JP2005509622A - ５’−カルバモイル−２’−メチル−１，１’−ビフェニル−４−カルボキサミド誘導体及びそのｐ３８キナーゼ阻害薬としての使用 - Google Patents

５’−カルバモイル−２’−メチル−１，１’−ビフェニル−４−カルボキサミド誘導体及びそのｐ３８キナーゼ阻害薬としての使用 Download PDF

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JP2005509622A
JP2005509622A JP2003535774A JP2003535774A JP2005509622A JP 2005509622 A JP2005509622 A JP 2005509622A JP 2003535774 A JP2003535774 A JP 2003535774A JP 2003535774 A JP2003535774 A JP 2003535774A JP 2005509622 A JP2005509622 A JP 2005509622A
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methyl
biphenyl
alkyl
mmol
dicarboxamide
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JP2003535774A
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Japanese (ja)
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JP2005509622A5 (OSRAM
Inventor
アンジェル，リチャード，マーティン
アストン，ニコラ，マリー
バムボロー，ポール
バムフォード，マーク，ジェームズ
コッカリル，ジョージ，スチュアート
マーリック，スザンヌ，ジョイ
スミス，キャスリン，ジェーン
ウォルカー，アン，ルイーズ
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Glaxo Group Ltd
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Glaxo Group Ltd
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Publication of JP2005509622A publication Critical patent/JP2005509622A/ja
Publication of JP2005509622A5 publication Critical patent/JP2005509622A5/ja
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JP2007506664A (ja) * 2003-06-20 2007-03-22 グラクソ　グループ　リミテッド マトリックスメタロプロテイナーゼの阻害剤
JP2009508835A (ja) * 2005-09-16 2009-03-05 アロー セラピューティクス リミテッド ビフェニル誘導体及びｃ型肝炎の治療におけるその使用
JP2014525425A (ja) * 2011-08-31 2014-09-29 アマケン エンヴェー 新規のｒｏｃｋキナーゼ阻害剤
JP2017506237A (ja) * 2014-02-19 2017-03-02 ハー・ルンドベック・アクチエゼルスカベット アルツハイマー病治療用のｂａｃｅ１阻害剤としての２−アミノ−３，５，５−トリフルオロ−３，４，５，６−テトラヒドロピリジン
JP2024505646A (ja) * 2021-01-29 2024-02-07 プレイザーセラピューティクス インコーポレイテッド ｐ３８ ＭＡＰキナーゼ阻害剤で抗炎症活性を示す新規な化合物

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BRPI0307351B8 (pt) 2002-02-12 2021-05-25 Smithkline Beecham Corp composto, composição farmacêutica, uso de um composto, e, processo para preparar um composto
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MA40941A (fr) 2014-11-10 2017-09-19 H Lundbeck As 2-amino-5,5-difluoro-6-(fluorométhyl)-6-phényl-3,4,5,6-tétrahydropyridines comme inhibiteurs de bace1
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JP2009508835A (ja) * 2005-09-16 2009-03-05 アロー セラピューティクス リミテッド ビフェニル誘導体及びｃ型肝炎の治療におけるその使用
JP2014525425A (ja) * 2011-08-31 2014-09-29 アマケン エンヴェー 新規のｒｏｃｋキナーゼ阻害剤
JP2017506237A (ja) * 2014-02-19 2017-03-02 ハー・ルンドベック・アクチエゼルスカベット アルツハイマー病治療用のｂａｃｅ１阻害剤としての２−アミノ−３，５，５−トリフルオロ−３，４，５，６−テトラヒドロピリジン
JP2024505646A (ja) * 2021-01-29 2024-02-07 プレイザーセラピューティクス インコーポレイテッド ｐ３８ ＭＡＰキナーゼ阻害剤で抗炎症活性を示す新規な化合物

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