JP2004502682A5 - - Google Patents
Download PDFInfo
- Publication number
- JP2004502682A5 JP2004502682A5 JP2002507795A JP2002507795A JP2004502682A5 JP 2004502682 A5 JP2004502682 A5 JP 2004502682A5 JP 2002507795 A JP2002507795 A JP 2002507795A JP 2002507795 A JP2002507795 A JP 2002507795A JP 2004502682 A5 JP2004502682 A5 JP 2004502682A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- substituted
- pharmaceutical composition
- heterocyclic ring
- aryl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US21634100P | 2000-07-05 | 2000-07-05 | |
| PCT/FI2001/000637 WO2002002541A2 (en) | 2000-07-05 | 2001-07-04 | Inhibitors of copper-containing amine oxidases |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2004502682A JP2004502682A (ja) | 2004-01-29 |
| JP2004502682A5 true JP2004502682A5 (https=) | 2005-03-03 |
Family
ID=22806663
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002507795A Withdrawn JP2004502682A (ja) | 2000-07-05 | 2001-07-04 | 銅含有アミン・オキシダーゼの阻害剤 |
| JP2002506712A Withdrawn JP2004501962A (ja) | 2000-07-05 | 2001-07-04 | 銅含有アミン・オキシダーゼの阻害剤 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2002506712A Withdrawn JP2004501962A (ja) | 2000-07-05 | 2001-07-04 | 銅含有アミン・オキシダーゼの阻害剤 |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US6624202B2 (https=) |
| EP (2) | EP1301495A2 (https=) |
| JP (2) | JP2004502682A (https=) |
| CN (2) | CN1450998A (https=) |
| AU (3) | AU2001282162A1 (https=) |
| CA (2) | CA2414799A1 (https=) |
| HU (2) | HUP0301336A3 (https=) |
| IL (2) | IL153767A0 (https=) |
| NO (2) | NO20026283L (https=) |
| NZ (2) | NZ523464A (https=) |
| PL (2) | PL360353A1 (https=) |
| RU (2) | RU2003103286A (https=) |
| WO (2) | WO2002002541A2 (https=) |
| ZA (2) | ZA200300064B (https=) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2004502682A (ja) | 2000-07-05 | 2004-01-29 | バイオティ セラピーズ コーポレイション | 銅含有アミン・オキシダーゼの阻害剤 |
| US6982286B2 (en) * | 2001-07-12 | 2006-01-03 | Biotie Therapies Corp. | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
| EP1587800A1 (en) | 2003-01-27 | 2005-10-26 | Astellas Pharma Inc. | Thiazole derivatives and their use as vap-1 inhibitors |
| JP4758337B2 (ja) * | 2003-03-31 | 2011-08-24 | 株式会社アールテック・ウエノ | 血管透過性亢進疾患を治療する方法 |
| ES2335769T3 (es) * | 2003-05-26 | 2010-04-05 | Biotie Therapies Corp. | Vap-1 cristalina y sus usos. |
| FI20031927A0 (fi) * | 2003-12-31 | 2003-12-31 | Faron Pharmaceuticals Oy | Terapeuttisesti vaikuttavia aineita ja niiden käyttö |
| US8119651B2 (en) | 2004-01-30 | 2012-02-21 | Biotie Therapies Corp. | Compositions useful especially for treatment or prevention of metabolic syndrome |
| JP2007519688A (ja) * | 2004-01-30 | 2007-07-19 | ファロン ファーマシューティカルズ オサケ ユキチュア | メタボリックシンドロームの治療または予防に特に有効な組成物 |
| FI20040136A0 (fi) * | 2004-01-30 | 2004-01-30 | Faron Pharmaceuticals Oy | Erityisesti diabeetikoille soveltuvia koostumuksia |
