JP2009179634A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2009179634A5 JP2009179634A5 JP2009115279A JP2009115279A JP2009179634A5 JP 2009179634 A5 JP2009179634 A5 JP 2009179634A5 JP 2009115279 A JP2009115279 A JP 2009115279A JP 2009115279 A JP2009115279 A JP 2009115279A JP 2009179634 A5 JP2009179634 A5 JP 2009179634A5
- Authority
- JP
- Japan
- Prior art keywords
- escitalopram
- salt
- oxalate
- base
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200500912 | 2005-06-22 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008517323A Division JP4906852B2 (ja) | 2005-06-22 | 2006-06-22 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2009179634A JP2009179634A (ja) | 2009-08-13 |
| JP2009179634A5 true JP2009179634A5 (enExample) | 2012-01-19 |
Family
ID=37546630
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008517323A Active JP4906852B2 (ja) | 2005-06-22 | 2006-06-22 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2008260742A Active JP4415056B2 (ja) | 2005-06-22 | 2008-10-07 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2009115279A Pending JP2009179634A (ja) | 2005-06-22 | 2009-05-12 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2009115280A Pending JP2009179635A (ja) | 2005-06-22 | 2009-05-12 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2011255804A Active JP5731957B2 (ja) | 2005-06-22 | 2011-11-24 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008517323A Active JP4906852B2 (ja) | 2005-06-22 | 2006-06-22 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2008260742A Active JP4415056B2 (ja) | 2005-06-22 | 2008-10-07 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009115280A Pending JP2009179635A (ja) | 2005-06-22 | 2009-05-12 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
| JP2011255804A Active JP5731957B2 (ja) | 2005-06-22 | 2011-11-24 | エスシタロプラムの結晶質塩基、およびエスシタロプラム塩基を含む口腔内分散性錠剤 |
Country Status (39)
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0123400D0 (en) | 2001-09-28 | 2001-11-21 | Novartis Ag | Organic compounds |
| WO2008059514A2 (en) * | 2006-07-31 | 2008-05-22 | Cadila Healthcare Limited | Process for preparing escitalopram |
| EP2134325A2 (en) * | 2007-03-01 | 2009-12-23 | Aurobindo Pharma Limited | Stable solid dosage forms of an antidepressant |
| HUE028897T2 (en) | 2010-07-23 | 2017-01-30 | H Lundbeck As | A method of purifying pharmaceutically acceptable salts of escitalopram |
| CN103360353A (zh) * | 2013-08-07 | 2013-10-23 | 中国药科大学 | 草酸艾司西酞普兰杂质的制备方法 |
| JP2018016569A (ja) * | 2016-07-26 | 2018-02-01 | 株式会社トクヤマ | (1s)−1−[3−(ジメチルアミノ)プロピル]−1−(4−フルオロフェニル)−1,3−ジヒドロイソベンゾフラン−5−カルボニトリル蓚酸塩の製造方法 |
| JP6423133B1 (ja) * | 2017-04-10 | 2018-11-14 | 東和薬品株式会社 | エスシタロプラム医薬組成物 |
| CN110711198B (zh) * | 2018-07-12 | 2022-03-15 | 山东大学 | D-甘露糖在制备抗抑郁药物中的应用 |
| KR102331187B1 (ko) | 2019-04-09 | 2021-11-26 | 주식회사 라이트팜텍 | 에스시탈로프람을 함유하는 안정성이 우수한 경구용 액제 조성물 및 그의 제조방법 |
| EP4277661A1 (en) * | 2021-01-18 | 2023-11-22 | Anton Frenkel | Pharmaceutical dosage form |
Family Cites Families (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1526331A (en) | 1976-01-14 | 1978-09-27 | Kefalas As | Phthalanes |
| GB8814057D0 (en) | 1988-06-14 | 1988-07-20 | Lundbeck & Co As H | New enantiomers & their isolation |
| JPH05222041A (ja) * | 1992-02-13 | 1993-08-31 | Mitsubishi Gas Chem Co Inc | アデニン誘導体の精製法 |
| EP0743850B1 (en) * | 1994-01-27 | 1999-10-06 | The Board Of Regents Of The University Of Oklahoma | Rapidly dissolving oral dosage form |
