JP2006517944A - 手術後の悪心嘔吐を治療するパロノセトロンの使用 - Google Patents
手術後の悪心嘔吐を治療するパロノセトロンの使用 Download PDFInfo
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- JP2006517944A JP2006517944A JP2006501881A JP2006501881A JP2006517944A JP 2006517944 A JP2006517944 A JP 2006517944A JP 2006501881 A JP2006501881 A JP 2006501881A JP 2006501881 A JP2006501881 A JP 2006501881A JP 2006517944 A JP2006517944 A JP 2006517944A
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- Prior art keywords
- palonosetron
- pharmaceutically acceptable
- ponv
- acceptable salt
- use according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4748—Quinolines; Isoquinolines forming part of bridged ring systems
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Hospice & Palliative Care (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Otolaryngology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
Applications Claiming Priority (2)
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| PCT/EP2004/001558 WO2004073714A1 (en) | 2003-02-18 | 2004-02-18 | Use of palonosetron treating post-operative nausea and vomiting |
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| JP2006517944A true JP2006517944A (ja) | 2006-08-03 |
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| JP2006501881A Pending JP2006517944A (ja) | 2003-02-18 | 2004-02-18 | 手術後の悪心嘔吐を治療するパロノセトロンの使用 |
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Cited By (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009507933A (ja) * | 2006-10-24 | 2009-02-26 | ヘルシン ヘルスケア ソシエテ アノニム | 改良された安定性と生物学的利用能をもつ塩酸パロノセトロンの投与形態 |
| WO2009139411A1 (ja) | 2008-05-15 | 2009-11-19 | 久光製薬株式会社 | パロノセトロンを含有する経皮吸収製剤 |
| JP2014501273A (ja) * | 2010-12-27 | 2014-01-20 | サムヤン バイオファーマシューティカルズ コーポレイション | 悪心または嘔吐防止用組成物 |
| JP2018024621A (ja) * | 2016-08-12 | 2018-02-15 | 武田テバファーマ株式会社 | パロノセトロン又はその薬学的に許容される塩を含む医薬組成物 |
| JP2018048096A (ja) * | 2016-09-23 | 2018-03-29 | ニプロ株式会社 | 液体製剤、及び、パロノセトロンの安定性を向上する方法 |
| JP2019533700A (ja) * | 2016-11-01 | 2019-11-21 | アカシア ファーマ リミテッドＡｃａｃｉａ Ｐｈａｒｍａ Ｌｉｍｉｔｅｄ | アミスルプリドによる術後嘔吐の治療法 |
| US12005042B2 (en) | 2017-02-10 | 2024-06-11 | Acacia Pharma Ltd. | Rescue treatment of post operative nausea and vomiting |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| JP5690461B2 (ja) * | 2002-11-15 | 2015-03-25 | ヘルシン ヘルスケア ソシエテ アノニム | 化学療法誘導嘔吐を治療するためのパロノセトロン |
| JO2735B1 (en) * | 2003-01-30 | 2013-09-15 | هيلسين هيلث كير أس ايه. | Liquid pharmaceutical formulations of palonosetron |
| US8598219B2 (en) | 2003-01-30 | 2013-12-03 | Helsinn Healthcare Sa | Liquid pharmaceutical formulations of palonosetron |
| US20070196491A1 (en) * | 2006-01-27 | 2007-08-23 | Eurand, Inc. | Drug delivery systems comprising weakly basic drugs and organic acids |
| JP5433236B2 (ja) * | 2006-01-27 | 2014-03-05 | アプタリス ファーマテック，インコーポレイテッド | 弱塩基性選択性セロトニン５−ｈｔ３遮断剤および有機酸を含む薬物送達系 |