| FI20040270A0 (fi) * | 2004-02-20 | 2004-02-20 | Biotie Therapies Oyj | Kuparia sisältävien amiinioksidaasien imhibiittoreina käyttökelpoiset hydratsinoalkoholijohdannaiset |
| DE602005013793D1 (de) * | 2004-07-27 | 2009-05-20 | Astellas Pharma Inc | Thiazolderivate mit vap-1-hemmender wirkung |
| CA2579889A1 (en) * | 2004-09-09 | 2006-03-16 | Astellas Pharma Inc. | Thiazole derivatives having vap-1 inhibitory activity |
| JP4140630B2 (ja) * | 2005-11-10 | 2008-08-27 | Ｔｄｋ株式会社 | 磁気ヘッドアセンブリ及び磁気ヘッドアセンブリの製造方法 |
| US8636995B2 (en) * | 2006-08-31 | 2014-01-28 | Cardiac Pacemakers, Inc. | Methods and devices to regulate stem cell homing |
| US8372399B2 (en) | 2006-08-31 | 2013-02-12 | Cardiac Pacemakers, Inc. | Bispecific antibodies and agents to enhance stem cell homing |
| US20080058922A1 (en) * | 2006-08-31 | 2008-03-06 | Cardiac Pacemakers, Inc. | Methods and devices employing vap-1 inhibitors |
| FI20061156A0 (fi) | 2006-12-27 | 2006-12-27 | Elina Kivi | Uusia peptidejä |
| WO2009061830A1 (en) * | 2007-11-06 | 2009-05-14 | Massachusetts Eye & Ear Infirmary | Methods and compositions for treating conditions associated with angiogenesis using a vascular adhesion protein-1 (vap-1) inhibitor |
| JP2011504485A (ja) * | 2007-11-21 | 2011-02-10 | ファーマクシス リミテッド | Ｓｓａｏ／ｖａｐ−１のハロアリルアミン阻害剤およびその用途 |
| TWI437986B (zh) | 2008-01-31 | 2014-05-21 | R Tech Ueno Ltd | 噻唑衍生物及使用該衍生物作為ｖａｐ－１抑制劑之用途 |
| TWI490214B (zh) | 2008-05-30 | 2015-07-01 | 艾德克 上野股份有限公司 | 苯或噻吩衍生物及該等作為ｖａｐ－１抑制劑之用途 |
| US8906642B2 (en) | 2008-09-03 | 2014-12-09 | Universitat Autonoma De Barcelona | Methods and compositions for the treatment and diagnosis of haemorrhagic conversion |
| RU2400233C1 (ru) | 2009-07-07 | 2010-09-27 | Общество с ограниченной ответственностью "Вирфарм" | Способ лечения заболеваний печени различного генеза |
| UA112154C2 (uk) | 2009-09-08 | 2016-08-10 | Біоті Терапіс Корп. | Застосування повністю людського анти-vap-1-антитіла для лікування фіброзних станів |
| JP5640983B2 (ja) | 2009-09-16 | 2014-12-17 | アステラス製薬株式会社 | グリシン化合物 |
| RU2010145439A (ru) * | 2010-11-08 | 2012-05-20 | Виктор Вениаминович Тец (RU) | Средство для лечения поражений печени, вызванных воздействием химических или биологических агентов |
| FI20115234A0 (fi) | 2011-03-08 | 2011-03-08 | Biotie Therapies Corp | Uusia pyridatsinoni- ja pyridoniyhdisteitä |
| SG193307A1 (en) | 2011-03-15 | 2013-10-30 | Astellas Pharma Inc | Guanidine compound |
| WO2014199171A1 (en) | 2013-06-12 | 2014-12-18 | Proximagen Limited | New therapeutic uses of enzyme inhibitors |
| EP3131539B1 (en) | 2014-04-15 | 2018-12-05 | Pécsi Tudományegyetem | Semicarbazide-sensitive amine oxidase inhibitors for use as analgesics in traumatic neuropathy and neurogenic inflammation |
| WO2015189534A1 (en) | 2014-06-12 | 2015-12-17 | Proximagen Limited | Vap-1 inhibitors for treating muscular dystrophy |
