JP2009537542A5 - - Google Patents

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Publication number
JP2009537542A5
JP2009537542A5 JP2009511057A JP2009511057A JP2009537542A5 JP 2009537542 A5 JP2009537542 A5 JP 2009537542A5 JP 2009511057 A JP2009511057 A JP 2009511057A JP 2009511057 A JP2009511057 A JP 2009511057A JP 2009537542 A5 JP2009537542 A5 JP 2009537542A5
Authority
JP
Japan
Prior art keywords
pyrrolidin
dimethylamino
carbonyl
phenyl
benzoyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2009511057A
Other languages
English (en)
Japanese (ja)
Other versions
JP2009537542A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2007/011765 external-priority patent/WO2007136668A2/en
Publication of JP2009537542A publication Critical patent/JP2009537542A/ja
Publication of JP2009537542A5 publication Critical patent/JP2009537542A5/ja
Withdrawn legal-status Critical Current

Links

JP2009511057A 2006-05-19 2007-05-16 ヒスタミン−３アンタゴニストとしてのｎ−ベンゾイルピロリジン−３−イルアミンおよびｎ−ベンジルピロリジン−３−イルアミン Withdrawn JP2009537542A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US80190506P 2006-05-19 2006-05-19
PCT/US2007/011765 WO2007136668A2 (en) 2006-05-19 2007-05-16 N-benzoyl-and n-benzylpyrrolidin-3-ylamines as histamine-3 antagonists

Publications (2)

Publication Number Publication Date
JP2009537542A JP2009537542A (ja) 2009-10-29
JP2009537542A5 true JP2009537542A5 (https=) 2010-07-08

Family

ID=38616614

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009511057A Withdrawn JP2009537542A (ja) 2006-05-19 2007-05-16 ヒスタミン−３アンタゴニストとしてのｎ−ベンゾイルピロリジン−３−イルアミンおよびｎ−ベンジルピロリジン−３−イルアミン

Country Status (12)

Country Link
US (1) US7842715B2 (https=)
EP (1) EP2027086B1 (https=)
JP (1) JP2009537542A (https=)
CN (1) CN101432261A (https=)
AR (1) AR061015A1 (https=)
AT (1) ATE533744T1 (https=)
AU (1) AU2007254232A1 (https=)
CA (1) CA2649913A1 (https=)
MX (1) MX2008014743A (https=)
PE (1) PE20080371A1 (https=)
TW (1) TW200811165A (https=)
WO (1) WO2007136668A2 (https=)

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EP1994022A2 (en) * 2006-03-15 2008-11-26 Wyeth a Corporation of the State of Delaware N-substituted-azacyclylamines as histamine-3 antagonists
TW200823204A (en) * 2006-10-17 2008-06-01 Arena Pharm Inc Biphenyl sulfonyl and phenyl-heteroaryl sulfonyl modulators of the histamine H3-receptor useful for the treatment of disorders related thereto
EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2009097995A1 (de) * 2008-02-07 2009-08-13 Sanofi-Aventis Neue phenyl-substituierte imidazolidine, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
US8236792B2 (en) * 2008-05-23 2012-08-07 Janssen Pharmaceutica Nv Substituted pyrrolidine amides as modulators of the histamine H3 receptor
CN102186479A (zh) * 2008-09-10 2011-09-14 凯利普西斯公司 用于治疗疾病的组胺受体的氨基嘧啶抑制剂
WO2012059443A2 (en) * 2010-11-01 2012-05-10 Neurotune Ag Novel neurotrypsin inhibitors
US8828994B2 (en) 2011-03-08 2014-09-09 Sanofi Di- and tri-substituted oxathiazine derivatives, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
EP2683699B1 (de) 2011-03-08 2015-06-24 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2766349B1 (de) 2011-03-08 2016-06-01 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
EP2683704B1 (de) 2011-03-08 2014-12-17 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
CN102784146A (zh) * 2011-05-19 2012-11-21 复旦大学 N-苯基喹唑啉-4-胺类衍生物的药用用途

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