JP2005526808A5 - - Google Patents
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- Publication number
- JP2005526808A5 JP2005526808A5 JP2003579830A JP2003579830A JP2005526808A5 JP 2005526808 A5 JP2005526808 A5 JP 2005526808A5 JP 2003579830 A JP2003579830 A JP 2003579830A JP 2003579830 A JP2003579830 A JP 2003579830A JP 2005526808 A5 JP2005526808 A5 JP 2005526808A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- rhinitis
- asthma
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 150000001875 compounds Chemical class 0.000 claims 14
- 208000006673 asthma Diseases 0.000 claims 3
- 230000004968 inflammatory condition Effects 0.000 claims 3
- 238000000034 method Methods 0.000 claims 3
- 206010039083 rhinitis Diseases 0.000 claims 3
- -1 benzenesulfonate (besylate) anion Chemical class 0.000 claims 2
- 239000003814 drug Substances 0.000 claims 2
- 125000000217 alkyl group Chemical group 0.000 claims 1
- FKBKHPCMPAOJOE-FCQHKQNSSA-N benzenesulfonic acid;4-[[[(2s)-4-[(3,4-dichlorophenyl)methyl]morpholin-2-yl]methylcarbamoylamino]methyl]benzamide;dihydrate Chemical compound O.O.OS(=O)(=O)C1=CC=CC=C1.C1=CC(C(=O)N)=CC=C1CNC(=O)NC[C@@H]1OCCN(CC=2C=C(Cl)C(Cl)=CC=2)C1 FKBKHPCMPAOJOE-FCQHKQNSSA-N 0.000 claims 1
- 239000000969 carrier Substances 0.000 claims 1
- 239000003085 diluting agent Substances 0.000 claims 1
- 238000004519 manufacturing process Methods 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
- 229940124597 therapeutic agent Drugs 0.000 claims 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0207432.6A GB0207432D0 (en) | 2002-03-28 | 2002-03-28 | Novel compounds |
| PCT/EP2003/003345 WO2003082293A1 (en) | 2002-03-28 | 2003-03-27 | Benzenesulphonate salt of a morpholine urea derivative for use as a ccr-3 antagonist in the treatment of inflammatory conditions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005526808A JP2005526808A (ja) | 2005-09-08 |
| JP2005526808A5 true JP2005526808A5 (enExample) | 2006-05-18 |
Family
ID=9933984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003579830A Pending JP2005526808A (ja) | 2002-03-28 | 2003-03-27 | 炎症状態の治療においてccr−3拮抗薬として使用するためのモルホリン尿素誘導体のベンゼンスルホン酸塩 |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7531651B2 (enExample) |
| EP (1) | EP1487456B1 (enExample) |
| JP (1) | JP2005526808A (enExample) |
| KR (1) | KR20040099375A (enExample) |
| CN (1) | CN1642554A (enExample) |
| AR (1) | AR039179A1 (enExample) |
| AT (1) | ATE317698T1 (enExample) |
| AU (1) | AU2003226761A1 (enExample) |
| BR (1) | BR0308480A (enExample) |
| CA (1) | CA2479912A1 (enExample) |
| DE (1) | DE60303603T2 (enExample) |
| ES (1) | ES2258724T3 (enExample) |
| GB (1) | GB0207432D0 (enExample) |
| IL (1) | IL163847A0 (enExample) |
| IS (1) | IS7432A (enExample) |
| MX (1) | MXPA04009456A (enExample) |
| NO (1) | NO20044323L (enExample) |
| PL (1) | PL372623A1 (enExample) |
| RU (1) | RU2004126948A (enExample) |
| TW (1) | TW200407145A (enExample) |
| WO (1) | WO2003082293A1 (enExample) |
| ZA (1) | ZA200407463B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20140335083A1 (en) * | 2011-12-01 | 2014-11-13 | Glaxo Group Limited | Methods of treatment and prevention of eye diseases |
| FR3022142B1 (fr) | 2014-06-16 | 2019-07-12 | Universite Paul Sabatier - Toulouse Iii | Inhibition de la chimiokine ccl7 ou de son recepteur ccr3 pour le traitement et le diagnostic du cancer de la prostate |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1995031431A1 (en) | 1994-05-18 | 1995-11-23 | Nisshin Flour Milling Co., Ltd. | Novel diaminomethylidene derivative |
| BR9915520A (pt) | 1998-11-20 | 2001-07-17 | Hoffmann La Roche | Antagonistas receptores ccr-3 derivados de pirrolidina |
| IL155092A0 (en) | 2000-09-29 | 2003-10-31 | Glaxo Group Ltd | Compounds useful in the treatment of inflammatory diseases |
-
2002
- 2002-03-28 GB GBGB0207432.6A patent/GB0207432D0/en not_active Ceased
-
2003
- 2003-03-26 TW TW092106768A patent/TW200407145A/zh unknown
- 2003-03-27 AR ARP030101092A patent/AR039179A1/es unknown
- 2003-03-27 ES ES03745298T patent/ES2258724T3/es not_active Expired - Lifetime
- 2003-03-27 AU AU2003226761A patent/AU2003226761A1/en not_active Abandoned
- 2003-03-27 BR BR0308480-9A patent/BR0308480A/pt not_active Application Discontinuation
- 2003-03-27 AT AT03745298T patent/ATE317698T1/de not_active IP Right Cessation
- 2003-03-27 PL PL03372623A patent/PL372623A1/xx not_active Application Discontinuation
- 2003-03-27 RU RU2004126948/04A patent/RU2004126948A/ru not_active Application Discontinuation
- 2003-03-27 KR KR10-2004-7015442A patent/KR20040099375A/ko not_active Withdrawn
- 2003-03-27 CN CNA038073641A patent/CN1642554A/zh active Pending
- 2003-03-27 EP EP03745298A patent/EP1487456B1/en not_active Expired - Lifetime
- 2003-03-27 WO PCT/EP2003/003345 patent/WO2003082293A1/en not_active Ceased
- 2003-03-27 MX MXPA04009456A patent/MXPA04009456A/es unknown
- 2003-03-27 IL IL16384703A patent/IL163847A0/xx unknown
- 2003-03-27 DE DE60303603T patent/DE60303603T2/de not_active Expired - Lifetime
- 2003-03-27 JP JP2003579830A patent/JP2005526808A/ja active Pending
- 2003-03-27 US US10/509,521 patent/US7531651B2/en not_active Expired - Fee Related
- 2003-03-27 CA CA002479912A patent/CA2479912A1/en not_active Abandoned
-
2004
- 2004-08-31 IS IS7432A patent/IS7432A/is unknown
- 2004-09-16 ZA ZA200407463A patent/ZA200407463B/en unknown
- 2004-10-12 NO NO20044323A patent/NO20044323L/no not_active Application Discontinuation
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