JP2007530550A5 - - Google Patents

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Publication number
JP2007530550A5
JP2007530550A5 JP2007505054A JP2007505054A JP2007530550A5 JP 2007530550 A5 JP2007530550 A5 JP 2007530550A5 JP 2007505054 A JP2007505054 A JP 2007505054A JP 2007505054 A JP2007505054 A JP 2007505054A JP 2007530550 A5 JP2007530550 A5 JP 2007530550A5
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JP
Japan
Prior art keywords
alkyl
cycloalkyl
aryl
alkenyl
trifluoromethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2007505054A
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English (en)
Japanese (ja)
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JP2007530550A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2005/009301 external-priority patent/WO2005097806A1/en
Publication of JP2007530550A publication Critical patent/JP2007530550A/ja
Publication of JP2007530550A5 publication Critical patent/JP2007530550A5/ja
Pending legal-status Critical Current

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JP2007505054A 2004-03-26 2005-03-17 異脂肪血症を治療するための化合物および方法 Pending JP2007530550A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55713404P 2004-03-26 2004-03-26
US62116204P 2004-10-22 2004-10-22
PCT/US2005/009301 WO2005097806A1 (en) 2004-03-26 2005-03-17 Compounds and methods for treating dyslipidemia

Publications (2)

Publication Number Publication Date
JP2007530550A JP2007530550A (ja) 2007-11-01
JP2007530550A5 true JP2007530550A5 (https=) 2008-04-24

Family

ID=34963426

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2007505054A Pending JP2007530550A (ja) 2004-03-26 2005-03-17 異脂肪血症を治療するための化合物および方法

Country Status (21)

Country Link
US (2) US20070208003A1 (https=)
EP (2) EP1732933B1 (https=)
JP (1) JP2007530550A (https=)
KR (1) KR20070007112A (https=)
AT (2) ATE402180T1 (https=)
AU (1) AU2005230915A1 (https=)
BR (1) BRPI0508966A (https=)
CA (1) CA2557010A1 (https=)
CY (1) CY1110398T1 (https=)
DE (2) DE602005014955D1 (https=)
DK (1) DK1732933T3 (https=)
EA (1) EA200601785A1 (https=)
EC (1) ECSP066886A (https=)
ES (2) ES2326326T3 (https=)
IL (1) IL177962A0 (https=)
MA (1) MA28550B1 (https=)
NO (1) NO20064763L (https=)
PL (1) PL1732933T3 (https=)
PT (1) PT1732933E (https=)
SI (1) SI1732933T1 (https=)
WO (2) WO2005097806A1 (https=)

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US8455522B2 (en) 2009-05-15 2013-06-04 Novartis Ag Benzoxazolone derivatives as aldosterone synthase inhibitors
NZ596302A (en) 2009-05-15 2014-01-31 Novartis Ag Aryl pyridine as aldosterone synthase inhibitors
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US8519134B2 (en) 2009-11-17 2013-08-27 Novartis Ag Aryl-pyridine derivatives as aldosterone synthase inhibitors
JO2967B1 (en) 2009-11-20 2016-03-15 نوفارتس ايه جي Acetic acid derivatives of carbamoyl methyl amino are substituted as new NEP inhibitors
ES2472446T3 (es) 2009-11-30 2014-07-01 Novartis Ag Derivados de imidazol como inhibidores de aldosterona sintasa
CN102858347B (zh) * 2010-02-24 2016-11-02 瑞立普萨公司 用作胆汁酸螯合剂的聚咪唑
CN103025348B (zh) 2010-05-06 2015-09-02 阿尔法科制药有限责任公司 传递类固醇到胆甾醇酯合成组织
US8877815B2 (en) 2010-11-16 2014-11-04 Novartis Ag Substituted carbamoylcycloalkyl acetic acid derivatives as NEP
US8673974B2 (en) 2010-11-16 2014-03-18 Novartis Ag Substituted amino bisphenyl pentanoic acid derivatives as NEP inhibitors
SG10201605304VA (en) 2011-07-08 2016-08-30 Novartis Ag Method of treating atherosclerosis in high triglyceride subjects
EP2744803A2 (en) 2011-08-18 2014-06-25 Dr. Reddy's Laboratories Ltd. Substituted heterocyclic amine compounds as cholestryl ester-transfer protein (cetp) inhibitors
MX352074B (es) 2011-09-27 2017-11-08 Dr Reddys Laboratories Ltd Derivados de 5-bencilaminometil-6-aminopirazolo [3,4-b] piridina como inhibidores de proteina de transferencia de ester de colesterilo (cetp) utiles para el tratamiento de aterosclerosis.
JO3210B1 (ar) 2011-10-28 2018-03-08 Merck Sharp & Dohme مثبط منصهر لبروتين نقل الكوليسترليستير اوكسازوليدينون ثمائي الحلقة
WO2013080999A1 (ja) 2011-11-29 2013-06-06 興和株式会社 ＮＰＣ１Ｌ１及び／又はＬＩＰＧ ｍＲＮＡの発現抑制剤並びに肥満症の予防及び／又は治療剤
UY35144A (es) 2012-11-20 2014-06-30 Novartis Ag Miméticos lineales sintéticos de apelina para el tratamiento de insuficiencia cardiaca
TR201808541T4 (tr) 2013-02-14 2018-07-23 Novartis Ag Nep (nötr endopeptidaz) inhibitörleri olarak ikame edilmiş bisfenil butanoik fosfonik asit türevleri.
KR20160031551A (ko) 2013-07-25 2016-03-22 노파르티스 아게 심부전의 치료를 위한 시클릭 폴리펩티드
HK1218252A1 (zh) 2013-07-25 2017-02-10 Novartis Ag 合成apelin多肽之生物结合物
MA41580A (fr) 2015-01-23 2017-11-29 Novartis Ag Conjugués d'acides gras de l'apeline synthétique présentant une demi-vie améliorée
JOP20190086A1 (ar) 2016-10-21 2019-04-18 Novartis Ag مشتقات نافثيريدينون جديدة واستخدامها في معالجة عدم انتظام ضربات القلب
UY38072A (es) 2018-02-07 2019-10-01 Novartis Ag Compuestos derivados de éster butanoico sustituido con bisfenilo como inhibidores de nep, composiciones y combinaciones de los mismos
AR127698A1 (es) 2021-11-23 2024-02-21 Novartis Ag Derivados de naftiridinona para el tratamiento de una enfermedad o un trastorno
KR20260015867A (ko) 2023-05-24 2026-02-03 노파르티스 아게 질환 또는 장애 치료용 나프티리디논 유도체

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TWI345568B (en) * 2004-04-02 2011-07-21 Mitsubishi Tanabe Pharma Corp Tetrahydronaphthyridine derivatives and a process for preparing the same
EA200700119A1 (ru) * 2004-06-24 2007-10-26 Эли Лилли Энд Компани Соединения и способы лечения дислипидемии

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