JP2005526808A - 炎症状態の治療においてｃｃｒ−３拮抗薬として使用するためのモルホリン尿素誘導体のベンゼンスルホン酸塩 - Google Patents
炎症状態の治療においてｃｃｒ−３拮抗薬として使用するためのモルホリン尿素誘導体のベンゼンスルホン酸塩 Download PDFInfo
- Publication number
- JP2005526808A JP2005526808A JP2003579830A JP2003579830A JP2005526808A JP 2005526808 A JP2005526808 A JP 2005526808A JP 2003579830 A JP2003579830 A JP 2003579830A JP 2003579830 A JP2003579830 A JP 2003579830A JP 2005526808 A JP2005526808 A JP 2005526808A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- mixture
- added
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0207432.6A GB0207432D0 (en) | 2002-03-28 | 2002-03-28 | Novel compounds |
| PCT/EP2003/003345 WO2003082293A1 (en) | 2002-03-28 | 2003-03-27 | Benzenesulphonate salt of a morpholine urea derivative for use as a ccr-3 antagonist in the treatment of inflammatory conditions |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005526808A true JP2005526808A (ja) | 2005-09-08 |
| JP2005526808A5 JP2005526808A5 (enExample) | 2006-05-18 |
Family
ID=9933984
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003579830A Pending JP2005526808A (ja) | 2002-03-28 | 2003-03-27 | 炎症状態の治療においてｃｃｒ−３拮抗薬として使用するためのモルホリン尿素誘導体のベンゼンスルホン酸塩 |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7531651B2 (enExample) |
| EP (1) | EP1487456B1 (enExample) |
| JP (1) | JP2005526808A (enExample) |
| KR (1) | KR20040099375A (enExample) |
| CN (1) | CN1642554A (enExample) |
| AR (1) | AR039179A1 (enExample) |
| AT (1) | ATE317698T1 (enExample) |
| AU (1) | AU2003226761A1 (enExample) |
| BR (1) | BR0308480A (enExample) |
| CA (1) | CA2479912A1 (enExample) |
| DE (1) | DE60303603T2 (enExample) |
| ES (1) | ES2258724T3 (enExample) |
| GB (1) | GB0207432D0 (enExample) |
| IL (1) | IL163847A0 (enExample) |
| IS (1) | IS7432A (enExample) |
| MX (1) | MXPA04009456A (enExample) |
| NO (1) | NO20044323L (enExample) |
| PL (1) | PL372623A1 (enExample) |
| RU (1) | RU2004126948A (enExample) |
| TW (1) | TW200407145A (enExample) |
| WO (1) | WO2003082293A1 (enExample) |
| ZA (1) | ZA200407463B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20140335083A1 (en) * | 2011-12-01 | 2014-11-13 | Glaxo Group Limited | Methods of treatment and prevention of eye diseases |
| FR3022142B1 (fr) | 2014-06-16 | 2019-07-12 | Universite Paul Sabatier - Toulouse Iii | Inhibition de la chimiokine ccl7 ou de son recepteur ccr3 pour le traitement et le diagnostic du cancer de la prostate |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1995031431A1 (en) | 1994-05-18 | 1995-11-23 | Nisshin Flour Milling Co., Ltd. | Novel diaminomethylidene derivative |
| BR9915520A (pt) | 1998-11-20 | 2001-07-17 | Hoffmann La Roche | Antagonistas receptores ccr-3 derivados de pirrolidina |
| IL155092A0 (en) | 2000-09-29 | 2003-10-31 | Glaxo Group Ltd | Compounds useful in the treatment of inflammatory diseases |
-
2002
- 2002-03-28 GB GBGB0207432.6A patent/GB0207432D0/en not_active Ceased
-
2003
- 2003-03-26 TW TW092106768A patent/TW200407145A/zh unknown
- 2003-03-27 AR ARP030101092A patent/AR039179A1/es unknown
- 2003-03-27 ES ES03745298T patent/ES2258724T3/es not_active Expired - Lifetime
- 2003-03-27 AU AU2003226761A patent/AU2003226761A1/en not_active Abandoned
- 2003-03-27 BR BR0308480-9A patent/BR0308480A/pt not_active Application Discontinuation
- 2003-03-27 AT AT03745298T patent/ATE317698T1/de not_active IP Right Cessation
- 2003-03-27 PL PL03372623A patent/PL372623A1/xx not_active Application Discontinuation
- 2003-03-27 RU RU2004126948/04A patent/RU2004126948A/ru not_active Application Discontinuation
- 2003-03-27 KR KR10-2004-7015442A patent/KR20040099375A/ko not_active Withdrawn
- 2003-03-27 CN CNA038073641A patent/CN1642554A/zh active Pending
- 2003-03-27 EP EP03745298A patent/EP1487456B1/en not_active Expired - Lifetime
- 2003-03-27 WO PCT/EP2003/003345 patent/WO2003082293A1/en not_active Ceased
- 2003-03-27 MX MXPA04009456A patent/MXPA04009456A/es unknown
- 2003-03-27 IL IL16384703A patent/IL163847A0/xx unknown
- 2003-03-27 DE DE60303603T patent/DE60303603T2/de not_active Expired - Lifetime
- 2003-03-27 JP JP2003579830A patent/JP2005526808A/ja active Pending
- 2003-03-27 US US10/509,521 patent/US7531651B2/en not_active Expired - Fee Related
- 2003-03-27 CA CA002479912A patent/CA2479912A1/en not_active Abandoned
-
2004
- 2004-08-31 IS IS7432A patent/IS7432A/is unknown
- 2004-09-16 ZA ZA200407463A patent/ZA200407463B/en unknown
- 2004-10-12 NO NO20044323A patent/NO20044323L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2479912A1 (en) | 2003-10-09 |
| IS7432A (is) | 2004-08-31 |
| EP1487456B1 (en) | 2006-02-15 |
| EP1487456A1 (en) | 2004-12-22 |
| GB0207432D0 (en) | 2002-05-08 |
| CN1642554A (zh) | 2005-07-20 |
| TW200407145A (en) | 2004-05-16 |
| ES2258724T3 (es) | 2006-09-01 |
| AU2003226761A1 (en) | 2003-10-13 |
| RU2004126948A (ru) | 2005-07-10 |
| IL163847A0 (en) | 2005-12-18 |
| WO2003082293A1 (en) | 2003-10-09 |
| US20060089497A1 (en) | 2006-04-27 |
| BR0308480A (pt) | 2005-01-18 |
| US7531651B2 (en) | 2009-05-12 |
| PL372623A1 (en) | 2005-07-25 |
| ZA200407463B (en) | 2005-10-12 |
| DE60303603T2 (de) | 2006-10-26 |
| AR039179A1 (es) | 2005-02-09 |
| ATE317698T1 (de) | 2006-03-15 |
| NO20044323L (no) | 2004-10-27 |
| MXPA04009456A (es) | 2005-01-25 |
| DE60303603D1 (de) | 2006-04-20 |
| KR20040099375A (ko) | 2004-11-26 |
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