| RU2595868C1 (ru) | 2015-03-27 | 2016-08-27 | Виктор Вениаминович Тец | Лекарственное средство с гепатопротекторной активностью |
| JP2018076236A (ja) | 2015-06-05 | 2018-05-17 | 株式会社アールテック・ウエノ | がんを処置するための医薬組成物 |
| HK1256174A1 (zh) | 2015-12-07 | 2019-09-13 | Benevolentai Cambridge Limited | 用於治疗疼痛的 vap-1 抑制剂 |
| CN109810041B (zh) * | 2017-11-21 | 2023-08-15 | 药捷安康(南京)科技股份有限公司 | 卤代烯丙基胺类ssao/vap-1抑制剂及其应用 |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3377345A (en) * | 1966-09-23 | 1968-04-09 | Dow Chemical Co | Substituted 3, 4, 5, 6-tetrahydro-2h-1, 3, 4-oxadiazin-2-one compounds and method ofpreparation thereof |
| US3486916A (en) | 1966-12-22 | 1969-12-30 | William A Cordon | Cement mixes and the production of articles therefrom |
| SE320311B (https=) | 1968-07-15 | 1970-02-02 | Mo Och Domsjoe Ab | |
| EP0639972A1 (en) * | 1992-05-15 | 1995-03-01 | University Of Saskatchewan | Method for preventing endothelium damage in mammals and for alleviating pain associated with gout and arthritis |
| US5413634A (en) | 1993-08-06 | 1995-05-09 | Arco Chemical Technology, L.P. | Cement composition |
| CA2117585C (en) | 1993-09-14 | 2001-06-05 | Edward T. Shawl | Cement composition |
| WO1996006058A1 (en) | 1994-08-25 | 1996-02-29 | W.R. Grace & Co.-Conn. | Shrinkage reduction cement composition |
| US5618344A (en) | 1995-03-06 | 1997-04-08 | W. R. Grace & Co.-Conn. | Cement composition |
| US5603760A (en) | 1995-09-18 | 1997-02-18 | W. R. Grace & Co.-Conn. | Cement admixture capable of inhibiting drying shrinkage and method of using same |
| US5556460A (en) | 1995-09-18 | 1996-09-17 | W.R. Grace & Co.-Conn. | Drying shrinkage cement admixture |
| JP2004502682A (ja) | 2000-07-05 | 2004-01-29 | バイオティ セラピーズ コーポレイション | 銅含有アミン・オキシダーゼの阻害剤 |
-
2001
- 2001-07-04 JP JP2002507795A patent/JP2004502682A/ja not_active Withdrawn
- 2001-07-04 RU RU2003103286/15A patent/RU2003103286A/ru not_active Application Discontinuation
- 2001-07-04 CN CN01815102A patent/CN1450998A/zh active Pending
- 2001-07-04 CN CN01815101A patent/CN1450997A/zh active Pending
- 2001-07-04 EP EP01960763A patent/EP1301495A2/en not_active Withdrawn
- 2001-07-04 IL IL15376701A patent/IL153767A0/xx unknown
- 2001-07-04 WO PCT/FI2001/000637 patent/WO2002002541A2/en not_active Ceased
- 2001-07-04 CA CA002414799A patent/CA2414799A1/en not_active Abandoned
- 2001-07-04 EP EP01960764A patent/EP1313718A2/en not_active Withdrawn
- 2001-07-04 JP JP2002506712A patent/JP2004501962A/ja not_active Withdrawn
- 2001-07-04 RU RU2003103291/04A patent/RU2003103291A/ru not_active Application Discontinuation
- 2001-07-04 HU HU0301336A patent/HUP0301336A3/hu unknown
- 2001-07-04 PL PL36035301A patent/PL360353A1/xx not_active Application Discontinuation
- 2001-07-04 IL IL15376601A patent/IL153766A0/xx unknown
- 2001-07-04 AU AU2001282162A patent/AU2001282162A1/en not_active Abandoned
- 2001-07-04 AU AU8216301A patent/AU8216301A/xx active Pending
