JP2009533393A5 - - Google Patents

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Publication number
JP2009533393A5
JP2009533393A5 JP2009504750A JP2009504750A JP2009533393A5 JP 2009533393 A5 JP2009533393 A5 JP 2009533393A5 JP 2009504750 A JP2009504750 A JP 2009504750A JP 2009504750 A JP2009504750 A JP 2009504750A JP 2009533393 A5 JP2009533393 A5 JP 2009533393A5
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JP
Japan
Prior art keywords
alkyl
heteroaryl
aryl
alkynyl
alkenyl
Prior art date
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Abandoned
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JP2009504750A
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English (en)
Japanese (ja)
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JP2009533393A (ja
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Publication date
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Priority claimed from PCT/EP2007/053560 external-priority patent/WO2007116092A1/en
Publication of JP2009533393A publication Critical patent/JP2009533393A/ja
Publication of JP2009533393A5 publication Critical patent/JP2009533393A5/ja
Abandoned legal-status Critical Current

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JP2009504750A 2006-04-12 2007-04-12 酵素阻害薬 Abandoned JP2009533393A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US79130206P 2006-04-12 2006-04-12
US87016506P 2006-12-15 2006-12-15
PCT/EP2007/053560 WO2007116092A1 (en) 2006-04-12 2007-04-12 Enzyme inhibitors

Publications (2)

Publication Number Publication Date
JP2009533393A JP2009533393A (ja) 2009-09-17
JP2009533393A5 true JP2009533393A5 (OSRAM) 2010-05-27

Family

ID=38256669

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2009504750A Abandoned JP2009533393A (ja) 2006-04-12 2007-04-12 酵素阻害薬

Country Status (12)

Country Link
US (2) US7728146B2 (OSRAM)
EP (1) EP2007734A1 (OSRAM)
JP (1) JP2009533393A (OSRAM)
KR (1) KR20090004950A (OSRAM)
AU (1) AU2007235876A1 (OSRAM)
BR (1) BRPI0709984A2 (OSRAM)
CA (1) CA2649209A1 (OSRAM)
EA (1) EA200802054A1 (OSRAM)
IL (1) IL194339A0 (OSRAM)
MX (1) MX2008013130A (OSRAM)
NZ (1) NZ571761A (OSRAM)
WO (1) WO2007116092A1 (OSRAM)

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EP2025674A1 (de) 2007-08-15 2009-02-18 sanofi-aventis Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
US8933024B2 (en) 2010-06-18 2015-01-13 Sanofi Azolopyridin-3-one derivatives as inhibitors of lipases and phospholipases
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
US8710050B2 (en) 2011-03-08 2014-04-29 Sanofi Di and tri- substituted oxathiazine derivatives, method for the production, method for the production thereof, use thereof as medicine and drug containing said derivatives and use thereof
WO2012120052A1 (de) 2011-03-08 2012-09-13 Sanofi Mit carbozyklen oder heterozyklen substituierte oxathiazinderivate, verfahren zu deren herstellung, diese verbindungen enthaltende arzneimittel und deren verwendung
WO2012120056A1 (de) 2011-03-08 2012-09-13 Sanofi Tetrasubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
EP2683705B1 (de) 2011-03-08 2015-04-22 Sanofi Di- und trisubstituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2012120053A1 (de) 2011-03-08 2012-09-13 Sanofi Verzweigte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2014064215A1 (en) 2012-10-24 2014-05-01 INSERM (Institut National de la Santé et de la Recherche Médicale) TPL2 KINASE INHIBITORS FOR PREVENTING OR TREATING DIABETES AND FOR PROMOTING β-CELL SURVIVAL
KR20230098711A (ko) 2013-01-22 2023-07-04 비스타젠 쎄라퓨틱스, 인크. L-4-클로로키뉴레닌의 투여형 및 치료적 용도
EP3273981B1 (en) 2015-03-24 2020-04-29 INSERM - Institut National de la Santé et de la Recherche Médicale Method and pharmaceutical composition for use in the treatment of diabetes
JP2018521007A (ja) * 2015-05-22 2018-08-02 ヴィスタゲン セラピューティクス、インコーポレイテッド Ｌ−４−クロロキヌレニンの治療的使用
JP2019089710A (ja) * 2016-03-22 2019-06-13 国立研究開発法人科学技術振興機構 イミダゾール化合物及びこれを含有する医薬
RU2614737C1 (ru) * 2016-04-12 2017-03-28 Общество с ограниченной ответственностью "Нормофарм" Способ улучшения памяти

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