| US5607697A (en) * | 1995-06-07 | 1997-03-04 | Cima Labs, Incorporated | Taste masking microparticles for oral dosage forms |
| EP0993524B1 (en) | 1997-06-30 | 2002-11-20 | Beloit Technologies, Inc. | Method and apparatus for the high speed application of coating to a traveling paper web |
| SK283309B6 (sk) | 1997-07-08 | 2003-05-02 | H. Lundbeck A/S | Spôsob výroby citalopramu a medziprodukty |
| DK1042310T3 (da) | 1997-11-11 | 2002-12-02 | Lundbeck & Co As H | Fremgangsmåde til fremstilling af citalopram |
| FR2785538B1 (fr) * | 1998-11-06 | 2004-04-09 | Prographarm Laboratoires | Comprime a delitement rapide perfectionne |
| US20020071864A1 (en) * | 1999-03-25 | 2002-06-13 | Yuhan Corporation | Rapidly disintegrable tablet for oral administration |
| ITMI991579A1 (it) | 1999-06-25 | 2001-01-15 | Lundbeck & Co As H | Metodo per la preparazione di citalopram |
| ITMI991581A1 (it) | 1999-06-25 | 2001-01-15 | Lundbeck & Co As H | Metodo per la preparazione di citalopram |
| JP2001226372A (ja) * | 1999-12-06 | 2001-08-21 | Sumika Fine Chemicals Co Ltd | ロサルタンの結晶性または結晶化された酸付加塩およびロサルタンの精製方法 |
| GB2357762B (en) * | 2000-03-13 | 2002-01-30 | Lundbeck & Co As H | Crystalline base of citalopram |
| AU2001294192A1 (en) * | 2000-10-06 | 2002-04-22 | Takeda Chemical Industries Ltd. | Solid preparations |
| WO2002032403A1 (fr) * | 2000-10-16 | 2002-04-25 | Daiichi Pharmaceutical Co., Ltd. | Compositions medicales pouvant se desintegrer rapidement dans la cavite buccale et leur procede de production |
| US7799342B2 (en) * | 2000-12-06 | 2010-09-21 | Wyeth Llc | Fast dissolving tablet |
| CA2360303C (en) * | 2000-12-22 | 2003-08-12 | Marco Villa | Process for the preparation of pure citalopram |
| SK284418B6 (sk) * | 2000-12-28 | 2005-04-01 | H. Lundbeck A/S | Spôsob výroby citalopramu |
| CZ20033267A3 (en) * | 2001-05-01 | 2004-06-16 | H. Lundbeck A/S | The use of enantiomeric pure escitalopram |
| US6872405B2 (en) * | 2001-05-10 | 2005-03-29 | Yamanouchi Pharmaceutical Co., Ltd. | Quick-disintegrating tablet in buccal cavity and manufacturing method thereof |
| GB0113842D0 (en) * | 2001-06-07 | 2001-08-01 | Boots Co Plc | Therapeutic agents |
| AR034612A1 (es) * | 2001-06-25 | 2004-03-03 | Lundbeck & Co As H | Proceso para la preparacion del citalopram racemico y/o del s- o r-citalopram mediante la separacion de una mezcla de r- y s-citalopram |
| AR034759A1 (es) | 2001-07-13 | 2004-03-17 | Lundbeck & Co As H | Metodo para la preparacion de escitalopram |
| PT1522539E (pt) * | 2001-07-31 | 2007-03-30 | Lundbeck & Co As H | Composição cristalina contendo escitalopram |
| IS7239A (is) * | 2001-12-14 | 2004-04-29 | H. Lundbeck A/S | Aðferð til framleiðslu á essítalóprami |
| AU2003222435A1 (en) * | 2002-01-07 | 2003-07-24 | Sun Pharmaceutical Industries Limited | Process for the preparation of 1-(3-(dimethylamino)propyl)-1-(4-fluorophenyl)- 1,3-dihydro-5-isobenzofuran carbonitrile |
| FR2834889B1 (fr) * | 2002-01-18 | 2004-04-02 | Roquette Freres | Forme pharmaceutique solide orodispersible |
| GB0204607D0 (en) * | 2002-02-27 | 2002-04-10 | Matrix Lab Ltd | Process |
| WO2003092659A1 (en) * | 2002-05-03 | 2003-11-13 | Skyepharma Canada Inc. | Oral dosage forms comprising fenofibrate |
| MEP5808A (xx) | 2002-12-23 | 2010-02-10 | Lundbeck & Co As H | Ecitalopram bromhidrat i postupak za njegovo pripremanje |
| CN1510024A (zh) * | 2002-12-24 | 2004-07-07 | 北京德众万全药物技术开发有限公司 | 可用于制备西酞普兰(s)-对映异构体的新的化合物及其制备方法 |
| DE10305984A1 (de) * | 2003-02-13 | 2004-09-02 | Helm Ag | Salze organischer Säuren mit Clopidogrel und deren Verwendung zur Herstellung phamazeutischer Formulierungen |
