JP2006528643A5 - - Google Patents

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JP2006528643A5
JP2006528643A5 JP2006521295A JP2006521295A JP2006528643A5 JP 2006528643 A5 JP2006528643 A5 JP 2006528643A5 JP 2006521295 A JP2006521295 A JP 2006521295A JP 2006521295 A JP2006521295 A JP 2006521295A JP 2006528643 A5 JP2006528643 A5 JP 2006528643A5
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halo
membered
alkyl
alkenyl
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JP2006521295A
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JP4521777B2 (ja
JP2006528643A (ja
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Priority claimed from PCT/US2004/023914 external-priority patent/WO2005009988A1/en
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JP2006521295A 2003-07-24 2004-07-23 疼痛治療または予防に有用な４−ヘテロアリール−テトラヒドロピペリジル化合物 Expired - Fee Related JP4521777B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US48951603P 2003-07-24 2003-07-24
PCT/US2004/023914 WO2005009988A1 (en) 2003-07-24 2004-07-23 Heteroaryl-tetrahydropiperidyl compounds useful for treating or preventing pain

Publications (3)

Publication Number Publication Date
JP2006528643A JP2006528643A (ja) 2006-12-21
JP2006528643A5 true JP2006528643A5 (enExample) 2008-03-06
JP4521777B2 JP4521777B2 (ja) 2010-08-11

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Family Applications (1)

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JP2006521295A Expired - Fee Related JP4521777B2 (ja) 2003-07-24 2004-07-23 疼痛治療または予防に有用な４−ヘテロアリール−テトラヒドロピペリジル化合物

Country Status (28)

Country Link
US (4) US7776861B2 (enExample)
EP (2) EP1648879B1 (enExample)
JP (1) JP4521777B2 (enExample)
KR (2) KR100896499B1 (enExample)
CN (3) CN1856484B (enExample)
AT (2) ATE411988T1 (enExample)
AU (1) AU2004259358B2 (enExample)
BR (1) BRPI0412248B1 (enExample)
CA (1) CA2533515C (enExample)
CY (1) CY1109318T1 (enExample)
DE (2) DE602004017316D1 (enExample)
DK (2) DK1648879T3 (enExample)
EA (1) EA009480B1 (enExample)
EG (1) EG25185A (enExample)
ES (1) ES2327684T3 (enExample)
GE (1) GEP20094675B (enExample)
HR (1) HRP20090442T1 (enExample)
IL (2) IL173344A (enExample)
IS (1) IS2593B (enExample)
MA (1) MA27948A1 (enExample)
MX (1) MXPA06000940A (enExample)
NO (1) NO331675B1 (enExample)
NZ (1) NZ544009A (enExample)
PT (1) PT1867644E (enExample)
SI (1) SI1867644T1 (enExample)
UA (1) UA83855C2 (enExample)
WO (1) WO2005009988A1 (enExample)
ZA (1) ZA200509997B (enExample)

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PL1867644T3 (pl) 2003-07-24 2009-10-30 Euro Celtique Sa Związki heteroarylo-tetrahydropiperydylowe przydatne w leczeniu lub zapobieganiu bólu
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US8759362B2 (en) * 2008-10-24 2014-06-24 Purdue Pharma L.P. Bicycloheteroaryl compounds and their use as TRPV1 ligands
US8703962B2 (en) * 2008-10-24 2014-04-22 Purdue Pharma L.P. Monocyclic compounds and their use as TRPV1 ligands
US8921373B2 (en) 2010-06-22 2014-12-30 Shionogi & Co., Ltd. Compounds having TRPV1 antagonistic activity and uses thereof
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US9394293B2 (en) 2011-08-10 2016-07-19 Purdue Pharma L.P. TRPV1 antagonists including dihydroxy substituent and uses thereof
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WO2017202376A1 (zh) * 2016-05-26 2017-11-30 南京明德新药研发股份有限公司 磺酰胺衍生物
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WO2021144720A1 (en) 2020-01-13 2021-07-22 Intrabio Ltd Treatment of late-onset neurodegenerative diseases in heterozygous npc1 gene mutation carriers
DE102022104759A1 (de) 2022-02-28 2023-08-31 SCi Kontor GmbH Co-Kristall-Screening Verfahren, insbesondere zur Herstellung von Co-Kristallen
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