IT1231760B - Derivati di acido piridoncarbossilico e loro sali, procedimento per produrre gli stessi e agenti antibatterici che li contengono - Google Patents

Derivati di acido piridoncarbossilico e loro sali, procedimento per produrre gli stessi e agenti antibatterici che li contengono

Info

Publication number
IT1231760B
IT1231760B IT8947875A IT4787589A IT1231760B IT 1231760 B IT1231760 B IT 1231760B IT 8947875 A IT8947875 A IT 8947875A IT 4787589 A IT4787589 A IT 4787589A IT 1231760 B IT1231760 B IT 1231760B
Authority
IT
Italy
Prior art keywords
salts
procedure
contain
produce
same
Prior art date
Application number
IT8947875A
Other languages
English (en)
Other versions
IT8947875A0 (it
Inventor
Hirokazu Narita
Yozo Todo
Jun Nitta
Hiroyasu Takagi
Fumihiko Iino
Original Assignee
Toyama Chemical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Toyama Chemical Co Ltd filed Critical Toyama Chemical Co Ltd
Publication of IT8947875A0 publication Critical patent/IT8947875A0/it
Application granted granted Critical
Publication of IT1231760B publication Critical patent/IT1231760B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/06—Peri-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
IT8947875A 1988-04-23 1989-04-21 Derivati di acido piridoncarbossilico e loro sali, procedimento per produrre gli stessi e agenti antibatterici che li contengono IT1231760B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10062888 1988-04-23
JP1075873A JPH0228178A (ja) 1988-04-23 1989-03-28 新規なピリドンカルボン酸誘導体およびその塩並びにそれらの製造法

Publications (2)

Publication Number Publication Date
IT8947875A0 IT8947875A0 (it) 1989-04-21
IT1231760B true IT1231760B (it) 1991-12-21

Family

ID=26417038

Family Applications (1)

Application Number Title Priority Date Filing Date
IT8947875A IT1231760B (it) 1988-04-23 1989-04-21 Derivati di acido piridoncarbossilico e loro sali, procedimento per produrre gli stessi e agenti antibatterici che li contengono

Country Status (21)