| TWI429436B (zh) * | 2007-04-10 | 2014-03-11 | Helsinn Therapeutics Us Inc | 使用生長激素促泌素治療或預防嘔吐之方法 |
| US20090155363A1 (en) * | 2007-12-14 | 2009-06-18 | Todd Maibach | Methods for oral administration of active drugs |
| EP2364138A2 (en) * | 2008-12-08 | 2011-09-14 | Teva Pharmaceutical Industries Ltd. | Palonosetron formulation |
| ES2432618T3 (es) * | 2009-05-20 | 2013-12-04 | Inserm (Institut National De La Santé Et De La Recherche Medicale) | Antagonistas del receptor 5-HT3 de serotonina para usar en el tratamiento o prevención de una patología del oído interno con déficit vestibular |
| EP2432467B1 (en) | 2009-05-20 | 2018-02-21 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Serotonin 5-ht3 receptor antagonists for use in the treatment of lesional vestibular disorders |
| US20110003005A1 (en) * | 2009-07-06 | 2011-01-06 | Gopi Venkatesh | Methods of Treating PDNV and PONV with Extended Release Ondansetron Compositions |
| EP2499137A1 (en) | 2009-11-13 | 2012-09-19 | Helsinn Healthcare S.A. | Palonosetron metabolites |
| EP2722045B1 (en) | 2009-11-18 | 2016-07-06 | Helsinn Healthcare SA | Compositions for treating centrally mediated nausea and vomiting |
| PE20121483A1 (es) | 2009-11-18 | 2012-12-02 | Helsinn Healthcare Sa | Composiciones para tratar nausea y vomito centralmente mediados |
| US10071088B2 (en) | 2012-06-26 | 2018-09-11 | Precondit, Llc | Anti-nausea drug combinations |
| EP3087987A4 (en) | 2013-12-23 | 2017-08-02 | Samyang Biopharmaceuticals Corporation | Pharmaceutical composition containing palonosetron |
| HRP20240453T1 (hr) | 2016-04-14 | 2024-06-21 | Sensorion | (+)-azasetron za uporabu u liječenju poremećaja uha |
| KR101802183B1 (ko) * | 2016-11-16 | 2017-11-28 | 주식회사 유영제약 | 팔로노세트론을 활성성분으로 함유하는 약제학적 조성물 |
| US11433021B2 (en) | 2018-01-12 | 2022-09-06 | Orion Corporation | Palonosetron for the treatment or prevention of nausea and vomiting |
| CN108703960A (zh) * | 2018-07-25 | 2018-10-26 | 无锡鑫连鑫生物医药科技有限公司 | 一种帕洛诺司琼缓释微球及其制备方法和使用方法 |
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| JP2006516583A (ja) * | 2003-01-30 | 2006-07-06 | ヘルシン ヘルスケア ソシエテ アノニム | パロノセトロン液状医薬製剤 |
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-
2004
- 2004-02-17 TW TW093103716A patent/TWI355936B/zh not_active IP Right Cessation
- 2004-02-17 MY MYPI20040515A patent/MY143789A/en unknown
- 2004-02-18 MX MXPA05008757A patent/MXPA05008757A/es active IP Right Grant
- 2004-02-18 PL PL378122A patent/PL378122A1/pl not_active Application Discontinuation
- 2004-02-18 BR BRPI0407549-8A patent/BRPI0407549A/pt not_active Application Discontinuation
- 2004-02-18 EP EP04712041A patent/EP1596862B1/en not_active Revoked
- 2004-02-18 NZ NZ541862A patent/NZ541862A/en not_active IP Right Cessation
- 2004-02-18 UA UAA200508834A patent/UA96254C2/uk unknown
- 2004-02-18 UY UY28193A patent/UY28193A1/es not_active Application Discontinuation
