JP2010523599A5 - - Google Patents

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Publication number
JP2010523599A5
JP2010523599A5 JP2010502352A JP2010502352A JP2010523599A5 JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5 JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010502352 A JP2010502352 A JP 2010502352A JP 2010523599 A5 JP2010523599 A5 JP 2010523599A5
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JP
Japan
Prior art keywords
alkyl
aryl
group
heteroaryl
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2010502352A
Other languages
English (en)
Japanese (ja)
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JP2010523599A (ja
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Publication date
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Priority claimed from PCT/US2008/059599 external-priority patent/WO2008124703A2/en
Publication of JP2010523599A publication Critical patent/JP2010523599A/ja
Publication of JP2010523599A5 publication Critical patent/JP2010523599A5/ja
Pending legal-status Critical Current

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JP2010502352A 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発 Pending JP2010523599A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92206507P 2007-04-05 2007-04-05
PCT/US2008/059599 WO2008124703A2 (en) 2007-04-05 2008-04-07 Development of molecular imaging probes for carbonic anhydrase-ix using click chemistry

Publications (2)

Publication Number Publication Date
JP2010523599A JP2010523599A (ja) 2010-07-15
JP2010523599A5 true JP2010523599A5 (enExample) 2010-12-02

Family

ID=39743771

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2010502352A Pending JP2010523599A (ja) 2007-04-05 2008-04-07 クリックケミストリーを使用した炭酸脱水酵素−ｉｘのための分子イメージングプローブの開発

Country Status (7)

Country Link
US (2) US7829063B2 (enExample)
EP (2) EP2468734A1 (enExample)
JP (1) JP2010523599A (enExample)
KR (2) KR20090127433A (enExample)
CN (1) CN101679318A (enExample)
CA (1) CA2683434A1 (enExample)
WO (1) WO2008124703A2 (enExample)

Families Citing this family (32)

