JP2005500363A - 安定化経口懸濁液製剤 - Google Patents

安定化経口懸濁液製剤 Download PDF

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JP2005500363A
JP2005500363A JP2003518483A JP2003518483A JP2005500363A JP 2005500363 A JP2005500363 A JP 2005500363A JP 2003518483 A JP2003518483 A JP 2003518483A JP 2003518483 A JP2003518483 A JP 2003518483A JP 2005500363 A JP2005500363 A JP 2005500363A
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composition
drug
present
polyoxyethylene
amount
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Japanese (ja)
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JP2005500363A5 (enExample
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ル，グァン・ウェイ
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ファルマシア・コーポレーション
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Publication of JP2005500363A publication Critical patent/JP2005500363A/ja
Publication of JP2005500363A5 publication Critical patent/JP2005500363A5/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Dental Preparations (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2003518483A 2001-08-06 2002-08-05 安定化経口懸濁液製剤 Pending JP2005500363A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US31037201P 2001-08-06 2001-08-06
PCT/US2002/024746 WO2003013473A1 (en) 2001-08-06 2002-08-05 Stabilized oral suspension formulation

Publications (2)

Publication Number Publication Date
JP2005500363A true JP2005500363A (ja) 2005-01-06
JP2005500363A5 JP2005500363A5 (enExample) 2005-12-22

Family

ID=23202195

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003518483A Pending JP2005500363A (ja) 2001-08-06 2002-08-05 安定化経口懸濁液製剤

Country Status (33)

Country Link
US (2) US20030108575A1 (enExample)
EP (1) EP1414409B1 (enExample)
JP (1) JP2005500363A (enExample)
KR (1) KR20040025740A (enExample)
CN (1) CN1287768C (enExample)
AP (1) AP1817A (enExample)
AT (1) ATE353627T1 (enExample)
BR (1) BR0211736A (enExample)
CA (1) CA2454173A1 (enExample)
CO (1) CO5560559A2 (enExample)
CY (1) CY1106548T1 (enExample)
DE (1) DE60218175T2 (enExample)
DK (1) DK1414409T3 (enExample)
EA (1) EA007901B1 (enExample)
EC (1) ECSP044974A (enExample)
ES (1) ES2280560T3 (enExample)
GE (1) GEP20074027B (enExample)
HR (1) HRP20040118A2 (enExample)
IL (1) IL159551A0 (enExample)
IS (1) IS7126A (enExample)
MA (1) MA27054A1 (enExample)
MX (1) MXPA04001109A (enExample)
MY (1) MY135119A (enExample)
NZ (1) NZ530844A (enExample)
OA (1) OA12646A (enExample)
PL (1) PL366382A1 (enExample)
PT (1) PT1414409E (enExample)
SI (1) SI1414409T1 (enExample)
TN (1) TNSN04023A1 (enExample)
UA (1) UA80682C2 (enExample)
WO (1) WO2003013473A1 (enExample)
YU (1) YU7404A (enExample)
ZA (1) ZA200400639B (enExample)

Cited By (3)

* Cited by examiner, † Cited by third party
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JP2014503512A (ja) * 2010-12-10 2014-02-13 ビオプロジェ エンケファリナーゼ阻害剤の新規投与形態
JP2018516279A (ja) * 2015-05-29 2018-06-21 コーダドース・インコーポレーテッド 経口投与用のセレコキシブの液状配合物
JP2019531309A (ja) * 2016-10-19 2019-10-31 サインパス ファルマ, インク.Signpath Pharma, Inc. チャネル病を引き起こす薬物に対するｄｍｐｃ、ｄｍｐｇ、ｄｍｐｃ／ｄｍｐｇ、ｌｙｓｏｐｇ及びｌｙｓｏｐｃの防御効果

