JP2010523599A5 - - Google Patents

Download PDF

Info

Publication number
JP2010523599A5
JP2010523599A5 JP2010502352A JP2010502352A JP2010523599A5 JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5 JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5
Authority
JP
Japan
Prior art keywords
alkyl
aryl
group
heteroaryl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010502352A
Other languages
English (en)
Japanese (ja)
Other versions
JP2010523599A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2008/059599 external-priority patent/WO2008124703A2/en
Publication of JP2010523599A publication Critical patent/JP2010523599A/ja
Publication of JP2010523599A5 publication Critical patent/JP2010523599A5/ja
Pending legal-status Critical Current

Links

JP2010502352A 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発 Pending JP2010523599A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92206507P 2007-04-05 2007-04-05
PCT/US2008/059599 WO2008124703A2 (en) 2007-04-05 2008-04-07 Development of molecular imaging probes for carbonic anhydrase-ix using click chemistry

Publications (2)

Publication Number Publication Date
JP2010523599A JP2010523599A (ja) 2010-07-15
JP2010523599A5 true JP2010523599A5 (enExample) 2010-12-02

Family

ID=39743771

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010502352A Pending JP2010523599A (ja) 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発

Country Status (7)

Country Link
US (2) US7829063B2 (enExample)
EP (2) EP2129666A2 (enExample)
JP (1) JP2010523599A (enExample)
KR (2) KR20120003499A (enExample)
CN (1) CN101679318A (enExample)
CA (1) CA2683434A1 (enExample)
WO (1) WO2008124703A2 (enExample)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2010004880A (es) * 2007-10-29 2010-07-28 Schering Corp Derivados heterociclicos de urea y tiourea, y metodos de uso de los mismos.
RU2498798C2 (ru) * 2008-01-09 2013-11-20 Моликьюлар Инсайт Фармасьютикалз, Инк. Ингибиторы карбоангидразы iх
EP2706057B1 (en) 2008-12-05 2016-04-20 Molecular Insight Pharmaceuticals, Inc. Bis(imidazolyl)compounds and radionuclide complexes
EA026557B1 (ru) 2008-12-09 2017-04-28 Джилид Сайэнс, Инк. Промежуточные соединения для получения модуляторов толл-подобных рецепторов
BR112012000209B8 (pt) 2009-06-15 2021-07-27 Molecular Insight Pharm Inc heterodímeros de ácido glutâmico e seus processos de preparação
WO2011018798A2 (en) * 2009-08-14 2011-02-17 Indian Association For The Cultivation Of Science Morpholino-based antisense agent
EP2491014A1 (en) * 2009-10-21 2012-08-29 Bayer Pharma Aktiengesellschaft Substituted halophenoxybenzamide derivatives
JP6245981B2 (ja) * 2010-04-08 2017-12-13 シーメンス メディカル ソリューションズ ユーエスエー インコーポレイテッドＳｉｅｍｅｎｓ Ｍｅｄｉｃａｌ Ｓｏｌｕｔｉｏｎｓ ＵＳＡ，Ｉｎｃ． 含水有機溶媒中の１８ｆ−標識化トレーサーの合成
US10639608B2 (en) 2010-04-08 2020-05-05 Siemens Medical Solutions Usa, Inc. System, device and method for preparing tracers and transferring materials during radiosynthesis
DK2634177T3 (en) * 2010-10-29 2016-08-15 Clino Ltd TAU IMAGE SOUND
CA2817691C (en) * 2010-11-13 2020-09-01 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
US9180209B2 (en) * 2011-02-28 2015-11-10 The Board Of Trustees Of The Leland Stanford Junior University Non-peptidic quenched fluorescent imaging probes
CN102219753B (zh) * 2011-04-21 2012-10-31 山东大学 一种三氮唑类化合物及其制备方法与应用
WO2012154885A2 (en) 2011-05-09 2012-11-15 Visen Medical, Inc. Carbonic anhydrase targeting agents and methods of using same
JP2014156400A (ja) * 2011-05-24 2014-08-28 Astellas Pharma Inc 腫瘍の画像診断用標識誘導体
US9120837B2 (en) 2012-01-06 2015-09-01 Molecular Insight Pharmaceuticals Metal complexes of poly(carboxyl)amine-containing ligands having an affinity for carbonic anhydrase IX
WO2013148319A1 (en) 2012-03-30 2013-10-03 Visen Medical, Inc. Bacterial imaging agents and methods of using same
WO2014110372A1 (en) 2013-01-14 2014-07-17 Molecular Insight Pharmaceuticals Triazine based radiopharmaceuticals and radioimaging agents
CA2929401A1 (en) 2013-11-05 2015-05-14 Bayer Cropscience Aktiengesellschaft Novel compounds for combating arthropods
PT3166607T (pt) 2014-07-11 2022-12-07 Gilead Sciences Inc Moduladores de receptores de tipo toll para o tratamento do vih
CN104212440B (zh) * 2014-09-03 2016-03-30 无锡艾德美特生物科技有限公司 一类喹唑啉类荧光探针及其制备和应用
CN107074860B (zh) * 2014-09-16 2022-07-15 吉利德科学公司 制备toll样受体调节剂的方法
AU2015318061B2 (en) 2014-09-16 2018-05-17 Gilead Sciences, Inc. Solid forms of a toll-like receptor modulator
CN107428776B (zh) 2015-03-24 2020-10-23 H.隆德贝克有限公司 制造4,5,6,7-四氢异噁唑并[5,4-c]吡啶-3-醇
LT6401B (lt) 2015-07-28 2017-06-12 Vilniaus Universitetas Karboanhidrazės selektyvūs inhibitoriai
CN105541825A (zh) * 2015-12-28 2016-05-04 中国药科大学 三氮唑衍生物制备方法及其作为药物的用途
KR102531494B1 (ko) * 2016-05-13 2023-05-10 더 존스 홉킨스 유니버시티 탄산 탈수효소 ix를 표적으로 하는 핵 영상화 및 방사선치료 제제 및 이의 용도
US10695450B2 (en) 2016-07-26 2020-06-30 Laboratoires Cyclopharma Synthesis of a radioactive agent composition
AU2018255413A1 (en) * 2017-04-20 2019-12-05 Leidos Biomedical Research, Inc. K-Ras modulators
DK3668856T3 (da) 2017-08-17 2021-09-20 Glaxosmithkline Ip Dev Ltd Hidtil ukendte tetrazolforbindelser og anvendelse deraf til behandling af tuberkulose
KR102147971B1 (ko) * 2019-11-22 2020-08-25 국방과학연구소 반응용매에 대한 혼화성 차이를 이용한 화학선택적 트리아졸의 제조방법
WO2025113696A1 (zh) * 2023-11-30 2025-06-05 赣州和美药业股份有限公司 一种化合物及其应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6562319B2 (en) * 2001-03-12 2003-05-13 Yissum Research Development Company Of The Hebrew University Of Jerusalem Radiolabeled irreversible inhibitors of epidermal growth factor receptor tyrosine kinase and their use in radioimaging and radiotherapy
HUE028349T2 (en) * 2002-11-26 2016-12-28 Inst Virology CAIX-specific inhibitors
US20060269942A1 (en) * 2005-04-27 2006-11-30 Kolb Hartmuth C In situ click chemistry method for screening high affinity molecular imaging probes
EP1733742A1 (en) 2005-06-17 2006-12-20 Universiteit Utrecht Holding B.V. Dendrimers multivalently substituted with active groups
US8158590B2 (en) 2005-08-05 2012-04-17 Syntarga B.V. Triazole-containing releasable linkers, conjugates thereof, and methods of preparation
US8470587B2 (en) * 2006-08-28 2013-06-25 The Trustees Of The University Of Pennsylvania 129Xe biosensors and their use
WO2008033557A2 (en) 2006-09-15 2008-03-20 Siemens Medical Solutions Usa, Inc. Click chemistry-derived cyclic peptidomimetics as integrin markers

