JP2010523599A5 - - Google Patents

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Publication number
JP2010523599A5
JP2010523599A5 JP2010502352A JP2010502352A JP2010523599A5 JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5 JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5
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JP
Japan
Prior art keywords
alkyl
aryl
group
heteroaryl
compound
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010502352A
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English (en)
Japanese (ja)
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JP2010523599A (ja
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Publication date
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Priority claimed from PCT/US2008/059599 external-priority patent/WO2008124703A2/en
Publication of JP2010523599A publication Critical patent/JP2010523599A/ja
Publication of JP2010523599A5 publication Critical patent/JP2010523599A5/ja
Pending legal-status Critical Current

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JP2010502352A 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発 Pending JP2010523599A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92206507P 2007-04-05 2007-04-05
PCT/US2008/059599 WO2008124703A2 (en) 2007-04-05 2008-04-07 Development of molecular imaging probes for carbonic anhydrase-ix using click chemistry

Publications (2)

Publication Number Publication Date
JP2010523599A JP2010523599A (ja) 2010-07-15
JP2010523599A5 true JP2010523599A5 (enExample) 2010-12-02

Family

ID=39743771

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010502352A Pending JP2010523599A (ja) 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発

Country Status (7)

Country Link
US (2) US7829063B2 (enExample)
EP (2) EP2468734A1 (enExample)
JP (1) JP2010523599A (enExample)
KR (2) KR20120003499A (enExample)
CN (1) CN101679318A (enExample)
CA (1) CA2683434A1 (enExample)
WO (1) WO2008124703A2 (enExample)

