JP2003522766A5 - - Google Patents

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Publication number
JP2003522766A5
JP2003522766A5 JP2001558440A JP2001558440A JP2003522766A5 JP 2003522766 A5 JP2003522766 A5 JP 2003522766A5 JP 2001558440 A JP2001558440 A JP 2001558440A JP 2001558440 A JP2001558440 A JP 2001558440A JP 2003522766 A5 JP2003522766 A5 JP 2003522766A5
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JP
Japan
Prior art keywords
amino
thiophenecarboxamide
aminocarbonyl
phenyl
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2001558440A
Other languages
English (en)
Japanese (ja)
Other versions
JP4812999B2 (ja
JP2003522766A (ja
Filing date
Publication date
Priority claimed from GBGB0003154.2A external-priority patent/GB0003154D0/en
Application filed filed Critical
Publication of JP2003522766A publication Critical patent/JP2003522766A/ja
Publication of JP2003522766A5 publication Critical patent/JP2003522766A5/ja
Application granted granted Critical
Publication of JP4812999B2 publication Critical patent/JP4812999B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2001558440A 2000-02-12 2001-02-07 ヘテロ芳香族カルボキサミド誘導体及び酵素ｉｋｋ−２のインヒビターとしてのそれらの使用 Expired - Fee Related JP4812999B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0003154.2A GB0003154D0 (en) 2000-02-12 2000-02-12 Novel compounds
GB0003154.2 2000-02-12
PCT/SE2001/000248 WO2001058890A1 (en) 2000-02-12 2001-02-07 Heteroaromatic carboxamide derivatives and their use as inhibitors of the enzyme ikk-2

Publications (3)

Publication Number Publication Date
JP2003522766A JP2003522766A (ja) 2003-07-29
JP2003522766A5 true JP2003522766A5 (enExample) 2008-03-27
JP4812999B2 JP4812999B2 (ja) 2011-11-09

Family

ID=9885396

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001558440A Expired - Fee Related JP4812999B2 (ja) 2000-02-12 2001-02-07 ヘテロ芳香族カルボキサミド誘導体及び酵素ｉｋｋ−２のインヒビターとしてのそれらの使用

Country Status (21)

Country Link
US (2) US7358376B2 (enExample)
EP (1) EP1261600B1 (enExample)
JP (1) JP4812999B2 (enExample)
KR (1) KR100738165B1 (enExample)
CN (1) CN1243747C (enExample)
AT (1) ATE266019T1 (enExample)
AU (1) AU781047B2 (enExample)
BR (1) BR0108143A (enExample)
CA (1) CA2396824C (enExample)
DE (1) DE60103132T2 (enExample)
DK (1) DK1261600T3 (enExample)
ES (1) ES2218376T3 (enExample)
GB (1) GB0003154D0 (enExample)
IL (2) IL150482A0 (enExample)
MX (1) MXPA02007734A (enExample)
NO (1) NO327741B1 (enExample)
NZ (1) NZ519947A (enExample)
PT (1) PT1261600E (enExample)
TR (1) TR200401962T4 (enExample)
WO (1) WO2001058890A1 (enExample)
ZA (1) ZA200205300B (enExample)

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WO2005037797A1 (en) * 2003-10-21 2005-04-28 Pharmacia Corporation Substituted pyrazole urea compounds for the treatment of inflammation
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WO2006036031A1 (ja) * 2004-09-30 2006-04-06 Takeda Pharmaceutical Company Limited 縮合フラン誘導体およびその用途
JP5000490B2 (ja) 2005-04-28 2012-08-15 武田薬品工業株式会社 チエノピリミドン化合物
US8063071B2 (en) 2007-10-31 2011-11-22 GlaxoSmithKline, LLC Chemical compounds
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