JP2009511513A5 - - Google Patents
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- Publication number
- JP2009511513A5 JP2009511513A5 JP2008534890A JP2008534890A JP2009511513A5 JP 2009511513 A5 JP2009511513 A5 JP 2009511513A5 JP 2008534890 A JP2008534890 A JP 2008534890A JP 2008534890 A JP2008534890 A JP 2008534890A JP 2009511513 A5 JP2009511513 A5 JP 2009511513A5
- Authority
- JP
- Japan
- Prior art keywords
- group
- radical
- formula
- alkyl
- solvate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 0 C*(*C(C*1c2ccc(*(CCOC3)C3=O)cc2)OC1=O)C(c1ccc(N)[n]1)=O Chemical compound C*(*C(C*1c2ccc(*(CCOC3)C3=O)cc2)OC1=O)C(c1ccc(N)[n]1)=O 0.000 description 11
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005048824A DE102005048824A1 (de) | 2005-10-10 | 2005-10-10 | Behandlung und Prophylaxe von Mikroangiopathien |
| PCT/EP2006/009373 WO2007042146A1 (de) | 2005-10-10 | 2006-09-27 | Behandlung und prophylaxe von mikroangiopathien |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009511513A JP2009511513A (ja) | 2009-03-19 |
| JP2009511513A5 true JP2009511513A5 (https=) | 2009-11-12 |
Family
ID=37492407
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008534890A Pending JP2009511513A (ja) | 2005-10-10 | 2006-09-27 | 微小血管障害の処置および予防 |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US20100160301A1 (https=) |
| EP (1) | EP1937271A1 (https=) |
| JP (1) | JP2009511513A (https=) |
| KR (1) | KR20080067647A (https=) |
| CN (1) | CN101325957A (https=) |
| AU (1) | AU2006301650A1 (https=) |
| BR (1) | BRPI0617202A2 (https=) |
| CA (1) | CA2624963A1 (https=) |
| CR (1) | CR9878A (https=) |
| DE (1) | DE102005048824A1 (https=) |
| EC (1) | ECSP088358A (https=) |
| IL (1) | IL190745A0 (https=) |
| NO (1) | NO20082120L (https=) |
| RU (1) | RU2008118100A (https=) |
| SV (1) | SV2009002865A (https=) |
| WO (1) | WO2007042146A1 (https=) |
| ZA (1) | ZA200803048B (https=) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| EP1685841A1 (en) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention and treatment of thromboembolic disorders |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| US8188270B2 (en) | 2005-10-04 | 2012-05-29 | Bayer Schering Pharma Aktiengesellschaft | Polymorphous form of 5-chloro-N-({(5S)-2-oxo-3[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidine-5-yl}-methyl)-2-thiophene carboxamide |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| WO2007092961A2 (en) * | 2006-02-09 | 2007-08-16 | University Of New Orleans Research & Technologies Foundation | Antibacterial agents |
| MX2009009304A (es) * | 2007-03-01 | 2009-11-18 | Novartis Ag | Inhibidores de cinasa pim y metodos para su uso. |
| DE102007018662A1 (de) * | 2007-04-20 | 2008-10-23 | Bayer Healthcare Ag | Oxazolidinone zur Behandlung und Prophylaxe von pulmonaler Hypertonie |
| WO2009018807A1 (de) * | 2007-08-06 | 2009-02-12 | Schebo Biotech Ag | Oxazolidinone als faktor xa- inhibitoren, verfahren zu ihrer herstellung und ihre verwendung in der therapie |
| JP5422569B2 (ja) * | 2008-02-21 | 2014-02-19 | サノフイ | 凝固第Ｘａ因子及びトロンビンの阻害剤としてのクロロチオフェン−イソオキサゾール類 |
| US7816355B1 (en) | 2009-04-28 | 2010-10-19 | Apotex Pharmachem Inc | Processes for the preparation of rivaroxaban and intermediates thereof |
| CN104693139B (zh) * | 2011-01-07 | 2017-04-19 | 浙江九洲药业股份有限公司 | 一种合成利伐沙班中间体的新工艺 |
| CN102746287B (zh) * | 2012-06-21 | 2014-05-28 | 成都苑东药业有限公司 | 一种恶唑烷酮化合物及其制备方法 |
| CN103724336B (zh) * | 2013-12-24 | 2015-10-21 | 悦康药业集团有限公司 | 一种新型抗凝血药物的合成方法 |
