JP2009531292A5 - - Google Patents
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- JP2009531292A5 JP2009531292A5 JP2008555528A JP2008555528A JP2009531292A5 JP 2009531292 A5 JP2009531292 A5 JP 2009531292A5 JP 2008555528 A JP2008555528 A JP 2008555528A JP 2008555528 A JP2008555528 A JP 2008555528A JP 2009531292 A5 JP2009531292 A5 JP 2009531292A5
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- Prior art keywords
- substituted
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- compound
- pharmaceutical formulation
- Prior art date
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- 0 C*OB1N*CC2=C1****2 Chemical compound C*OB1N*CC2=C1****2 0.000 description 10
- JRGCEKUPJLWOMA-UHFFFAOYSA-N CC(Cc1ccccc1)(c1ccccc11)OB1O Chemical compound CC(Cc1ccccc1)(c1ccccc11)OB1O JRGCEKUPJLWOMA-UHFFFAOYSA-N 0.000 description 1
- MTWMLAABQMHLGF-UHFFFAOYSA-N COB1OCCc2cc(F)ccc12 Chemical compound COB1OCCc2cc(F)ccc12 MTWMLAABQMHLGF-UHFFFAOYSA-N 0.000 description 1
- HVONAVOROSIODW-UHFFFAOYSA-N Cc1cc(Oc(cc2)ccc2C#N)ccc1B(O)OC Chemical compound Cc1cc(Oc(cc2)ccc2C#N)ccc1B(O)OC HVONAVOROSIODW-UHFFFAOYSA-N 0.000 description 1
- WVDBMCNGKCSQFN-UHFFFAOYSA-N N#Cc(cc1)ccc1Oc1ccc(B(O)O)cc1 Chemical compound N#Cc(cc1)ccc1Oc1ccc(B(O)O)cc1 WVDBMCNGKCSQFN-UHFFFAOYSA-N 0.000 description 1
- UJEQOMQHKUCKBE-UHFFFAOYSA-N OB(c1ccccc11)OC1c1ccccc1 Chemical compound OB(c1ccccc11)OC1c1ccccc1 UJEQOMQHKUCKBE-UHFFFAOYSA-N 0.000 description 1
- GIENEGYOIYZESG-UHFFFAOYSA-N OB1OC(Cc(cc2)ccc2Cl)c2c1ccc(F)c2 Chemical compound OB1OC(Cc(cc2)ccc2Cl)c2c1ccc(F)c2 GIENEGYOIYZESG-UHFFFAOYSA-N 0.000 description 1
- ALCCZBHVEZPCSQ-UHFFFAOYSA-N OB1OC2(CCCCC2)c2ccccc12 Chemical compound OB1OC2(CCCCC2)c2ccccc12 ALCCZBHVEZPCSQ-UHFFFAOYSA-N 0.000 description 1
- TVMGRHFILUALSH-UHFFFAOYSA-N OB1Oc2ccccc2-c2ccccc12 Chemical compound OB1Oc2ccccc2-c2ccccc12 TVMGRHFILUALSH-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77453206P | 2006-02-16 | 2006-02-16 | |
| US60/774,532 | 2006-02-16 | ||
| US82388806P | 2006-08-29 | 2006-08-29 | |
| US60/823,888 | 2006-08-29 | ||
| PCT/US2007/062350 WO2007095638A2 (en) | 2006-02-16 | 2007-02-16 | Boron-containing small molecules as anti-inflammatory agents |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013173486A Division JP2013253097A (ja) | 2006-02-16 | 2013-08-23 | 抗炎症剤としてのホウ素含有小分子 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009531292A JP2009531292A (ja) | 2009-09-03 |
| JP2009531292A5 true JP2009531292A5 (enExample) | 2010-04-08 |
| JP5419466B2 JP5419466B2 (ja) | 2014-02-19 |
Family
ID=38372267
Family Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008555528A Active JP5419466B2 (ja) | 2006-02-16 | 2007-02-16 | 抗炎症剤としてのホウ素含有小分子 |
| JP2013173486A Pending JP2013253097A (ja) | 2006-02-16 | 2013-08-23 | 抗炎症剤としてのホウ素含有小分子 |
| JP2015082026A Pending JP2015147795A (ja) | 2006-02-16 | 2015-04-13 | 抗炎症剤としてのホウ素含有小分子 |
| JP2016139202A Active JP6266708B2 (ja) | 2006-02-16 | 2016-07-14 | 抗炎症剤としてのホウ素含有小分子 |
Family Applications After (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2013173486A Pending JP2013253097A (ja) | 2006-02-16 | 2013-08-23 | 抗炎症剤としてのホウ素含有小分子 |
| JP2015082026A Pending JP2015147795A (ja) | 2006-02-16 | 2015-04-13 | 抗炎症剤としてのホウ素含有小分子 |
| JP2016139202A Active JP6266708B2 (ja) | 2006-02-16 | 2016-07-14 | 抗炎症剤としてのホウ素含有小分子 |
Country Status (24)
| Country | Link |
|---|---|
| US (12) | US8168614B2 (enExample) |
| EP (2) | EP1988779B1 (enExample) |
| JP (4) | JP5419466B2 (enExample) |
| KR (7) | KR20150113219A (enExample) |
| CN (2) | CN101420854B (enExample) |
| AU (1) | AU2007214421B2 (enExample) |
| BR (1) | BRPI0708051A2 (enExample) |
| CA (2) | CA2642583C (enExample) |
| CY (1) | CY1121899T1 (enExample) |
| DK (2) | DK1988779T5 (enExample) |
| ES (2) | ES2728455T3 (enExample) |
| HR (1) | HRP20150710T1 (enExample) |
| HU (2) | HUE025048T2 (enExample) |
| IL (2) | IL193230A (enExample) |
| ME (1) | ME02188B (enExample) |
| MX (2) | MX2008010381A (enExample) |
| NZ (1) | NZ570257A (enExample) |
| PL (2) | PL1988779T3 (enExample) |
| PT (2) | PT2719388T (enExample) |
| RS (1) | RS54108B1 (enExample) |
| RU (2) | RU2508113C2 (enExample) |
| SI (2) | SI2719388T1 (enExample) |
| WO (1) | WO2007095638A2 (enExample) |
| ZA (1) | ZA200806754B (enExample) |
Families Citing this family (126)
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| BRPI0711155A2 (pt) | 2006-05-02 | 2011-08-23 | Anacor Pharmaceuticals Inc | terapêuticos contendo boro resistentes hidroliticamente e métodos de uso |
| JO3598B1 (ar) * | 2006-10-10 | 2020-07-05 | Infinity Discovery Inc | الاحماض والاسترات البورونية كمثبطات اميد هيدروليز الحامض الدهني |
| US10265265B2 (en) | 2007-03-15 | 2019-04-23 | Drug Delivery Solutions Limited | Topical composition |
| JO3396B1 (ar) * | 2007-06-20 | 2019-10-20 | Anacor Pharmaceuticals Inc | جزيئات صغيرة تحتوي على البورون |
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| US9745567B2 (en) | 2008-04-28 | 2017-08-29 | Revalesio Corporation | Compositions and methods for treating multiple sclerosis |
| US9523090B2 (en) | 2007-10-25 | 2016-12-20 | Revalesio Corporation | Compositions and methods for treating inflammation |
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| RU2015109165A (ru) | 2008-03-06 | 2015-11-10 | Анакор Фармасьютикалз, Инк. | Борсодержащие малые молекулы в качестве противовоспалительных агентов |
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