IL88086A - Azetidinyl quinolone carboxylic acids esters and amides antibacterial compositions containing said compounds and uses thereof - Google Patents

Azetidinyl quinolone carboxylic acids esters and amides antibacterial compositions containing said compounds and uses thereof

Info

Publication number
IL88086A
IL88086A IL8808688A IL8808688A IL88086A IL 88086 A IL88086 A IL 88086A IL 8808688 A IL8808688 A IL 8808688A IL 8808688 A IL8808688 A IL 8808688A IL 88086 A IL88086 A IL 88086A
Authority
IL
Israel
Prior art keywords
alkyl
azetidinyl
amino
amides
compounds
Prior art date
Application number
IL8808688A
Other languages
English (en)
Other versions
IL88086A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL88086A0 publication Critical patent/IL88086A0/xx
Publication of IL88086A publication Critical patent/IL88086A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Steroid Compounds (AREA)
IL8808688A 1987-10-26 1988-10-19 Azetidinyl quinolone carboxylic acids esters and amides antibacterial compositions containing said compounds and uses thereof IL88086A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1987/002792 WO1989003828A1 (en) 1987-10-26 1987-10-26 Azetidinyl quinolone carboxylic acids and esters

Publications (2)

Publication Number Publication Date
IL88086A0 IL88086A0 (en) 1989-06-30
IL88086A true IL88086A (en) 1997-01-10

Family

ID=22202632

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8808688A IL88086A (en) 1987-10-26 1988-10-19 Azetidinyl quinolone carboxylic acids esters and amides antibacterial compositions containing said compounds and uses thereof

Country Status (19)

Country Link
US (1) US5039683A (xx)
EP (1) EP0314362B1 (xx)
JP (1) JPH01146879A (xx)
KR (1) KR900006741B1 (xx)
AT (1) ATE100805T1 (xx)
AU (1) AU602431B2 (xx)
DE (1) DE3887443T2 (xx)
DK (1) DK591588A (xx)
ES (1) ES2061680T3 (xx)
FI (1) FI893048A (xx)
HU (1) HU205105B (xx)
IE (1) IE63284B1 (xx)
IL (1) IL88086A (xx)
MY (1) MY103436A (xx)
NO (1) NO892616D0 (xx)
NZ (1) NZ226689A (xx)
PT (1) PT88837B (xx)
WO (1) WO1989003828A1 (xx)
ZA (1) ZA887927B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2634483B2 (fr) * 1987-12-29 1994-03-04 Esteve Labor Dr Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments
US5173484A (en) * 1988-02-05 1992-12-22 Bayer Aktiengesellschaft Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them
EP0997466A1 (en) * 1988-10-24 2000-05-03 PROCTER & GAMBLE PHARMACEUTICALS, INC. Novel antimicrobial lactam-quinolones
FR2654728B2 (fr) * 1989-03-16 1994-09-23 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament.
FR2644455B1 (fr) * 1989-03-16 1994-09-23 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicaments
FR2649106A2 (fr) * 1989-06-29 1991-01-04 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament
NO177302C (no) * 1989-03-16 1995-08-23 Esteve Labor Dr Analogifremgangsmåte til fremstilling av terapeutisk aktive substituerte azetidinylkinolon(naftyridon)karboksylsyrederivater
FR2690161B1 (fr) * 1992-04-16 1995-06-30 Esteve Labor Dr Derives de pyridone azetidinyl substitues avec activite antimicrobienne.
US5885983A (en) * 1996-05-10 1999-03-23 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
WO2005019224A2 (en) * 2003-06-06 2005-03-03 Cadila Healthcare Limited Novel antiinfective compounds
WO2005026146A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Azetidinyl quinolones as antibacterial agents

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4670444B1 (en) * 1980-09-03 1999-02-09 Bayer Ag and-naphthyridine-3-carboxylic acids and antibacte7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-quinoline-rial agents containing these compounds
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
NZ208470A (en) * 1983-07-18 1988-06-30 Abbott Lab 6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such
JPS6089480A (ja) * 1983-10-21 1985-05-20 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体
JPS60126284A (ja) * 1983-12-09 1985-07-05 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体およびその塩
US4623650A (en) * 1984-12-06 1986-11-18 Pfizer Inc. Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids
JPS61137885A (ja) * 1984-12-08 1986-06-25 Dainippon Pharmaceut Co Ltd 1,8−ナフチリジン誘導体、そのエステルおよびその塩
JPS61152682A (ja) * 1984-12-27 1986-07-11 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体、そのエステルおよびその塩
JPS61282382A (ja) * 1985-06-06 1986-12-12 Dainippon Pharmaceut Co Ltd フエニル置換1,8−ナフチリジン誘導体、そのエステルおよびその塩
JPS62469A (ja) * 1985-06-27 1987-01-06 Dainippon Pharmaceut Co Ltd 新規キノロン誘導体、そのエステルおよびその塩
JPS6219883A (ja) * 1985-07-19 1987-01-28 Ricoh Co Ltd 色替え可能な現像装置
JPH0674260B2 (ja) * 1985-08-01 1994-09-21 大日本製薬株式会社 キノリン誘導体、そのエステルおよびその塩
JPS62215572A (ja) * 1986-03-17 1987-09-22 Kyorin Pharmaceut Co Ltd キノロンカルボン酸誘導体
CN1019114B (zh) * 1986-03-31 1992-11-18 三共株式会社 喹啉-3-羟酸衍生物的制备方法
JPH0689480A (ja) * 1992-09-09 1994-03-29 Ricoh Co Ltd 光磁気記録再生装置

Also Published As

Publication number Publication date
KR890006616A (ko) 1989-06-14
AU602431B2 (en) 1990-10-11
DK591588A (da) 1989-04-27
ES2061680T3 (es) 1994-12-16
NO892616L (no) 1989-06-23
MY103436A (en) 1993-06-30
IE63284B1 (en) 1995-04-05
FI893048A0 (fi) 1989-06-21
HU205105B (en) 1992-03-30
JPH01146879A (ja) 1989-06-08
ATE100805T1 (de) 1994-02-15
WO1989003828A1 (en) 1989-05-05
ZA887927B (en) 1990-06-27
KR900006741B1 (ko) 1990-09-20
FI893048A (fi) 1989-06-21
DE3887443T2 (de) 1994-05-11
EP0314362A3 (en) 1989-10-18
NO892616D0 (no) 1989-06-23
HUT52497A (en) 1990-07-28
AU2432588A (en) 1988-10-25
DE3887443D1 (de) 1994-03-10
US5039683A (en) 1991-08-13
NZ226689A (en) 1990-03-27
PT88837B (pt) 1993-01-29
IL88086A0 (en) 1989-06-30
EP0314362B1 (en) 1994-01-26
EP0314362A2 (en) 1989-05-03
DK591588D0 (da) 1988-10-25
IE883217L (en) 1989-04-26

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Legal Events

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FF Patent granted
KB Patent renewed
RH Patent void