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GB9720061D0 (en) 1997-09-19 1997-11-19 Crosfield Joseph & Sons Metal compounds as phosphate binders
US9101540B2 (en) 2002-04-12 2015-08-11 Alkermes Pharma Ireland Limited Nanoparticulate megestrol formulations
US20040105889A1 (en) * 2002-12-03 2004-06-03 Elan Pharma International Limited Low viscosity liquid dosage forms
US20050036956A1 (en) * 2003-08-15 2005-02-17 Lin Fei Non-aqueous liquid tooth whitening composition
TR200301552A1 (tr) * 2003-09-18 2005-10-21 Nobel İlaç Sanayi̇ Ve Ti̇caret A. Ş. Rofekoksib' in yeni oral farmakolojik formülasyonları.
US20050266031A1 (en) * 2004-05-25 2005-12-01 Jay Dickerson Pharmaceutical suspension composition
US8318210B2 (en) 2005-02-28 2012-11-27 Neos Therapeutics, Lp Compositions and methods of making sustained release liquid formulations
US8653145B2 (en) * 2005-09-22 2014-02-18 Eaton Scientific Systems, Ltd. Method for alleviating climacteric symptoms
MY157620A (en) 2006-01-31 2016-06-30 Cytochroma Dev Inc A granular material of a solid water-soluble mixed metal compound capable of binding phosphate
PL2018153T3 (pl) * 2006-04-26 2012-09-28 Rosemont Pharmaceuticals Ltd Ciekłe kompozycje doustne
CN100434072C (zh) * 2006-06-19 2008-11-19 西安交通大学 具有抗炎性作用及改善血液流变性和抑制血栓形成的药物
GB0714670D0 (en) 2007-07-27 2007-09-05 Ineos Healthcare Ltd Use
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WO2011107855A2 (en) 2010-03-04 2011-09-09 Torrent Pharmaceuticals Limited Sustained release oral liquid suspension dosage form
LT2544532T (lt) 2010-03-12 2017-06-12 Monsanto Technology Llc Agrocheminių gelių kompozicijos
JP6209446B2 (ja) * 2010-06-02 2017-10-04 アステラス ドイチュランド ゲゼルシャフト ミット ベシュレンクテル ハフツング ベンダムスチンの経口投与形
KR102075173B1 (ko) * 2011-01-18 2020-02-07 센주 세이야꾸 가부시키가이샤 보존 효력을 갖는 브롬페낙 수성 액제 조성물
CN113842362A (zh) 2012-11-14 2021-12-28 格雷斯公司 含有生物活性材料与无序无机氧化物的组合物
EP4353311A3 (en) 2015-07-20 2024-07-17 The Brigham and Women's Hospital, Inc. Shear-thinning compositions as an intravascular embolic agent
CN105902409B (zh) * 2016-05-13 2019-03-05 广东龙湖科技股份有限公司 一种温和且具有触变性的牙膏
WO2019070818A2 (en) * 2017-10-04 2019-04-11 Panacea Biomatx, Inc. SUSPENSION OF ENCAPSULATED PHARMACEUTICAL PRODUCTS AND METHODS OF MAKING AND USING SAME
CN112402376A (zh) * 2019-08-22 2021-02-26 上海上药信谊药厂有限公司 一种结肠靶向的柳氮磺吡啶口服混悬剂及其制备方法
CN117883379A (zh) * 2021-02-12 2024-04-16 浙江贝灵生物医药有限公司 一种口服碱性溶媒组合物及其制备方法与应用
WO2022185338A1 (en) * 2021-03-05 2022-09-09 Alkem Laboratories Limited Stable oral suspension of celecoxib and method of preparation thereof
KR20240161261A (ko) 2023-05-04 2024-11-12 주식회사 퍼슨 성상 안정성이 우수한 현탁액 조성물

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JP2014503512A (ja) * 2010-12-10 2014-02-13 ビオプロジェ エンケファリナーゼ阻害剤の新規投与形態
JP2018516279A (ja) * 2015-05-29 2018-06-21 コーダドース・インコーポレーテッド 経口投与用のセレコキシブの液状配合物
JP2019531309A (ja) * 2016-10-19 2019-10-31 サインパス ファルマ, インク.Signpath Pharma, Inc. チャネル病を引き起こす薬物に対するｄｍｐｃ、ｄｍｐｇ、ｄｍｐｃ／ｄｍｐｇ、ｌｙｓｏｐｇ及びｌｙｓｏｐｃの防御効果

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