JP2010506853A - 疼痛などのナトリウムチャネル媒介性の疾患の処置のための、スピロ（［３，２−フロ］ピリジン−３，３’−インドール）−２’（１’ｈ）−オン誘導体および関連化合物 - Google Patents
疼痛などのナトリウムチャネル媒介性の疾患の処置のための、スピロ（［３，２−フロ］ピリジン−３，３’−インドール）−２’（１’ｈ）−オン誘導体および関連化合物 Download PDFInfo
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- JP2010506853A JP2010506853A JP2009532605A JP2009532605A JP2010506853A JP 2010506853 A JP2010506853 A JP 2010506853A JP 2009532605 A JP2009532605 A JP 2009532605A JP 2009532605 A JP2009532605 A JP 2009532605A JP 2010506853 A JP2010506853 A JP 2010506853A
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US85123706P | 2006-10-12 | 2006-10-12 | |
| US95558207P | 2007-08-13 | 2007-08-13 | |
| PCT/US2007/081244 WO2008046049A1 (en) | 2006-10-12 | 2007-10-12 | Spiro (furo [3, 2-c] pyridine-3-3 ' -indol) -2' (1'h)-one derivatives and related compounds for the treatment of sodium-channel mediated diseases, such as pain |
Publications (2)
| Publication Number | Publication Date |
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| JP2010506853A true JP2010506853A (ja) | 2010-03-04 |
| JP2010506853A5 JP2010506853A5 (https=) | 2011-11-24 |
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| JP2009532605A Withdrawn JP2010506853A (ja) | 2006-10-12 | 2007-10-12 | 疼痛などのナトリウムチャネル媒介性の疾患の処置のための、スピロ（［３，２−フロ］ピリジン−３，３’−インドール）−２’（１’ｈ）−オン誘導体および関連化合物 |
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| Country | Link |
|---|---|
| US (1) | US20110294842A9 (https=) |
| EP (1) | EP2076514A1 (https=) |
| JP (1) | JP2010506853A (https=) |
| AR (1) | AR063278A1 (https=) |
| AU (1) | AU2007307638A1 (https=) |
| BR (1) | BRPI0719857A2 (https=) |
| CA (1) | CA2666143A1 (https=) |
| CL (1) | CL2007002953A1 (https=) |
| MX (1) | MX2009003875A (https=) |
| RU (1) | RU2009117605A (https=) |
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012505895A (ja) * | 2008-10-17 | 2012-03-08 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | 治療剤としてのスピロオキシインドール化合物およびそれらの使用 |
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| AR053710A1 (es) * | 2005-04-11 | 2007-05-16 | Xenon Pharmaceuticals Inc | Compuestos espiroheterociclicos y sus usos como agentes terapeuticos |
| AR056968A1 (es) | 2005-04-11 | 2007-11-07 | Xenon Pharmaceuticals Inc | Compuestos espiro-oxindol y composiciones farmacéuticas |
| WO2008060789A2 (en) | 2006-10-12 | 2008-05-22 | Xenon Pharmaceuticals Inc. | Use of spiro-oxindole compounds as therapeutic agents |
| CA2741024A1 (en) * | 2008-10-17 | 2010-04-22 | Xenon Pharmaceuticals Inc. | Spiro-oxindole compounds and their use as therapeutic agents |
| WO2010078307A1 (en) | 2008-12-29 | 2010-07-08 | Xenon Pharmaceuticals Inc. | Spiro-oxindole-derivatives as sodium channel blockers |
| AR077252A1 (es) | 2009-06-29 | 2011-08-10 | Xenon Pharmaceuticals Inc | Enantiomeros de compuestos de espirooxindol y sus usos como agentes terapeuticos |
| US20110086899A1 (en) * | 2009-10-14 | 2011-04-14 | Xenon Pharmaceuticals Inc. | Pharmaceutical compositions for oral administration |
| KR20120099429A (ko) | 2009-10-14 | 2012-09-10 | 제논 파마슈티칼스 인크. | 스피로-옥스인돌 화합물의 합성 방법 |
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| HK1205114A1 (en) | 2012-04-12 | 2015-12-11 | Xenon Pharmaceuticals Inc. | Asymmetric syntheses for spiro-oxindole compounds useful as therapeutic agents |
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| TW201722938A (zh) | 2015-09-04 | 2017-07-01 | 魯賓有限公司 | 作為電位閘控鈉通道調節子之磺醯胺化合物 |
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2007
- 2007-10-12 US US12/445,270 patent/US20110294842A9/en not_active Abandoned
- 2007-10-12 WO PCT/US2007/081244 patent/WO2008046049A1/en not_active Ceased
- 2007-10-12 MX MX2009003875A patent/MX2009003875A/es not_active Application Discontinuation
- 2007-10-12 TW TW096138359A patent/TW200825091A/zh unknown
- 2007-10-12 BR BRPI0719857-4A patent/BRPI0719857A2/pt not_active IP Right Cessation
- 2007-10-12 JP JP2009532605A patent/JP2010506853A/ja not_active Withdrawn
- 2007-10-12 EP EP07844225A patent/EP2076514A1/en not_active Withdrawn
- 2007-10-12 AR ARP070104539A patent/AR063278A1/es unknown
- 2007-10-12 CA CA002666143A patent/CA2666143A1/en not_active Abandoned
- 2007-10-12 RU RU2009117605/04A patent/RU2009117605A/ru not_active Application Discontinuation
- 2007-10-12 AU AU2007307638A patent/AU2007307638A1/en not_active Abandoned
- 2007-10-12 CL CL200702953A patent/CL2007002953A1/es unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012505895A (ja) * | 2008-10-17 | 2012-03-08 | ゼノン・ファーマシューティカルズ・インコーポレイテッド | 治療剤としてのスピロオキシインドール化合物およびそれらの使用 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2076514A1 (en) | 2009-07-08 |
| RU2009117605A (ru) | 2010-11-20 |
| US20100160362A1 (en) | 2010-06-24 |
| TW200825091A (en) | 2008-06-16 |
| CL2007002953A1 (es) | 2008-02-01 |
| BRPI0719857A2 (pt) | 2014-06-03 |
| MX2009003875A (es) | 2009-04-22 |
| US20110294842A9 (en) | 2011-12-01 |
| CA2666143A1 (en) | 2008-04-17 |
| AU2007307638A1 (en) | 2008-04-17 |
| WO2008046049A1 (en) | 2008-04-17 |
| AR063278A1 (es) | 2009-01-14 |
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