CA2580962A1 - 20-cycloalkyl,26,27-alkyl/haloalkyl vitamin d3 compounds and methods of use thereof - Google Patents
20-cycloalkyl,26,27-alkyl/haloalkyl vitamin d3 compounds and methods of use thereof Download PDFInfo
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- CA2580962A1 CA2580962A1 CA002580962A CA2580962A CA2580962A1 CA 2580962 A1 CA2580962 A1 CA 2580962A1 CA 002580962 A CA002580962 A CA 002580962A CA 2580962 A CA2580962 A CA 2580962A CA 2580962 A1 CA2580962 A1 CA 2580962A1
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- compound
- vitamin
- disorder
- cyclopropyl
- cholecalciferol
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/14—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
- A61P5/16—Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4 for decreasing, blocking or antagonising the activity of the thyroid hormones
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Virology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Obesity (AREA)
- Cardiology (AREA)
- Dermatology (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Gastroenterology & Hepatology (AREA)
- Ophthalmology & Optometry (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US61273204P | 2004-09-24 | 2004-09-24 | |
| US60/612,732 | 2004-09-24 | ||
| PCT/US2005/034213 WO2006036813A2 (en) | 2004-09-24 | 2005-09-23 | 20-cycloalkyl,26,27-alkyl/haloalkyl vitamin d3 compounds and methods of use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2580962A1 true CA2580962A1 (en) | 2006-04-06 |
Family
ID=36119461
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002580962A Abandoned CA2580962A1 (en) | 2004-09-24 | 2005-09-23 | 20-cycloalkyl,26,27-alkyl/haloalkyl vitamin d3 compounds and methods of use thereof |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20080318911A1 (enExample) |
| EP (1) | EP1797033A4 (enExample) |
| JP (1) | JP2008514621A (enExample) |
| CN (1) | CN101106985A (enExample) |
| AU (1) | AU2005289664A1 (enExample) |
| CA (1) | CA2580962A1 (enExample) |
| IL (1) | IL182145A0 (enExample) |
| WO (1) | WO2006036813A2 (enExample) |
| ZA (1) | ZA200703310B (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2588453A1 (en) * | 2004-12-02 | 2006-06-08 | Abbott Laboratories | Use of a compound that activates a vitamin d receptor for reducing intimal hyperplasia, smooth muscle cell proliferation and restenosis in mammals |
| US7286295B1 (en) | 2005-11-30 | 2007-10-23 | Sandia Corporation | Microoptical compound lens |
| WO2009115398A1 (en) * | 2008-03-18 | 2009-09-24 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Vitamin d compounds for the treatment of biliary diseases |
| SI2263677T1 (sl) * | 2009-05-20 | 2011-07-29 | Hybrigenics Sa | Nove terapevtske uporabe inecalcitola |
| PT2634171E (pt) * | 2010-10-25 | 2015-09-16 | Teijin Pharma Ltd | Derivado de 23-ino-vitamina d3 |
| WO2012118154A1 (ja) * | 2011-03-02 | 2012-09-07 | 学校法人日本大学 | パーシャルアゴニスト活性を持つ新規ビタミンd受容体モジュレーター |
| US9370527B2 (en) | 2012-12-28 | 2016-06-21 | The Regents Of The University Of Michigan | Amelioration of intestinal fibrosis and treatment of Crohn's disease |
