JP2009526761A - ヘテロ二環式チオフェン化合物および使用の方法 - Google Patents
ヘテロ二環式チオフェン化合物および使用の方法 Download PDFInfo
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- JP2009526761A JP2009526761A JP2008552481A JP2008552481A JP2009526761A JP 2009526761 A JP2009526761 A JP 2009526761A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2008552481 A JP2008552481 A JP 2008552481A JP 2009526761 A JP2009526761 A JP 2009526761A
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- alkyl
- aryl
- heteroaryl
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
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Applications Claiming Priority (2)
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| US76341406P | 2006-01-30 | 2006-01-30 | |
| PCT/US2007/002352 WO2008063202A2 (en) | 2006-01-30 | 2007-01-30 | Heterobicyclic thiophene compounds for the treatment of cancer |
Publications (2)
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| JP2009526761A true JP2009526761A (ja) | 2009-07-23 |
| JP2009526761A5 JP2009526761A5 (https=) | 2011-03-10 |
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| JP2008552481A Pending JP2009526761A (ja) | 2006-01-30 | 2007-01-30 | ヘテロ二環式チオフェン化合物および使用の方法 |
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| Country | Link |
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| US (1) | US8003662B2 (https=) |
| EP (1) | EP1989211A2 (https=) |
| JP (1) | JP2009526761A (https=) |
| CN (1) | CN101522687A (https=) |
| AR (1) | AR059246A1 (https=) |
| CA (1) | CA2636242A1 (https=) |
| TW (1) | TW200806675A (https=) |
| WO (1) | WO2008063202A2 (https=) |
Cited By (9)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2010523568A (ja) * | 2007-04-05 | 2010-07-15 | アムジエン・インコーポレーテツド | オーロラキナーゼ調節物質及び使用方法 |
| WO2011162368A1 (ja) * | 2010-06-25 | 2011-12-29 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| JP2012525336A (ja) * | 2009-04-27 | 2012-10-22 | エラン ファーマシューティカルズ，インコーポレイテッド | α−４インテグリンのピリジノンアンタゴニスト |
| JP2013503903A (ja) * | 2009-09-03 | 2013-02-04 | アラーガン インコーポレイテッド | チロシンキナーゼモジュレーターとしての化合物 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| JP2021500378A (ja) * | 2018-03-08 | 2021-01-07 | ウェルマーカー・バイオ・カンパニー・リミテッドＷｅｌｌｍａｒｋｅｒ Ｂｉｏ ＣＯ．， Ｌｔｄ． | チエノピリジン誘導体およびそれを含む医薬組成物 |
| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| CN100406567C (zh) * | 2002-01-22 | 2008-07-30 | 生物材料公司 | 生物可降解聚合物的干燥方法 |
| AU2006229343A1 (en) * | 2005-03-28 | 2006-10-05 | Kirin Pharma Kabushiki Kaisha | Thienopyridine derivative, or quinoline derivative, or quinazoline derivative, having c-Met autophosphorylation inhibiting potency |
| AU2006313456B2 (en) | 2005-05-20 | 2011-06-23 | Methylgene Inc. | Inhibitors of VEGF receptor and HGF receptor signaling |
| CN101796055B (zh) | 2005-05-20 | 2013-09-04 | 梅特希尔基因公司 | Vegf受体和hgf受体信号的抑制剂 |
| EP2038289A2 (en) * | 2006-04-21 | 2009-03-25 | Amgen Inc. | Thieno-[2,3-d]pyrimidine and thieno-pyridazine compounds and methods of use |
| JP2009539878A (ja) * | 2006-06-08 | 2009-11-19 | アレイ バイオファーマ、インコーポレイテッド | キノリン化合物および使用方法 |
| US8778977B2 (en) | 2006-06-30 | 2014-07-15 | Sunesis Pharmaceuticals, Inc. | Pyridinonyl PDK1 inhibitors |
| US8907091B2 (en) * | 2007-08-29 | 2014-12-09 | Methylgene Inc. | Processes and intermediates for preparing fused heterocyclic kinase inhibitors |
| BRPI0816064B8 (pt) | 2007-08-29 | 2021-05-25 | Methylgene Inc | composto inibidor da atividade de proteína tirosina quinase, seu uso, e composição farmacêutica |
| JP5693239B2 (ja) | 2008-01-23 | 2015-04-01 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | ４−ピリジノン化合物および癌についてのその使用 |
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| JP2013503903A (ja) * | 2009-09-03 | 2013-02-04 | アラーガン インコーポレイテッド | チロシンキナーゼモジュレーターとしての化合物 |
| JP5889788B2 (ja) * | 2010-06-25 | 2016-03-22 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
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| WO2011162368A1 (ja) * | 2010-06-25 | 2011-12-29 | 興和株式会社 | 新規な縮合ピリジン又は縮合ピリミジン誘導体及びこれを含有する医薬 |
| WO2014038881A3 (ko) * | 2012-09-06 | 2014-05-08 | 씨제이제일제당 (주) | 피리돈 유도체를 포함하는 단백질 키나제 억제제 |
| JP2021500378A (ja) * | 2018-03-08 | 2021-01-07 | ウェルマーカー・バイオ・カンパニー・リミテッドＷｅｌｌｍａｒｋｅｒ Ｂｉｏ ＣＯ．， Ｌｔｄ． | チエノピリジン誘導体およびそれを含む医薬組成物 |
| JP2022535108A (ja) * | 2019-06-04 | 2022-08-04 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP7820152B2 (ja) | 2019-06-04 | 2026-02-25 | エグゼリクシス， インコーポレイテッド | キナーゼ依存性障害の処置のための化合物 |
| JP2023510296A (ja) * | 2020-01-07 | 2023-03-13 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP7434575B2 (ja) | 2020-01-07 | 2024-02-20 | メッドシャイン ディスカバリー インコーポレイテッド | 重水素化チエノピリジン系化合物 |
| JP2023550380A (ja) * | 2020-11-24 | 2023-12-01 | チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド | 重水素修飾チエノピリドン化合物 |
Also Published As
| Publication number | Publication date |
|---|---|
| CN101522687A (zh) | 2009-09-02 |
| WO2008063202A3 (en) | 2009-01-22 |
| AR059246A1 (es) | 2008-03-19 |
| EP1989211A2 (en) | 2008-11-12 |
| US20070197537A1 (en) | 2007-08-23 |
| US8003662B2 (en) | 2011-08-23 |
| CA2636242A1 (en) | 2008-05-29 |
| WO2008063202A2 (en) | 2008-05-29 |
| TW200806675A (en) | 2008-02-01 |
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