JP2001500496A - 医薬化合物の製造方法 - Google Patents

医薬化合物の製造方法

Info

Publication number
JP2001500496A
JP2001500496A JP10512921A JP51292198A JP2001500496A JP 2001500496 A JP2001500496 A JP 2001500496A JP 10512921 A JP10512921 A JP 10512921A JP 51292198 A JP51292198 A JP 51292198A JP 2001500496 A JP2001500496 A JP 2001500496A
Authority
JP
Japan
Prior art keywords
alkyl
aromatic group
formula
substituted
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP10512921A
Other languages
English (en)
Japanese (ja)
Inventor
マルティネリ，マイケル・ジェイ
モーアー，エリック・ディ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
University of Hawai'i at Hilo
Original Assignee
University of Hawaiʻi at Mānoa
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by University of Hawaiʻi at Mānoa, Eli Lilly and Co filed Critical University of Hawaiʻi at Mānoa
Publication of JP2001500496A publication Critical patent/JP2001500496A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/12—Cyclic peptides with only normal peptide bonds in the ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
  • Peptides Or Proteins (AREA)
JP10512921A 1996-09-06 1997-09-05 医薬化合物の製造方法 Pending JP2001500496A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US2543896P 1996-09-06 1996-09-06
US60/025,438 1996-09-06
PCT/US1997/015626 WO1998009988A1 (en) 1996-09-06 1997-09-05 Process to prepare pharmaceutical compounds

Publications (1)

Publication Number Publication Date
JP2001500496A true JP2001500496A (ja) 2001-01-16

Family

ID=21826074

Family Applications (1)

Application Number Title Priority Date Filing Date
JP10512921A Pending JP2001500496A (ja) 1996-09-06 1997-09-05 医薬化合物の製造方法

Country Status (10)

Country Link
US (1) US6252064B1 (enExample)
EP (1) EP0956295A1 (enExample)
JP (1) JP2001500496A (enExample)
KR (1) KR20010029474A (enExample)
AU (1) AU4182197A (enExample)
BR (1) BR9712805A (enExample)
CA (1) CA2264245A1 (enExample)
HU (1) HUP0000291A3 (enExample)
IL (1) IL128497A0 (enExample)
WO (1) WO1998009988A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0870506A1 (en) * 1997-04-11 1998-10-14 Eli Lilly And Company Compositions comprising a cryptophycin compound in combination with a synchronizing or activating agent for treating cancer
JP4776843B2 (ja) 1999-10-01 2011-09-21 イムノゲン インコーポレーティッド 免疫複合体及び化学療法剤を用いる癌治療用組成物及び方法
UA79293C2 (en) * 2002-07-03 2007-06-11 Univ Wayne State 4-(7'-halo-2-quino (xa-) linyloxy)phenoxy propionic acid derivatives as antineoplastic agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE203016T1 (de) * 1993-12-21 2001-07-15 Univ Hawaii Cryptophycine
DE69633667T2 (de) * 1995-03-07 2006-03-02 University Of Hawaii, Honolulu Neue synthetische cryptophycine
EP0957912A1 (en) * 1996-08-30 1999-11-24 Eli Lilly And Company Pharmaceutical compounds
WO1998008505A1 (en) * 1996-08-30 1998-03-05 Eli Lilly And Company Pharmaceutical compounds

Also Published As

Publication number Publication date
EP0956295A1 (en) 1999-11-17
KR20010029474A (ko) 2001-04-06
WO1998009988A1 (en) 1998-03-12
AU4182197A (en) 1998-03-26
HUP0000291A2 (hu) 2000-09-28
CA2264245A1 (en) 1998-03-12
BR9712805A (pt) 1999-11-23
US6252064B1 (en) 2001-06-26
HUP0000291A3 (en) 2000-10-30
EP0956295A4 (enExample) 1999-12-22
IL128497A0 (en) 2000-01-31

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