Country Link
US (1) US4990508A (it)
JP (1) JPH0228178A (it)
KR (1) KR910005833B1 (it)
AT (1) AT398422B (it)
AU (1) AU601324B2 (it)
BE (1) BE1003252A4 (it)
CA (1) CA1340493C (it)
CH (1) CH680793A5 (it)
DE (1) DE3913245C2 (it)
DK (1) DK175649B1 (it)
ES (1) ES2016012A6 (it)
FI (1) FI91529C (it)
FR (1) FR2630441B1 (it)
GB (1) GB2217710B (it)
HU (2) HU205759B (it)
IL (1) IL89931A (it)
IT (1) IT1231760B (it)
NL (1) NL192832C (it)
NO (1) NO171214C (it)
NZ (1) NZ228847A (it)
SE (1) SE504625C2 (it)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5104868A (en) * 1988-06-21 1992-04-14 Pfizer Inc. Tricyclic derivatives of 7-substituted-6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acids and esters
EP0997466A1 (en) * 1988-10-24 2000-05-03 PROCTER & GAMBLE PHARMACEUTICALS, INC. Novel antimicrobial lactam-quinolones
EP0449445A3 (en) * 1990-03-27 1993-08-25 Pfizer Inc. Preparation of beta-ketoesters useful in preparing quinolone antibiotics
IT1248011B (it) * 1991-06-07 1995-01-05 Mediolanum Farmaceutici Spa Procedimento per la preparazione dell'acido 9-fluoro-10- (4-metil-1-piperazinil)-7-oxo-2,3-diidro-7h-pirido (1,2,3-de) (1,4)benzotiadin-6-carbossilico cloridrato.
EG20543A (en) * 1992-10-30 1999-07-31 Procter & Gamble Process for preparing of novel antimicrobial -5- (n-heterosubstituted amino) quinolones
TW252107B (it) * 1993-08-27 1995-07-21 Hokuriku Pharmacetical Co Ltd
IT1270834B (it) * 1993-10-27 1997-05-13 Archimica Spa Disolfuro chinolico
IT1270836B (it) * 1993-10-27 1997-05-13 Archimica Spa Procedimento per la preparazione di rufloxacina e suoi sali
USH1480H (en) * 1993-12-09 1995-09-05 The Procter & Gamble Company Methods of using dyphylline for the promotion of hair growth
KR100768034B1 (ko) 1999-03-17 2007-10-17 다이이찌 세이야꾸 가부시기가이샤 의약 조성물
KR20040105772A (ko) 2002-03-21 2004-12-16 바스프 악티엔게젤샤프트 살진균성 트리아졸로피리미딘, 이의 제조방법 및 유해진균 방제를 위한 이의 용도 및 상기 성분을 함유하는조성물
CN1332962C (zh) * 2005-07-12 2007-08-22 武汉人福药业有限责任公司 一种合成甲磺酸帕珠沙星中间体的方法
PL2383271T3 (pl) * 2006-03-13 2013-12-31 Kyorin Seiyaku Kk Aminochinolony jako inhibitory GSK-3
EP2203458B1 (en) * 2007-09-11 2011-11-02 Kyorin Pharmaceutical Co., Ltd. Cyanoaminoquinolones as gsk-3 inhibitors
CA2699152C (en) 2007-09-12 2015-11-24 Activx Biosciences, Inc. Spirocyclic aminoquinolones as gsk-3 inhibitors
JP5502889B2 (ja) * 2009-03-11 2014-05-28 杏林製薬株式会社 ｇｓｋ−３阻害剤としての７−シクロアルキルアミノキノロン
CN101928290B (zh) * 2009-11-27 2011-11-09 浙江司太立制药股份有限公司 一种甲磺酸帕珠沙星的纯化方法
CN102295652A (zh) * 2011-06-27 2011-12-28 辽宁海神联盛制药有限公司 一种甲磺酸帕珠沙星合成工艺的改进方法
CN102850375A (zh) * 2012-03-06 2013-01-02 江西师范大学 一类多取代吡啶并[4, 3-d]噁嗪化合物及制备方法
CN103772412B (zh) * 2012-10-23 2016-03-16 浙江海森药业有限公司 一种帕珠沙星中间体的制备方法
CN105622632B (zh) * 2014-10-29 2018-06-29 浙江海森药业股份有限公司 一种喹诺酮类化合物及其制备方法