- 2001-07-04 NZ NZ523464A patent/NZ523464A/en unknown
- 2001-07-04 CA CA002414807A patent/CA2414807A1/en not_active Abandoned
- 2001-07-04 HU HU0301625A patent/HUP0301625A3/hu unknown
- 2001-07-04 AU AU2001282163A patent/AU2001282163B2/en not_active Ceased
- 2001-07-04 PL PL36037401A patent/PL360374A1/xx not_active Application Discontinuation
- 2001-07-04 NZ NZ523463A patent/NZ523463A/en unknown
- 2001-07-04 WO PCT/FI2001/000638 patent/WO2002002090A2/en not_active Ceased
- 2001-07-05 US US09/898,003 patent/US6624202B2/en not_active Expired - Fee Related
-
2002
- 2002-12-30 NO NO20026283A patent/NO20026283L/no not_active Application Discontinuation
- 2002-12-30 NO NO20026282A patent/NO20026282L/no not_active Application Discontinuation
-
2003
- 2003-01-03 ZA ZA200300064A patent/ZA200300064B/en unknown
- 2003-01-03 ZA ZA200300063A patent/ZA200300063B/en unknown
- 2003-07-21 US US10/622,581 patent/US20040106654A1/en not_active Abandoned
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| JP2004502682A5 (https=) | ||
| US20240050401A1 (en) | Methods of treating social function disorders | |
| RU2346945C2 (ru) | Производные n-гетероциклилметилбензамидов, их получение и их применение в терапии | |
| RU2003103291A (ru) | Ингибиторы медьсодержащих аминооксидаз | |
| US20240246936A1 (en) | Synthesis and novel salt forms of (r)-5-((e)-2-(pyrrolidin-3-ylvinyl)pyrimidine | |
| KR102602558B1 (ko) | Il-12, il-23 및/또는 ifn 알파 반응의 조정제로서의 포스핀 옥시드 알킬 아미드 치환된 헤테로아릴 화합물 | |
| JP2019501125A (ja) | ＩＬ−１２、ＩＬ−２３および／またはＩＦＮα応答のモジュレーターとして有用なイミダゾピリダジン化合物 | |
| JP2004501962A5 (https=) | ||
| US5426106A (en) | Pyrrolo-pyridazinone derivatives | |
| BR112021014709A2 (pt) | Compostos piridina ou piridazina dissubstituídos por amida | |
| JP2011513421A (ja) | サブタイプ選択的なジアザビシクロアルカンのアミド | |
| JP2019535723A (ja) | Ｉｌ−１２、ｉｌ−２３および／またはｉｆｎ−アルファのイミダゾピリダジン調節剤 | |
| JP2013512922A (ja) | 神経型ニコチン性アセチルコリン受容体リガンドとしての３，６−ジアザビシクロ［３．１．１］ヘプタン | |
| CN100436414C (zh) | 作为毒蕈碱受体拮抗剂的氮杂双环衍生物 | |
| JP4920408B2 (ja) | 向知性作用を有する化合物、その調製方法、これを有する薬学的組成物、及びその使用 | |
| CN1097459C (zh) | 用作磷酸二酯酶iv抑制剂的二氮杂䓬并吲哚 | |
| US20110118239A1 (en) | Preparation and enantiomeric separation of 7-(3-pyridinyl)-1,7-diazaspiro[4.4]nonane and novel salt forms of the racemate and enantiomers | |
| JP7618642B2 (ja) | インターロイキンの調節におけるプロドラッグ | |
| CA2742366A1 (en) | Synthesis and salt forms of (r)-5-((e)-2-(pyrrolidin-3-ylvinyl)pyrimidine | |
| RU2081870C1 (ru) | Производные диазепинона, способы их получения и фармацевтическая композиция | |
| GB2290292A (en) | 2-Phenylpyridazino[4,5-b]indole-1,4-dione derivatives as NMDA and AMPA antagonists | |
| CN116898854A (zh) | 一种吡唑并嘧啶类化合物的新用途 | |
| JPH032155A (ja) | カルバミド酸エステル誘導体 | |
| TW201206910A (en) | Substituted N-heterocycloalkyl bipyrrolidinylphenyl amide derivatives, preparation and therapeutic use thereof | |
| JP2861274B2 (ja) | アミノケトン誘導体 |