JP2005528459A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2005528459A5 JP2005528459A5 JP2004511291A JP2004511291A JP2005528459A5 JP 2005528459 A5 JP2005528459 A5 JP 2005528459A5 JP 2004511291 A JP2004511291 A JP 2004511291A JP 2004511291 A JP2004511291 A JP 2004511291A JP 2005528459 A5 JP2005528459 A5 JP 2005528459A5
- Authority
- JP
- Japan
- Prior art keywords
- amino
- het
- methyl
- independently
- unsubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02012590A EP1369420A1 (en) | 2002-06-06 | 2002-06-06 | Inhibitors of the GPib - vWF interaction |
| PCT/EP2003/005955 WO2003104221A1 (en) | 2002-06-06 | 2003-06-06 | Inhibitors of the gpib -vwf interaction, their preparation and use |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2005528459A JP2005528459A (ja) | 2005-09-22 |
| JP2005528459A5 true JP2005528459A5 (enExample) | 2006-04-06 |
| JP4455326B2 JP4455326B2 (ja) | 2010-04-21 |
Family
ID=29433122
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004511291A Expired - Fee Related JP4455326B2 (ja) | 2002-06-06 | 2003-06-06 | ＧＰＩｂ−ｖＷＦ相互作用の阻害薬、それらの製造および使用 |
Country Status (9)
| Country | Link |
|---|---|
| EP (2) | EP1369420A1 (enExample) |
| JP (1) | JP4455326B2 (enExample) |
| AT (1) | ATE353082T1 (enExample) |
| AU (1) | AU2003274686A1 (enExample) |
| BR (1) | BR0311826A (enExample) |
| CA (1) | CA2488193A1 (enExample) |
| DE (1) | DE60311578T2 (enExample) |
| MX (1) | MXPA04011408A (enExample) |
| WO (1) | WO2003104221A1 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR043507A1 (es) * | 2003-03-14 | 2005-08-03 | Lundbeck & Co As H | Derivados de anilina sustituidos y composiciones farmaceuticas |
| BRPI0408205A (pt) * | 2003-03-14 | 2006-02-14 | Lundbeck & Co As H | derivado de anilina substituìdo, composição farmacêutica, e, uso de uma composição farmacêutica |
| EP1669348A4 (en) | 2003-09-30 | 2009-03-11 | Eisai R&D Man Co Ltd | NEW ANTIPILIC AGENT CONTAINING A HETEROCYCLIC COMPOUND |
| WO2006016548A1 (ja) * | 2004-08-09 | 2006-02-16 | Eisai R & D Management Co., Ltd. | ヘテロ環化合物を含有する新規な抗マラリア剤 |
| WO2006106711A1 (ja) | 2005-03-30 | 2006-10-12 | Eisai R & D Management Co., Ltd. | ピリジン誘導体を含有する抗真菌剤 |
| TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
| WO2008035726A1 (en) | 2006-09-21 | 2008-03-27 | Eisai R & D Management Co., Ltd. | Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same |
| TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
| CA2685194A1 (en) | 2007-04-27 | 2008-11-13 | Eisai R&D Management Co., Ltd. | Heterocycle-substituted pyridine derivatives salt or crystal thereof |
| US8461189B2 (en) | 2007-06-27 | 2013-06-11 | Merck Sharp & Dohme Corp. | Pyridyl derivatives as histone deacetylase inhibitors |
| AU2008269154B2 (en) | 2007-06-27 | 2014-06-12 | Merck Sharp & Dohme Llc | 4-carboxybenzylamino derivatives as histone deacetylase inhibitors |
| US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
| US8188119B2 (en) | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
| AU2011313853A1 (en) * | 2010-10-11 | 2013-05-02 | Auckland Uniservices Limited | Substituted benzamides and their uses |