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EP2209779A1 (en) * 2007-10-29 2010-07-28 Schering Corporation Heterocyclic urea and thiourea derivatives and methods of use thereof
US8562945B2 (en) 2008-01-09 2013-10-22 Molecular Insight Pharmaceuticals, Inc. Technetium- and rhenium-bis(heteroaryl) complexes and methods of use thereof
RU2498798C2 (ru) 2008-01-09 2013-11-20 Моликьюлар Инсайт Фармасьютикалз, Инк. Ингибиторы карбоангидразы iх
RS53347B (sr) 2008-12-09 2014-10-31 Gilead Sciences, Inc. Modulatori toll-sličnih receptora
AU2010260195B2 (en) 2009-06-15 2014-11-20 Molecular Insight Pharmaceuticals, Inc. Process for production of heterodimers of glutamic acid
US9914745B2 (en) 2009-08-14 2018-03-13 Indian Association For The Cultivation Of Science Morpholino-based antisense agent
EP2491014A1 (en) * 2009-10-21 2012-08-29 Bayer Pharma Aktiengesellschaft Substituted halophenoxybenzamide derivatives
CA2795762C (en) * 2010-04-08 2017-03-28 Siemens Medical Solutions Usa, Inc. Synthesis of 18f-labeled tracers in hydrous organic solvents
US10639608B2 (en) 2010-04-08 2020-05-05 Siemens Medical Solutions Usa, Inc. System, device and method for preparing tracers and transferring materials during radiosynthesis
RU2627694C2 (ru) 2010-10-29 2017-08-10 Клино Лтд. Производные хинолина, визуализирующий белок тау
KR101848077B1 (ko) * 2010-11-13 2018-04-11 이노크린 파마슈티컬즈, 인크. 금속효소 억제제 화합물
WO2012118715A2 (en) * 2011-02-28 2012-09-07 The Board Of Trustees Of Leland Stanford Junior University Non-peptidic quenched fluorescent imaging probes
CN102219753B (zh) * 2011-04-21 2012-10-31 山东大学 一种三氮唑类化合物及其制备方法与应用
CN103687854A (zh) 2011-05-09 2014-03-26 文森医学公司 碳酸酐酶靶向剂及其使用方法
JP2014156400A (ja) * 2011-05-24 2014-08-28 Astellas Pharma Inc 腫瘍の画像診断用標識誘導体
EP2800471A4 (en) 2012-01-06 2015-11-04 Molecular Insight Pharm Inc METAL COMPLEX OF POLY (CARBOXYL) AMINE CONTAINING LIGANDS HAVING AFFINITY FOR CARBON IX ANHYDRASE
US9375493B2 (en) 2012-03-30 2016-06-28 Visen Medical, Inc. Bacterial imaging agents and methods of using same
EP3939972A1 (en) 2013-01-14 2022-01-19 Molecular Insight Pharmaceuticals, Inc. Triazine based radiopharmaceuticals and radioimaging agents
AR098311A1 (es) 2013-11-05 2016-05-26 Bayer Cropscience Ag Compuestos para el control de artrópodos
JP6522732B2 (ja) 2014-07-11 2019-05-29 ギリアード サイエンシーズ， インコーポレイテッド Ｈｉｖを治療するためのトール様受容体の調節因子
CN104212440B (zh) * 2014-09-03 2016-03-30 无锡艾德美特生物科技有限公司 一类喹唑啉类荧光探针及其制备和应用
SG11201701520TA (en) 2014-09-16 2017-04-27 Gilead Sciences Inc Solid forms of a toll-like receptor modulator
KR102306860B1 (ko) * 2014-09-16 2021-09-30 길리애드 사이언시즈, 인코포레이티드 톨-유사 수용체 조정제를 제조하는 방법
LT3274331T (lt) 2015-03-24 2020-04-10 H. Lundbeck A/S 4,5,6,7-tetrahidroizozaksolo[5,4-c]piridin-3-olio gamybos būdas
LT6401B (lt) 2015-07-28 2017-06-12 Vilniaus Universitetas Karboanhidrazės selektyvūs inhibitoriai
CN105541825A (zh) * 2015-12-28 2016-05-04 中国药科大学 三氮唑衍生物制备方法及其作为药物的用途
KR102531494B1 (ko) * 2016-05-13 2023-05-10 더 존스 홉킨스 유니버시티 탄산 탈수효소 ix를 표적으로 하는 핵 영상화 및 방사선치료 제제 및 이의 용도
US10695450B2 (en) 2016-07-26 2020-06-30 Laboratoires Cyclopharma Synthesis of a radioactive agent composition
EP3612526A2 (en) * 2017-04-20 2020-02-26 The Regents of the University of California K-ras modulators
WO2019034729A1 (en) * 2017-08-17 2019-02-21 Glaxosmithkline Intellectual Property Development Limited NOVEL TETRAZOLE COMPOUNDS AND THEIR USE IN THE TREATMENT OF TUBERCULOSIS
TWI810456B (zh) 2019-05-22 2023-08-01 美商基利科學股份有限公司 Tlr7調節化合物及hiv疫苗之組合
KR102147971B1 (ko) * 2019-11-22 2020-08-25 국방과학연구소 반응용매에 대한 혼화성 차이를 이용한 화학선택적 트리아졸의 제조방법
WO2025113696A1 (zh) * 2023-11-30 2025-06-05 赣州和美药业股份有限公司 一种化合物及其应用
CN117986213A (zh) * 2024-02-26 2024-05-07 厦门大学 一种5-氯甲基糠醛制备2,5-二（氨基甲基）呋喃的方法
WO2026060272A1 (en) * 2024-09-16 2026-03-19 Wisconsin Alumni Research Foundation Long-residence ca9 ligands and radioisotope carriers for inhibition, visualization and irradiation of ca9-expressing tumors

Family Cites Families (7)

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Publication number Priority date Publication date Assignee Title
US6562319B2 (en) * 2001-03-12 2003-05-13 Yissum Research Development Company Of The Hebrew University Of Jerusalem Radiolabeled irreversible inhibitors of epidermal growth factor receptor tyrosine kinase and their use in radioimaging and radiotherapy
US7550424B2 (en) * 2002-11-26 2009-06-23 Institute Of Virology Slovak Academy Of Sciences CA IX-specific inhibitors
ATE527542T1 (de) * 2005-04-27 2011-10-15 Siemens Medical Solutions Verfahren zur herstellung von abbildungssonden unter verwendung von click chemie
EP1733742A1 (en) 2005-06-17 2006-12-20 Universiteit Utrecht Holding B.V. Dendrimers multivalently substituted with active groups
US8158590B2 (en) 2005-08-05 2012-04-17 Syntarga B.V. Triazole-containing releasable linkers, conjugates thereof, and methods of preparation
WO2008027162A2 (en) * 2006-08-28 2008-03-06 The Trustees Of The University Of Pennsylvania 129xe biosensors and their use
US20080213175A1 (en) 2006-09-15 2008-09-04 Kolb Hartmuth C Click chemistry-derived cyclic peptidomimetics as integrin markers

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