JP2009138000A5 - - Google Patents

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Publication number
JP2009138000A5
JP2009138000A5 JP2009018865A JP2009018865A JP2009138000A5 JP 2009138000 A5 JP2009138000 A5 JP 2009138000A5 JP 2009018865 A JP2009018865 A JP 2009018865A JP 2009018865 A JP2009018865 A JP 2009018865A JP 2009138000 A5 JP2009138000 A5 JP 2009138000A5
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JP
Japan
Prior art keywords
formula
compound according
converted
compound
under sufficient
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JP2009018865A
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English (en)
Japanese (ja)
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JP5097724B2 (ja
JP2009138000A (ja
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Priority claimed from US08/985,876 external-priority patent/US6262283B1/en
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Publication of JP2009138000A publication Critical patent/JP2009138000A/ja
Publication of JP2009138000A5 publication Critical patent/JP2009138000A5/ja
Application granted granted Critical
Publication of JP5097724B2 publication Critical patent/JP5097724B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP2009018865A 1996-12-06 2009-01-29 アミノステロール、ビタミンｄ類似体および他の化合物の製造に有用な２４−ヒドロキシル化された化合物の立体選択的合成 Expired - Lifetime JP5097724B2 (ja)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US3237896P 1996-12-06 1996-12-06
US60/032,378 1996-12-06
US08/985,876 US6262283B1 (en) 1996-12-06 1997-12-05 Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds
US08/985,876 1997-12-05

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP52401298A Division JP4441769B2 (ja) 1996-12-06 1997-12-08 アミノステロール、ビタミンｄ類似体および他の化合物の製造に有用な２４−ヒドロキシル化された化合物の立体選択的合成

Publications (3)

Publication Number Publication Date
JP2009138000A JP2009138000A (ja) 2009-06-25
JP2009138000A5 true JP2009138000A5 (enExample) 2009-11-12
JP5097724B2 JP5097724B2 (ja) 2012-12-12

Family

ID=26708341

Family Applications (2)

Application Number Title Priority Date Filing Date
JP52401298A Expired - Lifetime JP4441769B2 (ja) 1996-12-06 1997-12-08 アミノステロール、ビタミンｄ類似体および他の化合物の製造に有用な２４−ヒドロキシル化された化合物の立体選択的合成
JP2009018865A Expired - Lifetime JP5097724B2 (ja) 1996-12-06 2009-01-29 アミノステロール、ビタミンｄ類似体および他の化合物の製造に有用な２４−ヒドロキシル化された化合物の立体選択的合成

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP52401298A Expired - Lifetime JP4441769B2 (ja) 1996-12-06 1997-12-08 アミノステロール、ビタミンｄ類似体および他の化合物の製造に有用な２４−ヒドロキシル化された化合物の立体選択的合成

Country Status (7)

Country Link
US (2) US6262283B1 (enExample)
EP (1) EP0942918A2 (enExample)
JP (2) JP4441769B2 (enExample)
AU (1) AU746559B2 (enExample)
CA (1) CA2272721C (enExample)
ES (1) ES2486840T3 (enExample)
WO (1) WO1998024800A2 (enExample)

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US8242294B2 (en) 2007-06-19 2012-08-14 Kythera Biopharmaceuticals, Inc. Synthetic bile acid compositions and methods
US20080318870A1 (en) 2007-06-19 2008-12-25 Kythera Biopharmaceuticals, Inc. Synthetic bile acid compositions and methods
JOP20180077A1 (ar) 2007-06-19 2019-01-30 Kythera Biopharmaceuticals Inc تركيبات وطرق لحمض صفراوي تخليقي
EP3293195A1 (en) * 2007-09-06 2018-03-14 OHR Pharmaceutical, Inc. Compounds for use in treating diabetes
KR100876857B1 (ko) * 2008-02-15 2008-12-31 경북대학교 산학협력단 7-플루오로-3-아미노스테로이드 유도체 또는 이의약학적으로 허용가능한 염, 이의 제조방법 및 이를유효성분으로 함유하는 항균용 약학적 조성물
BR112013003216A2 (pt) 2010-08-12 2016-05-17 Kythera Biopharmaceuticals Inc composições sintéticas de ácido biliar e métodos
AU2011292160B2 (en) 2010-08-17 2015-09-03 Ohr Pharmaceutical, Inc. Ophthalmic formulations of squalamine
WO2012047495A2 (en) * 2010-09-27 2012-04-12 Kythera Biopharmaceuticals, Inc. Methods for preparing synthetic bile acids and compositions comprising the same
EP4469466A1 (en) * 2022-01-25 2024-12-04 Enterin, Inc. C25 r and s isomers of aminosterols and methods of making and using the same
CN116836214B (zh) * 2022-03-25 2024-07-09 苏州恩泰新材料科技有限公司 一种7-酮石胆酸中间体的合成方法和应用

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