| AU2004238321B2 (en) * | 2003-05-07 | 2009-08-27 | Samyang Biopharmaceuticals Corporation | Highly plastic granules for making fast melting tablets |
| ES2688193T3 (es) * | 2003-10-15 | 2018-10-31 | Fuji Chemical Industry Co., Ltd. | Comprimido de disgregación rápida en la cavidad oral |
| WO2005049596A1 (en) * | 2003-11-20 | 2005-06-02 | Natco Pharma Limited | A process for the preparation of high purity escitalopram |
| HU227491B1 (en) * | 2003-11-25 | 2011-07-28 | Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag | Tablet containing citalopram hydrogen bromide |
| NZ549100A (en) * | 2004-03-05 | 2010-02-26 | Lundbeck & Co As H | Crystalline composition containing escitalopram oxalate |
| EP1877394A1 (en) * | 2005-04-04 | 2008-01-16 | Jubilant Organosys Limited | Process for the preparation of escitalopram or its acid addition salts |
-
2006
- 2006-06-15 TW TW100102601A patent/TWI358407B/zh not_active IP Right Cessation
- 2006-06-15 TW TW095121358A patent/TWI347942B/zh not_active IP Right Cessation
- 2006-06-21 MY MYPI20062933A patent/MY143252A/en unknown
- 2006-06-21 MY MYPI2010000618A patent/MY143239A/en unknown
- 2006-06-21 AR ARP060102654A patent/AR055062A1/es not_active Application Discontinuation
- 2006-06-22 PL PL06742481T patent/PL1896439T5/pl unknown
- 2006-06-22 MX MX2007015328A patent/MX2007015328A/es active IP Right Grant
- 2006-06-22 EA EA201001108A patent/EA201001108A1/ru unknown
- 2006-06-22 PT PT06742481T patent/PT1896439E/pt unknown
- 2006-06-22 GB GB0724557A patent/GB2442160B/en not_active Expired - Fee Related
- 2006-06-22 PL PL384185A patent/PL384185A1/pl unknown
- 2006-06-22 EP EP10179395A patent/EP2325177A1/en not_active Withdrawn
- 2006-06-22 EA EA200800102A patent/EA019239B1/ru not_active IP Right Cessation
- 2006-06-22 AU AU2006261452A patent/AU2006261452B2/en not_active Withdrawn - After Issue
- 2006-06-22 RS RS20110057A patent/RS51575B2/sr unknown
- 2006-06-22 CA CA002646780A patent/CA2646780A1/en not_active Abandoned
- 2006-06-22 FI FI20077133A patent/FI20077133L/fi unknown
- 2006-06-22 AT AT06742481T patent/ATE497500T1/de active
- 2006-06-22 ES ES06742481.2T patent/ES2356838T5/es active Active
- 2006-06-22 SK SK50040-2007A patent/SK500402007A3/sk unknown
- 2006-06-22 CA CA2612827A patent/CA2612827C/en not_active Expired - Fee Related
- 2006-06-22 SG SG201100648-3A patent/SG169358A1/en unknown
- 2006-06-22 KR KR1020117005777A patent/KR101340815B1/ko active Active
- 2006-06-22 WO PCT/DK2006/000366 patent/WO2006136169A2/en not_active Ceased
- 2006-06-22 CZ CZ20080430A patent/CZ300686B6/cs not_active IP Right Cessation
- 2006-06-22 DK DK06742481.2T patent/DK1896439T4/en active
- 2006-06-22 CZ CZ20070898A patent/CZ299906B6/cs not_active IP Right Cessation
- 2006-06-22 DE DE112006001619T patent/DE112006001619T5/de not_active Withdrawn
- 2006-06-22 CN CN201010286088XA patent/CN101928269A/zh active Pending
- 2006-06-22 DE DE602006019961T patent/DE602006019961D1/de active Active
- 2006-06-22 KR KR1020117015711A patent/KR20110084341A/ko not_active Ceased
- 2006-06-22 EP EP06742481.2A patent/EP1896439B2/en active Active
- 2006-06-22 EP EP10179318A patent/EP2385044A1/en not_active Withdrawn
- 2006-06-22 CN CNA2006800200393A patent/CN101189220A/zh active Pending
- 2006-06-22 HU HU0800135A patent/HUP0800135A3/hu unknown
- 2006-06-22 AT AT0900506U patent/AT10983U1/de not_active IP Right Cessation
- 2006-06-22 KR KR1020077028918A patent/KR20080018191A/ko not_active Ceased