| CN103193695B (zh) * | 2013-04-22 | 2015-08-05 | 中国药科大学 | 3-苯基-3-吡咯基戊烷类衍生物及其医药用途 |
| WO2016065042A1 (en) | 2014-10-22 | 2016-04-28 | Extend Biosciences, Inc. | Therapeutic vitamin d conjugates |
| US9616109B2 (en) | 2014-10-22 | 2017-04-11 | Extend Biosciences, Inc. | Insulin vitamin D conjugates |
| WO2021029318A1 (ja) * | 2019-08-13 | 2021-02-18 | 国立大学法人東北大学 | 免疫チェックポイント阻害剤、免疫チェックポイント関連疾患の治療剤、免疫抑制剤、抗フィブロネクチン抗体又はその誘導体、フィブロネクチンアナログ、フィブロネクチンまたはその部分タンパク質を検出するためのキット、及びフィブロネクチンまたはその部分タンパク質を検出する方法 |
| BR112022011790A2 (pt) | 2019-12-19 | 2022-08-30 | Ngm Biopharmaceuticals Inc | Agentes de ligação a ilt3 e métodos de uso dos mesmos |
| CN113274346A (zh) * | 2021-05-25 | 2021-08-20 | 满孝勇 | 一种莫匹罗星软膏的应用 |
| EP4593867A2 (en) | 2022-09-30 | 2025-08-06 | Extend Biosciences, Inc. | Long-acting parathyroid hormone |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW403735B (en) * | 1995-11-22 | 2000-09-01 | Hoffmann La Roche | 25-hydroxy-16-ene-26, 27-bishomo-cholecalciferol |
| SG70010A1 (en) * | 1996-05-23 | 2000-01-25 | Hoffmann La Roche | Fluorinated vitamin d3 analogs |
| US6100294A (en) * | 1997-05-16 | 2000-08-08 | Women And Infants Hospital | Cyclic ether vitamin D3 compounds, 1α(OH) 3-epi-vitamin D3 compounds and uses thereof |
| DE69814109T2 (de) * | 1997-09-08 | 2004-02-26 | F. Hoffmann-La Roche Ag | 1,3-dihydroxy-20,20-dialkyl-vitamin d3 analoga |
| US6331642B1 (en) * | 1999-07-12 | 2001-12-18 | Hoffmann-La Roche Inc. | Vitamin D3 analogs |
| EP1430026A1 (en) * | 2001-09-21 | 2004-06-23 | F. Hoffmann-La Roche Ag | 3-desoxy-vitamin d3 analog esters |
| BRPI0414701A (pt) * | 2003-09-24 | 2006-11-14 | Bioxell Spa | uso de um composto de vitamina d, método de prevenção ou tratamnento de disfunção de bexiga em um paciente, composto de vitamina d, e, kit |
| US20080064668A1 (en) * | 2003-09-24 | 2008-03-13 | Bioxell S.P.A. | 1,3-Diacylated, 26,27-Alkyl/Haloakyl Vitamin D3 Compounds and Methods of Use Thereof |
| WO2005082375A2 (en) * | 2004-03-01 | 2005-09-09 | Bioxell Spa | Treatment of interstitial cystitis with vitamin d compounds |
-
2005
- 2005-09-23 WO PCT/US2005/034213 patent/WO2006036813A2/en not_active Ceased
- 2005-09-23 CN CNA2005800401650A patent/CN101106985A/zh active Pending
- 2005-09-23 EP EP05801186A patent/EP1797033A4/en not_active Withdrawn
- 2005-09-23 US US11/663,704 patent/US20080318911A1/en not_active Abandoned
- 2005-09-23 CA CA002580962A patent/CA2580962A1/en not_active Abandoned
- 2005-09-23 JP JP2007533665A patent/JP2008514621A/ja active Pending
- 2005-09-23 AU AU2005289664A patent/AU2005289664A1/en not_active Abandoned
-
2007
- 2007-03-22 IL IL182145A patent/IL182145A0/en unknown
- 2007-04-23 ZA ZA200703310A patent/ZA200703310B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL182145A0 (en) | 2007-07-24 |
| ZA200703310B (en) | 2008-06-25 |
| CN101106985A (zh) | 2008-01-16 |
| EP1797033A2 (en) | 2007-06-20 |
| WO2006036813A2 (en) | 2006-04-06 |
| JP2008514621A (ja) | 2008-05-08 |
| US20080318911A1 (en) | 2008-12-25 |
| AU2005289664A1 (en) | 2006-04-06 |
| EP1797033A4 (en) | 2010-04-28 |
| WO2006036813A3 (en) | 2006-09-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |