JP2008514621A - 20−シクロアルキル,26,27−アルキル/ハロアルキル−ビタミンd3化合物及びその使用方法 - Google Patents

20−シクロアルキル,26,27−アルキル/ハロアルキル−ビタミンd3化合物及びその使用方法 Download PDF

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JP2008514621A
JP2008514621A JP2007533665A JP2007533665A JP2008514621A JP 2008514621 A JP2008514621 A JP 2008514621A JP 2007533665 A JP2007533665 A JP 2007533665A JP 2007533665 A JP2007533665 A JP 2007533665A JP 2008514621 A JP2008514621 A JP 2008514621A
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compound
disease
vitamin
cyclopropyl
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JP2008514621A5 (enExample
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アール ウスココヴィッチ ミラン
アドリーニ ルシアーノ
ペンナ ジュゼッペ
コッリ エンリコ
スタニスラフ マルチャーク
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ビオクセル エッセ ピ ア
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JP2007533665A 2004-09-24 2005-09-23 20−シクロアルキル,26,27−アルキル/ハロアルキル−ビタミンd3化合物及びその使用方法 Pending JP2008514621A (ja)

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US61273204P 2004-09-24 2004-09-24
PCT/US2005/034213 WO2006036813A2 (en) 2004-09-24 2005-09-23 20-cycloalkyl,26,27-alkyl/haloalkyl vitamin d3 compounds and methods of use thereof

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JP2008514621A5 JP2008514621A5 (enExample) 2008-12-18

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US (1) US20080318911A1 (enExample)
EP (1) EP1797033A4 (enExample)
JP (1) JP2008514621A (enExample)
CN (1) CN101106985A (enExample)
AU (1) AU2005289664A1 (enExample)
CA (1) CA2580962A1 (enExample)
IL (1) IL182145A0 (enExample)
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Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012527424A (ja) * 2009-05-20 2012-11-08 イブリジェニク ソシエテ アノニム イネカルシトールの新しい治療的使用
JP5950413B2 (ja) * 2011-03-02 2016-07-13 学校法人日本大学 パーシャルアゴニスト活性を持つ新規ビタミンd受容体モジュレーター
WO2021029318A1 (ja) * 2019-08-13 2021-02-18 国立大学法人東北大学 免疫チェックポイント阻害剤、免疫チェックポイント関連疾患の治療剤、免疫抑制剤、抗フィブロネクチン抗体又はその誘導体、フィブロネクチンアナログ、フィブロネクチンまたはその部分タンパク質を検出するためのキット、及びフィブロネクチンまたはその部分タンパク質を検出する方法
US11760802B2 (en) 2019-12-19 2023-09-19 Ngm Biopharmaceuticals, Inc. ILT3-binding agents and methods of use thereof

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2588453A1 (en) * 2004-12-02 2006-06-08 Abbott Laboratories Use of a compound that activates a vitamin d receptor for reducing intimal hyperplasia, smooth muscle cell proliferation and restenosis in mammals
US7286295B1 (en) 2005-11-30 2007-10-23 Sandia Corporation Microoptical compound lens
WO2009115398A1 (en) * 2008-03-18 2009-09-24 INSERM (Institut National de la Santé et de la Recherche Médicale) Vitamin d compounds for the treatment of biliary diseases
PT2634171E (pt) * 2010-10-25 2015-09-16 Teijin Pharma Ltd Derivado de 23-ino-vitamina d3
US9370527B2 (en) 2012-12-28 2016-06-21 The Regents Of The University Of Michigan Amelioration of intestinal fibrosis and treatment of Crohn's disease
CN103193695B (zh) * 2013-04-22 2015-08-05 中国药科大学 3-苯基-3-吡咯基戊烷类衍生物及其医药用途
WO2016065042A1 (en) 2014-10-22 2016-04-28 Extend Biosciences, Inc. Therapeutic vitamin d conjugates
US9616109B2 (en) 2014-10-22 2017-04-11 Extend Biosciences, Inc. Insulin vitamin D conjugates
CN113274346A (zh) * 2021-05-25 2021-08-20 满孝勇 一种莫匹罗星软膏的应用
EP4593867A2 (en) 2022-09-30 2025-08-06 Extend Biosciences, Inc. Long-acting parathyroid hormone

Citations (9)

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JPH1045714A (ja) * 1996-05-23 1998-02-17 F Hoffmann La Roche Ag フッ素化ビタミンd3類似体
JP2000500476A (ja) * 1995-11-22 2000-01-18 エフ・ホフマン―ラ ロシュ アーゲー 25―ヒドロキシ―16―エン―26,27―ビスホモ―コレカルシフェロール類
JP2001515881A (ja) * 1997-09-08 2001-09-25 エフ.ホフマン−ラ ロシュ アーゲー 1,3−ジヒドロキシ−20,20−ジアルキル−ビタミンd3類似体
JP2002505668A (ja) * 1997-05-16 2002-02-19 ウィメン アンド インファンツ ホスピタル 環状エーテルビタミンD3化合物、1α(OH)3−エピ−ビタミンD3化合物及びそれらの使用法
JP2003504354A (ja) * 1999-07-12 2003-02-04 エフ.ホフマン−ラ ロシュ アーゲー ビタミンd3アナログ
WO2003027065A1 (en) * 2001-09-21 2003-04-03 F. Hoffmann-La Roche Ag 3-desoxy-vitamin d3 analog esters
JP2007506765A (ja) * 2003-09-24 2007-03-22 ビオクセル エッセ ピ ア 1,3−ジアシル化26,27−アルキル/ハロアルキルビタミンd3化合物及びその使用方法
JP2007506780A (ja) * 2003-09-24 2007-03-22 ビオエクセル エスピーエー 膀胱機能障害の治療方法
JP2007525533A (ja) * 2004-03-01 2007-09-06 ビオエクセル エスピーエー 間質性膀胱炎の治療方法、並びに関連化合物及び組成物

Patent Citations (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000500476A (ja) * 1995-11-22 2000-01-18 エフ・ホフマン―ラ ロシュ アーゲー 25―ヒドロキシ―16―エン―26,27―ビスホモ―コレカルシフェロール類
JPH1045714A (ja) * 1996-05-23 1998-02-17 F Hoffmann La Roche Ag フッ素化ビタミンd3類似体
JP2002505668A (ja) * 1997-05-16 2002-02-19 ウィメン アンド インファンツ ホスピタル 環状エーテルビタミンD3化合物、1α(OH)3−エピ−ビタミンD3化合物及びそれらの使用法
JP2001515881A (ja) * 1997-09-08 2001-09-25 エフ.ホフマン−ラ ロシュ アーゲー 1,3−ジヒドロキシ−20,20−ジアルキル−ビタミンd3類似体
JP2003504354A (ja) * 1999-07-12 2003-02-04 エフ.ホフマン−ラ ロシュ アーゲー ビタミンd3アナログ
WO2003027065A1 (en) * 2001-09-21 2003-04-03 F. Hoffmann-La Roche Ag 3-desoxy-vitamin d3 analog esters
JP2005503434A (ja) * 2001-09-21 2005-02-03 エフ.ホフマン−ラ ロシュ アーゲー 3−デスオキシ−ビタミンd3類似体
JP2007506765A (ja) * 2003-09-24 2007-03-22 ビオクセル エッセ ピ ア 1,3−ジアシル化26,27−アルキル/ハロアルキルビタミンd3化合物及びその使用方法
JP2007506780A (ja) * 2003-09-24 2007-03-22 ビオエクセル エスピーエー 膀胱機能障害の治療方法
JP2007525533A (ja) * 2004-03-01 2007-09-06 ビオエクセル エスピーエー 間質性膀胱炎の治療方法、並びに関連化合物及び組成物

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012527424A (ja) * 2009-05-20 2012-11-08 イブリジェニク ソシエテ アノニム イネカルシトールの新しい治療的使用
JP2016179994A (ja) * 2009-05-20 2016-10-13 イブリジェニク ソシエテ アノニム イネカルシトールの新しい治療的使用
JP5950413B2 (ja) * 2011-03-02 2016-07-13 学校法人日本大学 パーシャルアゴニスト活性を持つ新規ビタミンd受容体モジュレーター
WO2021029318A1 (ja) * 2019-08-13 2021-02-18 国立大学法人東北大学 免疫チェックポイント阻害剤、免疫チェックポイント関連疾患の治療剤、免疫抑制剤、抗フィブロネクチン抗体又はその誘導体、フィブロネクチンアナログ、フィブロネクチンまたはその部分タンパク質を検出するためのキット、及びフィブロネクチンまたはその部分タンパク質を検出する方法
US11760802B2 (en) 2019-12-19 2023-09-19 Ngm Biopharmaceuticals, Inc. ILT3-binding agents and methods of use thereof
US12187796B2 (en) 2019-12-19 2025-01-07 Ngm Biopharmaceuticals, Inc. ILT3-binding agents and methods of use thereof

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IL182145A0 (en) 2007-07-24
ZA200703310B (en) 2008-06-25
CN101106985A (zh) 2008-01-16
EP1797033A2 (en) 2007-06-20
WO2006036813A2 (en) 2006-04-06
CA2580962A1 (en) 2006-04-06
US20080318911A1 (en) 2008-12-25
AU2005289664A1 (en) 2006-04-06
EP1797033A4 (en) 2010-04-28
WO2006036813A3 (en) 2006-09-14

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