| SG11201406518XA (en) | 2012-04-12 | 2014-11-27 | Univ Leland Stanford Junior | Substituted benzamides and their uses |
| JP2023078557A (ja) * | 2021-11-26 | 2023-06-07 | 学校法人東海大学 | フォンヴィルブランド因子と血小板との結合を阻害するための医薬組成物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW301607B (enExample) * | 1993-03-09 | 1997-04-01 | Takeda Pharm Industry Co Ltd | |
| US5919776A (en) * | 1996-12-20 | 1999-07-06 | Merck & Co., Inc. | Substituted aminoquinolines as modulators of chemokine receptor activity |
| AU5812498A (en) * | 1996-12-20 | 1998-07-17 | Merck & Co., Inc. | Substituted aminoquinolines as modulators of chemokine receptor activity |
-
2002
- 2002-06-06 EP EP02012590A patent/EP1369420A1/en not_active Withdrawn
-
2003
- 2003-06-06 BR BR0311826-6A patent/BR0311826A/pt not_active IP Right Cessation
- 2003-06-06 MX MXPA04011408A patent/MXPA04011408A/es unknown
- 2003-06-06 JP JP2004511291A patent/JP4455326B2/ja not_active Expired - Fee Related
- 2003-06-06 AT AT03740199T patent/ATE353082T1/de not_active IP Right Cessation
- 2003-06-06 DE DE60311578T patent/DE60311578T2/de not_active Expired - Lifetime
- 2003-06-06 WO PCT/EP2003/005955 patent/WO2003104221A1/en not_active Ceased
- 2003-06-06 CA CA002488193A patent/CA2488193A1/en not_active Abandoned
- 2003-06-06 AU AU2003274686A patent/AU2003274686A1/en not_active Abandoned
- 2003-06-06 EP EP03740199A patent/EP1509516B1/en not_active Expired - Lifetime
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DE60217674T2 (de) | Derivate heterocyclischer verbindungen und arzneimittel | |
| JP2021119196A5 (enExample) | ||
| JP6513078B2 (ja) | 新規ヒストンデアセチラーゼインヒビター | |
| US9687479B2 (en) | Multisubstituted aromatic compounds as serine protease inhibitors | |
| RU2578602C2 (ru) | Способ получения 5-хлор-n-(5s)-2-оксо-3-[4-(3-оксо-морфолинил)-фенил]-1,3-оксазолидин-5-ил}-метил)-2-тиофенкарбоксамида в модификации ii (варианты) | |
| JP4594925B2 (ja) | 増殖亢進性、血管新生性及び炎症性疾患の治療に有用な２−オキソ−１，３，５−パーヒドロトリアザピン誘導体 | |
| JP2013121919A (ja) | 血漿カリクレイン阻害剤 | |
| JP2000504682A (ja) | 抗血栓性／抗凝血性効果を有するアミノ複素環式化合物 | |
| JP2000508334A (ja) | ピラジノン系トロンビン阻害薬 | |
| IL166855A (en) | Annals of compressed pyrimidine with azaleas that inhibit pi3k activity and drugs containing them. | |
| JP2001514227A (ja) | ピラジノン系トロンビン阻害薬 | |
| CN112204023A (zh) | 因子XIIa抑制剂 | |
| JP2010150275A (ja) | ピラジノントロンビン阻害剤 | |
| JP2017532358A (ja) | ポリヘテロアリールヒストンデアセチラーゼインヒビターおよび治療におけるその使用 | |
| JP2009543844A (ja) | 直接トロンビン阻害剤の新しい小児適応症 | |
| KR20160139067A (ko) | 테트라히드로이소퀴놀린-1-온 유도체 또는 그의 염 | |
| JP5178712B2 (ja) | アリール置換ヘテロ環およびそれらの使用 | |
| KR20080040692A (ko) | 단백질 키나제 억제제로서의 2-아미노아릴 피리딘 | |
| AU2014238478B2 (en) | Halogenopyrazoles as inhibitors of thrombin | |
| US6326386B1 (en) | Benzamide derivatives as thrombin inhibitors | |
| JPWO2004094407A1 (ja) | ５員複素環誘導体 | |
| JP2008517954A (ja) | 抗血小板剤としての置換ピリドキシン | |
| JP2005506970A (ja) | 置換イソインドール類およびそれらの使用 | |
| WO2001092234A1 (en) | Pyrazinone thrombin inhibitors | |
| JP3237107B2 (ja) | ブタジエン誘導体及びその製法 |