- 2006-06-22 KR KR1020107026804A patent/KR20100133023A/ko not_active Ceased
- 2006-06-22 CZ CZ20080429A patent/CZ301286B6/cs not_active IP Right Cessation
- 2006-06-22 TR TR2007/08792T patent/TR200708792T1/xx unknown
- 2006-06-22 GB GB0811164A patent/GB2448834B/en not_active Expired - Fee Related
- 2006-06-22 JP JP2008517323A patent/JP4906852B2/ja active Active
- 2006-06-22 HR HRP20110093TT patent/HRP20110093T4/hr unknown
- 2006-06-22 ES ES200750085A patent/ES2319073B1/es not_active Expired - Fee Related
- 2006-06-22 ZA ZA200711066A patent/ZA200711066B/xx unknown
- 2006-06-22 TR TR2010/00625T patent/TR201000625T1/xx unknown
- 2006-06-22 SI SI200630923T patent/SI1896439T2/sl unknown
- 2006-06-22 FI FI20080548A patent/FI20080548L/fi unknown
- 2006-06-22 KR KR1020127014205A patent/KR20120064140A/ko not_active Ceased
- 2006-06-22 EE EEU200800003U patent/EE00773U1/xx not_active IP Right Cessation
- 2006-06-22 BR BRPI0612295-7A patent/BRPI0612295A2/pt not_active IP Right Cessation
- 2006-06-22 UA UAA200800362A patent/UA86536C2/ru unknown
-
2007
- 2007-11-18 IL IL187454A patent/IL187454A0/en unknown
- 2007-12-19 BG BG10110024A patent/BG66086B1/bg unknown
- 2007-12-21 LV LVP-07-157A patent/LV13677B/lv unknown
-
2008
- 2008-01-14 IS IS8705A patent/IS8705A/is unknown
- 2008-01-18 NO NO20080359A patent/NO20080359L/no unknown
- 2008-01-21 DK DK200800075A patent/DK200800075A/da not_active Application Discontinuation
- 2008-01-21 LT LT2008005A patent/LT5550B/lt not_active IP Right Cessation
- 2008-10-07 JP JP2008260742A patent/JP4415056B2/ja active Active
-
2009
- 2009-02-27 DK DKPA200900284A patent/DK200900284A/da not_active Application Discontinuation
- 2009-03-10 ZA ZA200901698A patent/ZA200901698B/en unknown
- 2009-05-12 JP JP2009115279A patent/JP2009179634A/ja active Pending
- 2009-05-12 JP JP2009115280A patent/JP2009179635A/ja active Pending
- 2009-07-07 AT AT0041709U patent/AT11883U1/de not_active IP Right Cessation
-
2010
- 2010-03-05 AU AU2010200844A patent/AU2010200844A1/en not_active Withdrawn
- 2010-12-20 NO NO20101777A patent/NO20101777L/no not_active Application Discontinuation
- 2010-12-27 AR ARP100104958A patent/AR079750A2/es not_active Application Discontinuation
-
2011
- 2011-02-03 CY CY20111100116T patent/CY1112392T1/el unknown
- 2011-11-24 JP JP2011255804A patent/JP5731957B2/ja active Active
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2009179634A5 (enExample) | ||
| JP2006519255A5 (enExample) | ||
| JP2009138000A5 (enExample) | ||
| JP2018502909A5 (enExample) | ||
| CN1227233C (zh) | 纯晶形的5-氯-3-(4-甲磺酰基苯基)-6′-甲基-[2,3′]联吡啶及其合成方法 | |
| JP2010095546A5 (enExample) | ||
| JP2014501282A5 (enExample) | ||
| JP2014503001A5 (enExample) | ||
| JP2005520923A5 (enExample) | ||
| JP2004536093A5 (ja) | R−及びs−シタロプラムの混合物を分離することによってラセミシタロプラム及びs−もしくはr−シタロプラムを製造する方法 | |
| JP2018528948A5 (enExample) | ||
| JP2017520564A5 (enExample) | ||
| JP2013508368A5 (enExample) | ||
| JP2019524752A5 (enExample) | ||
| JP2012508747A5 (enExample) | ||
| JP2018009003A5 (enExample) | ||
| JP2005502603A5 (enExample) | ||
| CN103443084A (zh) | 制备苯达莫司汀的方法 | |
| JP2014503456A5 (enExample) | ||
| HRP20110093T1 (hr) | Kristalna baza escitaloprama i orodisperzibilne tablete koje sadrže bazu escitaloprama | |
| US9815801B2 (en) | Method of refining valsartan comprising more than or equal to 10% D-isomers | |
| JP2011529050A5 (enExample) | ||
| JP2006508646A5 (enExample) | ||
| JP2015535210A5 (enExample) | ||
| CN104703967B (zh) | 氟伏沙明游离碱的精制方法及利用其的高纯度马来酸氟伏沙明的制备方法 |