JP2009120598A5 - - Google Patents

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Publication number
JP2009120598A5
JP2009120598A5 JP2008273676A JP2008273676A JP2009120598A5 JP 2009120598 A5 JP2009120598 A5 JP 2009120598A5 JP 2008273676 A JP2008273676 A JP 2008273676A JP 2008273676 A JP2008273676 A JP 2008273676A JP 2009120598 A5 JP2009120598 A5 JP 2009120598A5
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JP
Japan
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group
pharmaceutically acceptable
solvate
acceptable salt
compound according
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JP2008273676A
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English (en)
Japanese (ja)
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JP4568779B2 (ja
JP2009120598A (ja
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Priority to JP2008273676A priority Critical patent/JP4568779B2/ja
Priority claimed from JP2008273676A external-priority patent/JP4568779B2/ja
Publication of JP2009120598A publication Critical patent/JP2009120598A/ja
Publication of JP2009120598A5 publication Critical patent/JP2009120598A5/ja
Application granted granted Critical
Publication of JP4568779B2 publication Critical patent/JP4568779B2/ja
Expired - Fee Related legal-status Critical Current
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JP2008273676A 2007-10-26 2008-10-24 スピロ環化合物及びその医薬用途 Expired - Fee Related JP4568779B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2008273676A JP4568779B2 (ja) 2007-10-26 2008-10-24 スピロ環化合物及びその医薬用途

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007279697 2007-10-26
JP2008273676A JP4568779B2 (ja) 2007-10-26 2008-10-24 スピロ環化合物及びその医薬用途

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2010165678A Division JP2010270137A (ja) 2007-10-26 2010-07-23 スピロ環化合物及びその医薬用途

Publications (3)

Publication Number Publication Date
JP2009120598A JP2009120598A (ja) 2009-06-04
JP2009120598A5 true JP2009120598A5 (enExample) 2010-04-22
JP4568779B2 JP4568779B2 (ja) 2010-10-27

Family

ID=40579581

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2008273676A Expired - Fee Related JP4568779B2 (ja) 2007-10-26 2008-10-24 スピロ環化合物及びその医薬用途
JP2010165678A Pending JP2010270137A (ja) 2007-10-26 2010-07-23 スピロ環化合物及びその医薬用途
JP2014158380A Pending JP2014221829A (ja) 2007-10-26 2014-08-04 スピロ環化合物及びその医薬用途
JP2016001396A Ceased JP2016102130A (ja) 2007-10-26 2016-01-06 スピロ環化合物及びその医薬用途
JP2017049246A Pending JP2017132787A (ja) 2007-10-26 2017-03-14 スピロ環化合物及びその医薬用途

Family Applications After (4)

Application Number Title Priority Date Filing Date
JP2010165678A Pending JP2010270137A (ja) 2007-10-26 2010-07-23 スピロ環化合物及びその医薬用途
JP2014158380A Pending JP2014221829A (ja) 2007-10-26 2014-08-04 スピロ環化合物及びその医薬用途
JP2016001396A Ceased JP2016102130A (ja) 2007-10-26 2016-01-06 スピロ環化合物及びその医薬用途
JP2017049246A Pending JP2017132787A (ja) 2007-10-26 2017-03-14 スピロ環化合物及びその医薬用途

Country Status (29)

Country Link
US (3) US8299296B2 (enExample)
EP (3) EP2202216B1 (enExample)
JP (5) JP4568779B2 (enExample)
KR (1) KR101565622B1 (enExample)
CN (1) CN101835737B (enExample)
AR (1) AR071055A1 (enExample)
AU (1) AU2008314933B2 (enExample)
BR (1) BRPI0818687A2 (enExample)
CA (1) CA2704013C (enExample)
CL (1) CL2008003153A1 (enExample)
CO (1) CO6321230A2 (enExample)
CY (1) CY1113352T1 (enExample)
DK (1) DK2202216T3 (enExample)
ES (1) ES2386596T3 (enExample)
HR (1) HRP20120696T1 (enExample)
IL (1) IL205283A (enExample)
ME (1) ME02338B (enExample)
MX (1) MX2010004435A (enExample)
MY (1) MY148469A (enExample)
NZ (1) NZ584161A (enExample)
PE (1) PE20091014A1 (enExample)
PL (1) PL2202216T3 (enExample)
PT (1) PT2202216E (enExample)
RS (1) RS52474B (enExample)
RU (1) RU2490250C2 (enExample)
SI (1) SI2202216T1 (enExample)
TW (1) TWI421070B (enExample)
WO (1) WO2009054479A1 (enExample)
ZA (1) ZA201002305B (enExample)