Similar Documents

Publication Publication Date Title
JP2010523599A5 (enExample)
WO2009155017A3 (en) Novel substituted azabenzoxazoles
JP2016534063A5 (enExample)
JP2013544846A5 (enExample)
JP2010511632A5 (enExample)
JP2015508103A5 (enExample)
DK2864329T3 (en) 18F-LABELED PHOLATE / ANTIFOLATE ANALOGS
JP2013523896A5 (enExample)
JP2017531619A5 (enExample)
JP2015518004A5 (enExample)
JP2017528498A5 (enExample)
JP2008195730A5 (enExample)
WO2015191506A3 (en) Pyrrolo[2,3-c]pyridines as imaging agents for neurofibrilary tangles
JP2013540114A5 (enExample)
JP2015511609A5 (enExample)
JP5500875B2 (ja) 新規化合物、該新規化合物を用いたプローブ及び該新規化合物もしくは該プローブを用いた蛍光イメージング用造影剤
JP2012506439A5 (enExample)
JP2010513441A5 (enExample)
RU2012124266A (ru) Хелаты марганца и их применение в качестве контрастных агентов в магнитно-резонансной визуализации (mpb)
JP2010505865A5 (enExample)
JP2007511494A5 (enExample)
JP2012504131A5 (enExample)
JP2012522841A5 (enExample)
JP2019527225A (ja) Ｉｄｏ１酵素イメージングのための放射性リガンド
JP2010502585A5 (enExample)