JOP20190177A1 - طريقة لعلاج أو تحسين اضطرابات أيضية باستخدام مساعدات مستقبل glp-1 مقترنة بمناهضات لمستقبل ببتيد مثبط معوي (gipr) - Google Patents

طريقة لعلاج أو تحسين اضطرابات أيضية باستخدام مساعدات مستقبل glp-1 مقترنة بمناهضات لمستقبل ببتيد مثبط معوي (gipr)

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Publication number
JOP20190177A1
JOP20190177A1 JOP/2019/0177A JOP20190177A JOP20190177A1 JO P20190177 A1 JOP20190177 A1 JO P20190177A1 JO P20190177 A JOP20190177 A JO P20190177A JO P20190177 A1 JOP20190177 A1 JO P20190177A1
Authority
JO
Jordan
Prior art keywords
glp
receptor
gipr
treating
antagonists
Prior art date
Application number
JOP/2019/0177A
Other languages
Arabic (ar)
English (en)
Inventor
Murielle M Veniant-Ellison
Leslie P Miranda
Yuan Cheng
James R Falsey
Chawita Netirojjanakul
Bradley J Herberich
Jing Xu
Jerry Ryan Holder
Bin Wu
Shanaka Stanislaus
Kelvin Sham
Junming Yie
Shu-Chen Lu
Original Assignee
Amgen Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=61832572&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JOP20190177(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Amgen Inc filed Critical Amgen Inc
Publication of JOP20190177A1 publication Critical patent/JOP20190177A1/ar

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    • A61K47/68Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an antibody, an immunoglobulin or a fragment thereof, e.g. an Fc-fragment
    • A61K47/6835Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an antibody, an immunoglobulin or a fragment thereof, e.g. an Fc-fragment the modifying agent being an antibody or an immunoglobulin bearing at least one antigen-binding site
    • A61K47/6847Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an antibody, an immunoglobulin or a fragment thereof, e.g. an Fc-fragment the modifying agent being an antibody or an immunoglobulin bearing at least one antigen-binding site the antibody targeting a hormone or a hormone-releasing or -inhibiting factor
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    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
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    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A61K47/6801Drug-antibody or immunoglobulin conjugates defined by the pharmacologically or therapeutically active agent
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
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    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
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    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
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    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2869Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against hormone receptors
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
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    • C07ORGANIC CHEMISTRY
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    • C07K2317/76Antagonist effect on antigen, e.g. neutralization or inhibition of binding
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    • C07ORGANIC CHEMISTRY
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    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/77Internalization into the cell

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JOP/2019/0177A 2017-01-17 2017-06-16 طريقة لعلاج أو تحسين اضطرابات أيضية باستخدام مساعدات مستقبل glp-1 مقترنة بمناهضات لمستقبل ببتيد مثبط معوي (gipr) JOP20190177A1 (ar)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201762447332P 2017-01-17 2017-01-17

Publications (1)

Publication Number Publication Date
JOP20190177A1 true JOP20190177A1 (ar) 2019-07-16

Family

ID=61832572

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Application Number Title Priority Date Filing Date
JOP/2019/0177A JOP20190177A1 (ar) 2017-01-17 2017-06-16 طريقة لعلاج أو تحسين اضطرابات أيضية باستخدام مساعدات مستقبل glp-1 مقترنة بمناهضات لمستقبل ببتيد مثبط معوي (gipr)

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US (3) US10905772B2 (enExample)
EP (2) EP4480537A3 (enExample)
JP (3) JP7175899B2 (enExample)
KR (3) KR102781241B1 (enExample)
CN (2) CN110662558B (enExample)
AR (1) AR110751A1 (enExample)
AU (2) AU2018210858B2 (enExample)
BR (1) BR112019014588A2 (enExample)
CA (1) CA3049023A1 (enExample)
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CO (1) CO2019007685A2 (enExample)
CR (2) CR20230302A (enExample)
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EA (1) EA201991721A1 (enExample)
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HU (1) HUE069334T2 (enExample)
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JO (1) JOP20190177A1 (enExample)
LT (1) LT3570885T (enExample)
MA (1) MA47314B1 (enExample)
MD (1) MD3570885T2 (enExample)
MX (2) MX2019008462A (enExample)
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PE (2) PE20250777A1 (enExample)
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