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AR078948A1 (es) * 2009-11-30 2011-12-14 Lilly Co Eli Compuestos de espiropiperidina, composicion farmaceutica que lo comprenden y su uso para preparar un medicamento util para tratar la diabetes
US8476287B2 (en) 2009-12-25 2013-07-02 Mochida Pharmaceutical Co., Ltd. 3-hydroxy-5-arylisothiazole derivative
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
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TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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CA2834465A1 (en) 2011-04-28 2012-11-01 Mochida Pharmaceutical Co., Ltd. Cyclic amide derivative
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
WO2013045413A1 (en) 2011-09-27 2013-04-04 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2875020B1 (en) 2012-07-19 2017-09-06 Boehringer Ingelheim International GmbH Process for the preparation of a fumaric acid salt of 9-[4-(3-chloro-2-fluoro-phenylamino)-7-methoxy- chinazolin-6-yloxy]-1,4-diaza-spiro[5.5]undecan-5-one
WO2014064215A1 (en) 2012-10-24 2014-05-01 INSERM (Institut National de la Santé et de la Recherche Médicale) TPL2 KINASE INHIBITORS FOR PREVENTING OR TREATING DIABETES AND FOR PROMOTING β-CELL SURVIVAL
TWI692469B (zh) 2012-11-09 2020-05-01 南韓商Ｌｇ化學股份有限公司 Ｇｐｒ４０受體促效劑，製造該促效劑的方法以及含有該促效劑作爲活性劑的醫藥組成物
PT2920165T (pt) 2012-11-16 2016-12-20 Bristol Myers Squibb Co Moduladores de diidropirazol gpr40
KR101569522B1 (ko) 2013-04-18 2015-11-17 현대약품 주식회사 신규한 3-(4-(벤질옥시)페닐)헥스-4-이노익 산 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 대사성 질환의 예방 또는 치료용 약학적 조성물
US9957219B2 (en) 2013-12-04 2018-05-01 Merck Sharp & Dohme Corp. Antidiabetic bicyclic compounds
EP3102198B1 (en) 2014-02-06 2020-08-26 Merck Sharp & Dohme Corp. Antidiabetic compounds
US10227360B2 (en) 2014-02-19 2019-03-12 Piramal Enterprises Limited Compounds for use as GPR120 agonists
US10273230B2 (en) 2014-07-25 2019-04-30 Piramal Enterprises Limited Substituted phenyl alkanoic acid compounds as GPR120 agonists and uses thereof
WO2016038540A1 (en) 2014-09-11 2016-03-17 Piramal Enterprises Limited Fused heterocyclic compounds as gpr120 agonists
ES2805743T3 (es) 2015-03-24 2021-02-15 Inst Nat Sante Rech Med Método y composición farmacéutica para uso en el tratamiento de la diabetes
JPWO2018181847A1 (ja) 2017-03-31 2020-03-05 武田薬品工業株式会社 芳香環化合物
WO2019160882A1 (en) 2018-02-13 2019-08-22 Gilead Sciences, Inc. Pd-1/pd-l1 inhibitors
WO2019204609A1 (en) 2018-04-19 2019-10-24 Gilead Sciences, Inc. Pd-1/pd-l1 inhibitors
BR112020026746A2 (pt) 2018-07-13 2021-03-30 Gilead Sciences, Inc. Composto, composição farmacêutica, métodos para inibir pd-1, pd-l1 e/ou a interação de pd-1/pd-l1 e para tratar câncer, e, kit para tratar ou prevenir câncer ou uma doença ou condição.
CN112955435B (zh) 2018-10-24 2024-09-06 吉利德科学公司 Pd-1/pd-l1抑制剂
JP2022552655A (ja) 2019-10-07 2022-12-19 キャリーオペ，インク． Ｇｐｒ１１９アゴニスト
PH12022552277A1 (en) 2020-02-28 2024-03-04 Kallyope Inc Gpr40 agonists
JP2023526625A (ja) 2020-05-19 2023-06-22 キャリーオペ，インク． Ａｍｐｋアクチベーター
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CN115181023B (zh) * 2022-05-17 2023-07-28 东华理工大学 螺环活性增塑剂及其制备方法
WO2025037230A1 (en) * 2023-08-11 2025-02-20 Life Code Limited Compositions, agents and preparations for promoting hair growth and/or mitigating hair loss

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