| CN104402876A (zh) * | 2014-11-25 | 2015-03-11 | 沈阳药科大学 | 噁唑烷酮类化合物及其应用 |
| CN104478866B (zh) * | 2014-12-05 | 2017-07-07 | 广东东阳光药业有限公司 | 噁唑烷酮类化合物及其在药物中的应用 |
| CN104447728B (zh) * | 2014-12-05 | 2017-01-04 | 广东东阳光药业有限公司 | 噁唑烷酮类化合物及其在药物中的应用 |
| CN104447730B (zh) * | 2014-12-05 | 2017-11-07 | 广东东阳光药业有限公司 | 噁唑烷酮类化合物及其在药物中的应用 |
| CN104478869B (zh) * | 2014-12-05 | 2017-04-12 | 广东东阳光药业有限公司 | 噁唑烷酮类化合物及其在药物中的应用 |
| CN104497008B (zh) * | 2014-12-09 | 2016-11-16 | 广东东阳光药业有限公司 | 取代噁唑烷酮类化合物及其使用方法和用途 |
| EP3078378B1 (en) | 2015-04-08 | 2020-06-24 | Vaiomer | Use of factor xa inhibitors for regulating glycemia |
| US11608320B2 (en) | 2020-02-02 | 2023-03-21 | Kuwait University | Oxazolidinone hydroxamic acid derivatives |
| WO2021184339A1 (en) | 2020-03-20 | 2021-09-23 | Merck Sharp & Dohme Corp. | Oxazolidinone compound and methods of use thereof as an antibacterial agent |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2811555A (en) * | 1955-05-02 | 1957-10-29 | Eastman Kodak Co | Reduction of 2-nitroso-5-diethylaminotoluene |
| LU80081A1 (fr) * | 1977-08-26 | 1979-05-15 | Delalande Sa | Nouvelles hydroxymethyl-5 oxazolidinones-2,leur procede de preparation et leur application therapeutique |
| US4128654A (en) * | 1978-02-10 | 1978-12-05 | E. I. Du Pont De Nemours And Company | 5-Halomethyl-3-phenyl-2-oxazolidinones |
| DE3822650A1 (de) * | 1988-07-05 | 1990-02-01 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
| ATE146783T1 (de) * | 1991-11-01 | 1997-01-15 | Upjohn Co | Substituierte aryl- und heteroaryl- phenyloxazolidinone |
| US5349045A (en) * | 1993-01-26 | 1994-09-20 | United States Surgical Corporation | Polymer derived from cyclic amide and medical devices manufactured therefrom |
| ATE181735T1 (de) * | 1993-05-01 | 1999-07-15 | Merck Patent Gmbh | Substituierte 1-phenyl-oxazolidin-2-on derivate, deren herstellung und deren verwendung als adhäsionsrezeptor-antagonisten |
| HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
| DE19524765A1 (de) * | 1995-07-07 | 1997-01-09 | Boehringer Mannheim Gmbh | Neue Oxazolidinonderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel |
| DE19962924A1 (de) * | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
-
2005
- 2005-10-10 DE DE102005048824A patent/DE102005048824A1/de not_active Withdrawn
-
2006
- 2006-09-27 EP EP06792284A patent/EP1937271A1/de not_active Withdrawn
- 2006-09-27 BR BRPI0617202-4A patent/BRPI0617202A2/pt not_active IP Right Cessation
- 2006-09-27 AU AU2006301650A patent/AU2006301650A1/en not_active Abandoned
- 2006-09-27 US US12/089,650 patent/US20100160301A1/en not_active Abandoned
- 2006-09-27 WO PCT/EP2006/009373 patent/WO2007042146A1/de not_active Ceased
- 2006-09-27 JP JP2008534890A patent/JP2009511513A/ja active Pending
- 2006-09-27 KR KR1020087011170A patent/KR20080067647A/ko not_active Withdrawn
- 2006-09-27 CA CA002624963A patent/CA2624963A1/en not_active Abandoned
- 2006-09-27 CN CNA2006800463670A patent/CN101325957A/zh active Pending
- 2006-09-27 RU RU2008118100/15A patent/RU2008118100A/ru not_active Application Discontinuation
-
2008
- 2008-04-07 ZA ZA200803048A patent/ZA200803048B/xx unknown
- 2008-04-09 IL IL190745A patent/IL190745A0/en unknown
- 2008-04-09 EC EC2008008358A patent/ECSP088358A/es unknown
- 2008-04-09 SV SV2008002865A patent/SV2009002865A/es not_active Application Discontinuation
- 2008-04-09 CR CR9878A patent/CR9878A/es not_active Application Discontinuation
- 2008-05-06 NO NO20082120A patent/NO20082120L/no not_active Application Discontinuation
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