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3883522A (en) * 1974-02-11 1975-05-13 Riker Laboratories Inc Substituted pyrido(1,2,3-de)-1,4-benzoxazines
DE3211984C2 (de) * 1981-05-21 1986-04-03 Dieter Dr. 7900 Ulm Benz Rotierende Zahnbürste
JPS591489A (ja) * 1982-06-29 1984-01-06 Dai Ichi Seiyaku Co Ltd ピリドベンゾオキサジン誘導体
DE3234529A1 (de) * 1982-09-17 1984-03-22 Bayer Ag, 5090 Leverkusen Substituierte benzoxazin-derivate
US4603199A (en) * 1982-10-25 1986-07-29 Riker Laboratories, Inc. Phenyl-substituted tricyclic antibacterial agent intermediates
US4607032A (en) * 1984-04-26 1986-08-19 Abbott Laboratories Quino-benoxazine antibacterial compounds
US4540694A (en) * 1984-04-26 1985-09-10 Abbott Laboratories 1-Pyridine substituted quino-benoxazines and antibacterial use
US4822801A (en) * 1984-07-20 1989-04-18 Warner-Lambert Company 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents
US4623650A (en) * 1984-12-06 1986-11-18 Pfizer Inc. Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids
DE3517709A1 (de) * 1985-01-05 1986-07-10 Bayer Ag Basische zubereitungen von chinoloncarbonsaeuren
DE3525108A1 (de) * 1985-06-07 1986-12-11 Bayer Ag, 5090 Leverkusen Antibakteriell wirksame chinoloncarbonsaeureester
DE3522406A1 (de) * 1985-06-22 1987-01-02 Bayer Ag Verfahren zur herstellung von 1,8-verbrueckten 4-chinolon-3-carbonsaeuren
DE3522405A1 (de) * 1985-06-22 1987-01-02 Bayer Ag 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln
DE3543513A1 (de) * 1985-12-10 1987-06-11 Bayer Ag Enantiomerenreine 1,8-verbrueckte 4-chinolon-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende arzneimittel und ihre verwendung zur herstellung von arzneimitteln
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
US4777253A (en) * 1986-04-25 1988-10-11 Abbott Laboratories Process for preparation of racemate and optically active ofloxacin and related derivatives
IT1196429B (it) * 1986-07-01 1988-11-16 Mediolanum Farmaceutici Srl Processo per la preparazione di pirido benzotiazine ad attivita' antibatterica e loro sali con acidi solfonici
DE3623757A1 (de) * 1986-07-15 1988-01-21 Bayer Ag Neue 1,8-verbrueckte 4-chinoloncarbonsaeuren und diese enthaltende arzneimittel
DE3639465A1 (de) * 1986-11-18 1988-05-19 Hoechst Ag Optisch aktive gyrasehemmer, ihre herstellung und verwendung als antibiotika
DE3641661A1 (de) * 1986-12-05 1988-06-30 Bayer Ag Verfahren zur herstellung von chinoloncarbonsaeureestern
DE3711193A1 (de) * 1987-04-02 1988-10-13 Bayer Ag 5-substituierte chinolon- und naphthyridoncarbonsaeure-derivate
JP2598921B2 (ja) * 1987-10-05 1997-04-09 富山化学工業株式会社 新規なキノリン誘導体およびその塩
DE3810080A1 (de) * 1988-03-25 1989-10-05 Bayer Ag Trisubstituierte 1,3,5-triazin-2,4,6-trione
DE3815481A1 (de) * 1988-05-06 1989-11-16 Sandoz Ag Sulfonsaeuregruppenfreie basische verbindung
US5039682A (en) * 1988-06-21 1991-08-13 Pfizer Inc. 6-fluoro-1,4-dihydroquinol-4-one-3-carboxylic acid derivatives and intermediates therefor

Also Published As

Publication number Publication date
US4990508A (en) 1991-02-05
CH680793A5 (it) 1992-11-13
FI91529B (fi) 1994-03-31
AU3266189A (en) 1989-10-26
FR2630441B1 (fr) 1994-10-14
CA1340493C (en) 1999-04-13
FI891910A (fi) 1989-10-24
SE8901464L (sv) 1989-10-24
FR2630441A1 (fr) 1989-10-27
DE3913245C2 (de) 1999-07-15
GB2217710B (en) 1991-12-04
DK192589A (da) 1989-10-24
GB8908096D0 (en) 1989-05-24
GB2217710A (en) 1989-11-01
JPH0228178A (ja) 1990-01-30
NL192832C (nl) 1998-03-04
FI891910A0 (fi) 1989-04-21
AT398422B (de) 1994-12-27
HU205759B (en) 1992-06-29
NL8901007A (nl) 1989-11-16
ES2016012A6 (es) 1990-10-01
SE8901464D0 (sv) 1989-04-21
IL89931A (en) 1993-06-10
HUT51621A (en) 1990-05-28
NZ228847A (en) 1990-04-26
DK192589D0 (da) 1989-04-20
HU211568A9 (en) 1995-12-28
FI91529C (fi) 1994-07-11
DE3913245A1 (de) 1989-11-02
KR910005833B1 (ko) 1991-08-05
AU601324B2 (en) 1990-09-06
KR900016222A (ko) 1990-11-12
DK175649B1 (da) 2005-01-03
NO891650L (no) 1989-10-24
ATA95989A (de) 1994-04-15
IT8947875A0 (it) 1989-04-21
NL192832B (nl) 1997-11-03
IL89931A0 (en) 1989-12-15
NO171214B (no) 1992-11-02
SE504625C2 (sv) 1997-03-17
JPH0588714B2 (it) 1993-12-24
NO171214C (no) 1993-02-10
BE1003252A4 (fr) 1992-02-11
NO891650D0 (no) 1989-04-21