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Publication number Priority date Publication date Assignee Title
CA2703981A1 (en) * 2007-10-29 2009-05-07 Schering Corporation Heterocyclic urea and thiourea derivatives and methods of use thereof
US8562945B2 (en) 2008-01-09 2013-10-22 Molecular Insight Pharmaceuticals, Inc. Technetium- and rhenium-bis(heteroaryl) complexes and methods of use thereof
AU2009204133B2 (en) 2008-01-09 2014-04-10 Molecular Insight Pharmaceuticals, Inc. Inhibitors of carbonic anhydrase IX
MX2011006152A (es) 2008-12-09 2011-07-28 Gilead Sciences Inc Moduladores de receptores tipo toll.
BR112012000210A2 (pt) 2009-06-15 2019-09-24 Molecular Insight Pharm Inc processo para a produção de heterodímeoros de ácido glutâmico.
WO2011018798A2 (en) * 2009-08-14 2011-02-17 Indian Association For The Cultivation Of Science Morpholino-based antisense agent
WO2011047796A1 (en) * 2009-10-21 2011-04-28 Bayer Schering Pharma Aktiengesellschaft Substituted halophenoxybenzamide derivatives
US10639608B2 (en) 2010-04-08 2020-05-05 Siemens Medical Solutions Usa, Inc. System, device and method for preparing tracers and transferring materials during radiosynthesis
KR101430422B1 (ko) * 2010-04-08 2014-08-14 지멘스 메디컬 솔루션즈 유에스에이, 인크. 함수 유기 용매에서 18ｆ-표지된 트레이서의 합성
HUE030172T2 (en) 2010-10-29 2017-05-29 Clino Ltd Tau imaging probe
CA2817691C (en) * 2010-11-13 2020-09-01 Viamet Pharmaceuticals, Inc. Metalloenzyme inhibitor compounds
US9180209B2 (en) * 2011-02-28 2015-11-10 The Board Of Trustees Of The Leland Stanford Junior University Non-peptidic quenched fluorescent imaging probes
CN102219753B (zh) * 2011-04-21 2012-10-31 山东大学 一种三氮唑类化合物及其制备方法与应用
WO2012154885A2 (en) 2011-05-09 2012-11-15 Visen Medical, Inc. Carbonic anhydrase targeting agents and methods of using same
JP2014156400A (ja) * 2011-05-24 2014-08-28 Astellas Pharma Inc 腫瘍の画像診断用標識誘導体
WO2013103813A1 (en) 2012-01-06 2013-07-11 Molecular Insight Pharmaceuticals Metal complexes of poly(carboxyl)amine-containing ligands having an affinity for carbonic anhydrase ix
CN104245954A (zh) 2012-03-30 2014-12-24 文森医学公司 细菌成像剂及其使用方法
HUE035739T2 (en) 2013-01-14 2018-05-28 Molecular Insight Pharm Inc Triazine-based radiopharmaceuticals and radiological imaging agents
BR112016010164A2 (pt) 2013-11-05 2017-08-08 Bayer Cropscience Ag novos compostos para o combate aos ártropodes
JP6522732B2 (ja) 2014-07-11 2019-05-29 ギリアード サイエンシーズ， インコーポレイテッド Ｈｉｖを治療するためのトール様受容体の調節因子
CN104212440B (zh) * 2014-09-03 2016-03-30 无锡艾德美特生物科技有限公司 一类喹唑啉类荧光探针及其制备和应用
EP3194401B1 (en) 2014-09-16 2020-10-21 Gilead Sciences, Inc. Solid forms of a toll-like receptor modulator
CN107074860B (zh) * 2014-09-16 2022-07-15 吉利德科学公司 制备toll样受体调节剂的方法
MA41802B1 (fr) 2015-03-24 2020-04-30 H Lundbeck As Fabrication de 4,5,6,7-tétrahydroisozaxolo[5,4-c]pyridine-3-ol
LT6401B (lt) 2015-07-28 2017-06-12 Vilniaus Universitetas Karboanhidrazės selektyvūs inhibitoriai
CN105541825A (zh) * 2015-12-28 2016-05-04 中国药科大学 三氮唑衍生物制备方法及其作为药物的用途
CN109476655B (zh) * 2016-05-13 2022-03-08 约翰霍普金斯大学 靶向碳酸酐酶ix的核成像剂和放射治疗剂及其用途
US10695450B2 (en) 2016-07-26 2020-06-30 Laboratoires Cyclopharma Synthesis of a radioactive agent composition
KR20200011426A (ko) * 2017-04-20 2020-02-03 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 K-ras 조절인자
SMT202100515T1 (it) * 2017-08-17 2021-11-12 Glaxosmithkline Ip Dev Ltd Nuovi composti tetrazolici e loro uso nel trattamento della tubercolosi
KR102147971B1 (ko) * 2019-11-22 2020-08-25 국방과학연구소 반응용매에 대한 혼화성 차이를 이용한 화학선택적 트리아졸의 제조방법
WO2025113696A1 (zh) * 2023-11-30 2025-06-05 赣州和美药业股份有限公司 一种化合物及其应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6562319B2 (en) * 2001-03-12 2003-05-13 Yissum Research Development Company Of The Hebrew University Of Jerusalem Radiolabeled irreversible inhibitors of epidermal growth factor receptor tyrosine kinase and their use in radioimaging and radiotherapy
EP2594265B1 (en) * 2002-11-26 2015-10-28 Institute Of Virology Ca ix-specific inhibitors
US20060269942A1 (en) * 2005-04-27 2006-11-30 Kolb Hartmuth C In situ click chemistry method for screening high affinity molecular imaging probes
EP1733742A1 (en) 2005-06-17 2006-12-20 Universiteit Utrecht Holding B.V. Dendrimers multivalently substituted with active groups
US8158590B2 (en) 2005-08-05 2012-04-17 Syntarga B.V. Triazole-containing releasable linkers, conjugates thereof, and methods of preparation
WO2008027162A2 (en) * 2006-08-28 2008-03-06 The Trustees Of The University Of Pennsylvania 129xe biosensors and their use
US20080213175A1 (en) 2006-09-15 2008-09-04 Kolb Hartmuth C Click chemistry-derived cyclic peptidomimetics as integrin markers

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