- 2004-02-18 GE GEAP20048984A patent/GEP20104908B/en unknown
- 2004-02-18 CA CA002515946A patent/CA2515946C/en not_active Expired - Fee Related
- 2004-02-18 KR KR1020057014589A patent/KR101113087B1/ko not_active Ceased
- 2004-02-18 AU AU2004212704A patent/AU2004212704B2/en not_active Expired
- 2004-02-18 DK DK04712041.5T patent/DK1596862T3/da active
- 2004-02-18 WO PCT/EP2004/001558 patent/WO2004073714A1/en not_active Ceased
- 2004-02-18 ES ES04712041T patent/ES2357769T3/es not_active Expired - Lifetime
- 2004-02-18 EP EP10177400A patent/EP2258367A3/en not_active Withdrawn
- 2004-02-18 SI SI200431601T patent/SI1596862T1/sl unknown
- 2004-02-18 CN CNA2004800045134A patent/CN1750822A/zh active Pending
- 2004-02-18 PT PT04712041T patent/PT1596862E/pt unknown
- 2004-02-18 EA EA200501318A patent/EA013836B1/ru not_active IP Right Cessation
- 2004-02-18 AT AT04712041T patent/ATE490774T1/de active
- 2004-02-18 HR HR20050709A patent/HRP20050709A2/xx not_active Application Discontinuation
- 2004-02-18 JP JP2006501881A patent/JP2006517944A/ja active Pending
- 2004-02-18 DE DE602004030424T patent/DE602004030424D1/de not_active Expired - Lifetime
-
2005
- 2005-08-10 US US11/201,035 patent/US20060074101A1/en not_active Abandoned
- 2005-08-15 IS IS7983A patent/IS7983A/is unknown
- 2005-08-17 CU CU20050158A patent/CU23587B7/es active IP Right Grant
- 2005-08-17 ZA ZA200506580A patent/ZA200506580B/en unknown
- 2005-08-18 EC EC2005005970A patent/ECSP055970A/es unknown
- 2005-09-16 NO NO20054296A patent/NO20054296L/no unknown
-
2011
- 2011-03-04 CY CY20111100257T patent/CY1111312T1/el unknown
Patent Citations (3)
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| JPH03176486A (ja) * | 1989-11-28 | 1991-07-31 | Syntex Usa Inc | 新規三環式化合物 |
| JP2006508977A (ja) * | 2002-11-15 | 2006-03-16 | ヘルシン ヘルスケア ソシエテ アノニム | 化学療法誘導嘔吐を治療するためのパロノセトロン |
| JP2006516583A (ja) * | 2003-01-30 | 2006-07-06 | ヘルシン ヘルスケア ソシエテ アノニム | パロノセトロン液状医薬製剤 |
Cited By (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2009507933A (ja) * | 2006-10-24 | 2009-02-26 | ヘルシン ヘルスケア ソシエテ アノニム | 改良された安定性と生物学的利用能をもつ塩酸パロノセトロンの投与形態 |
| WO2009139411A1 (ja) | 2008-05-15 | 2009-11-19 | 久光製薬株式会社 | パロノセトロンを含有する経皮吸収製剤 |
| JP2014501273A (ja) * | 2010-12-27 | 2014-01-20 | サムヤン バイオファーマシューティカルズ コーポレイション | 悪心または嘔吐防止用組成物 |
| JP2018024621A (ja) * | 2016-08-12 | 2018-02-15 | 武田テバファーマ株式会社 | パロノセトロン又はその薬学的に許容される塩を含む医薬組成物 |
| JP2018048096A (ja) * | 2016-09-23 | 2018-03-29 | ニプロ株式会社 | 液体製剤、及び、パロノセトロンの安定性を向上する方法 |
| JP2019533700A (ja) * | 2016-11-01 | 2019-11-21 | アカシア ファーマ リミテッドＡｃａｃｉａ Ｐｈａｒｍａ Ｌｉｍｉｔｅｄ | アミスルプリドによる術後嘔吐の治療法 |
| JP2023058654A (ja) * | 2016-11-01 | 2023-04-25 | アカシア ファーマ リミテッド | アミスルプリドによる術後嘔吐の治療法 |
| US12005042B2 (en) | 2017-02-10 | 2024-06-11 | Acacia Pharma Ltd. | Rescue treatment of post operative nausea and vomiting |
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