Similar Documents

Publication Publication Date Title
IT1231760B (it) Derivati di acido piridoncarbossilico e loro sali, procedimento per produrre gli stessi e agenti antibatterici che li contengono
IT1209953B (it) Derivati di 1,4-diidro-4-ossonaftiridina e relativi sali, procedimento per la loro produzione e agenti antibatterici che comprendono i medesimi
IT1193211B (it) Derivati dell'acido 2,4,6-triiodo-isoftalico,metodo per la loro preparazione e mezzi di contrasto che li contengono
IT8449339A0 (it) Composti eterociclici, loro preparazione e loro impiego come medicamenti
IT8567743A0 (it) Derivati di benzimidazolo procedimento per la loro preparazione e agenti antiulcera che li contengono
IT1207226B (it) Derivati dell'acido 2,4,6-triiodo-isoftalico, metodo per la loro preparazione e mezzi di contrasto che li contengono.
IT1218336B (it) Derivati di acido 4-osso-1,4-diidro-nicotinico e loro sali,procedimentoper produrli ed agenti antibatterici che li contengono
IT1197759B (it) Derivati acidi idrossicarbossilici oligomeri,loro preparazione e loro impiego
IT8123602A0 (it) Sali stabili della s-adenosilmetionina, processo per la loro preparazione e composizioni terapeutiche che li comprendono come principio attivo.
IT8448889A1 (it) Composti azolici loro preparazione e loro impiego come funghicidi e antimicotici
IT1242004B (it) Derivati di isoindolo e loro sali, procedimenti per produrli ed agenteantitumore che li contiene.
IT8947598A0 (it) Composti carbonilati, loro preparazione e loro impiego come erbicidi
IT8123603A0 (it) Sali stabili della s-adenosilmetionina, processo per la loro preparazione e composizioni terapeutiche che li comprendono come principio attivo.
IT1205715B (it) Derivati di piroglutammide,agenti nootropici che li contengono e procedimento per la loro preparazione
IT1129264B (it) Derivati di acido cicloesancarbossilico particolarmente utili come antiulcera e procedimento per la loro preparazione
IT7949927A0 (it) Imidazochinossaline e loro sali,loro procedimento di produzione,loro impiego come medicamenti e composizioni farmaceutiche che le contengono
IT1199860B (it) Polieteri glicosilati,composizioni che li comprendono,procedimento per la loro preparazione e impiego
IT1174760B (it) Derivati di acido 4-idrossi 3-chinolin carbossilico sostituiti in 2,loro preparazione,loro applicazione come medicamenti,composizioni che li contengono ed imtermedi ottenuti
IT1178330B (it) Composti tiofensolfonammididici sostituiti, loro sali, erbicidi che li contengono e procedimento per prepararli
IT1147839B (it) Derivati di acido ciclopropan carbossilico per la lotta contro i parassiti,composizioni che li contengono e procedimento per la loro preparazione
IT8548298A0 (it) Nuovi derivati steroidei sostituiti in posizione 11-beta, procedimento per la loro preparazione e loro applicazione come medicamenti
IT1211960B (it) Derivati di azaspirodecano,loro sali,procedimento di preparazione,applicazione quali medicamenti e composizioni che li contengono
IT1247696B (it) Penam-derivati e loro sali, procedimento per la loro produzione ed agente antibatterico che li contiene.
IT1185067B (it) Derivati di tiocianopirimidina,processo per la loro produzione e funghicidi per uso agricolo e orticolo che li contengono
IT1168389B (it) Derivati di alcandioli con attivita' ipolipidemizzante,metodi per la loro preparazione e composizioni farmaceutiche che li contengono

Legal Events

Date Code Title Description
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19970222