022409A2 (pt) 2020-05-06 2023-02-07 Ajax Therapeutics Inc 6-heteroarilóxi benzimidazóis e azabenzimidazóis como inibidores de jak2
CN119454695A (zh) * 2020-09-23 2025-02-18 上海润石医药科技有限公司 Csf1r激酶抑制剂及其用途
WO2022140527A1 (en) 2020-12-23 2022-06-30 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
WO2023009712A1 (en) * 2021-07-29 2023-02-02 Ajax Therapeutics, Inc. Heteroaryloxy thiazolo azines as jak2 inhibitors
CA3234638A1 (en) 2021-11-09 2023-05-19 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
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