DE3887443D1 - Azetidinylchinoloncarbonsäure und Ester. - Google Patents

Azetidinylchinoloncarbonsäure und Ester.

Info

Publication number
DE3887443D1
DE3887443D1 DE88309722T DE3887443T DE3887443D1 DE 3887443 D1 DE3887443 D1 DE 3887443D1 DE 88309722 T DE88309722 T DE 88309722T DE 3887443 T DE3887443 T DE 3887443T DE 3887443 D1 DE3887443 D1 DE 3887443D1
Authority
DE
Germany
Prior art keywords
alkyl
azetidinyl
amino
halo
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE88309722T
Other languages
English (en)
Other versions
DE3887443T2 (de
Inventor
Susumi Nakanishi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of DE3887443D1 publication Critical patent/DE3887443D1/de
Application granted granted Critical
Publication of DE3887443T2 publication Critical patent/DE3887443T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Quinoline Compounds (AREA)
DE88309722T 1987-10-26 1988-10-17 Azetidinylchinoloncarbonsäure und Ester. Expired - Fee Related DE3887443T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1987/002792 WO1989003828A1 (en) 1987-10-26 1987-10-26 Azetidinyl quinolone carboxylic acids and esters

Publications (2)

Publication Number Publication Date
DE3887443D1 true DE3887443D1 (de) 1994-03-10
DE3887443T2 DE3887443T2 (de) 1994-05-11

Family

ID=22202632

Family Applications (1)

Application Number Title Priority Date Filing Date
DE88309722T Expired - Fee Related DE3887443T2 (de) 1987-10-26 1988-10-17 Azetidinylchinoloncarbonsäure und Ester.

Country Status (19)

Country Link
US (1) US5039683A (de)
EP (1) EP0314362B1 (de)
JP (1) JPH01146879A (de)
KR (1) KR900006741B1 (de)
AT (1) ATE100805T1 (de)
AU (1) AU602431B2 (de)
DE (1) DE3887443T2 (de)
DK (1) DK591588A (de)
ES (1) ES2061680T3 (de)
FI (1) FI893048A (de)
HU (1) HU205105B (de)
IE (1) IE63284B1 (de)
IL (1) IL88086A (de)
MY (1) MY103436A (de)
NO (1) NO892616L (de)
NZ (1) NZ226689A (de)
PT (1) PT88837B (de)
WO (1) WO1989003828A1 (de)
ZA (1) ZA887927B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2634483B2 (fr) * 1987-12-29 1994-03-04 Esteve Labor Dr Derives des acides 7-(1-azetidinyl)-1,4-dihydro-4-oxoquinoleine-3-carboxyliques, leur preparation et leur application en tant que medicaments
US5173484A (en) * 1988-02-05 1992-12-22 Bayer Aktiengesellschaft Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them
EP0366189A3 (de) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Antimikrobielle Lactam-Quinolone
FR2654728B2 (fr) * 1989-03-16 1994-09-23 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament.
FR2644455B1 (fr) * 1989-03-16 1994-09-23 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicaments
FR2649106A2 (fr) * 1989-06-29 1991-01-04 Esteve Labor Dr Derives d'acides pyridone carboxyliques azetidinyl substitues, leur preparation et leur application en tant que medicament
NO177302C (no) * 1989-03-16 1995-08-23 Esteve Labor Dr Analogifremgangsmåte til fremstilling av terapeutisk aktive substituerte azetidinylkinolon(naftyridon)karboksylsyrederivater
FR2690161B1 (fr) * 1992-04-16 1995-06-30 Esteve Labor Dr Derives de pyridone azetidinyl substitues avec activite antimicrobienne.
US5885983A (en) * 1996-05-10 1999-03-23 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
WO2005019224A2 (en) * 2003-06-06 2005-03-03 Cadila Healthcare Limited Novel antiinfective compounds
WO2005026146A1 (en) * 2003-09-12 2005-03-24 Warner-Lambert Company Llc Azetidinyl quinolones as antibacterial agents

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4670444B1 (en) * 1980-09-03 1999-02-09 Bayer Ag and-naphthyridine-3-carboxylic acids and antibacte7-amino-1-cyclopropyl-4-oxo-1,4-dihydro-quinoline-rial agents containing these compounds
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
NZ208470A (en) * 1983-07-18 1988-06-30 Abbott Lab 6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid derivatives and antibacterial compositions containing such
JPS6089480A (ja) * 1983-10-21 1985-05-20 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体
JPS60126284A (ja) * 1983-12-09 1985-07-05 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体およびその塩
US4623650A (en) * 1984-12-06 1986-11-18 Pfizer Inc. Antibiotic derivatives of 7-phenyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids
JPS61137885A (ja) * 1984-12-08 1986-06-25 Dainippon Pharmaceut Co Ltd １，８−ナフチリジン誘導体、そのエステルおよびその塩
JPS61152682A (ja) * 1984-12-27 1986-07-11 Dainippon Pharmaceut Co Ltd ピリドンカルボン酸誘導体、そのエステルおよびその塩
JPS61282382A (ja) * 1985-06-06 1986-12-12 Dainippon Pharmaceut Co Ltd フエニル置換１，８−ナフチリジン誘導体、そのエステルおよびその塩
JPS62469A (ja) * 1985-06-27 1987-01-06 Dainippon Pharmaceut Co Ltd 新規キノロン誘導体、そのエステルおよびその塩
JPS6219883A (ja) * 1985-07-19 1987-01-28 Ricoh Co Ltd 色替え可能な現像装置
JPH0674260B2 (ja) * 1985-08-01 1994-09-21 大日本製薬株式会社 キノリン誘導体、そのエステルおよびその塩
JPS62215572A (ja) * 1986-03-17 1987-09-22 Kyorin Pharmaceut Co Ltd キノロンカルボン酸誘導体
EP0241206A3 (de) * 1986-03-31 1989-05-10 Sankyo Company Limited Chinolin-3-carbonsäurederivate, ihre Herstellung und Verwendung
JPH0689480A (ja) * 1992-09-09 1994-03-29 Ricoh Co Ltd 光磁気記録再生装置

Also Published As

Publication number Publication date
JPH01146879A (ja) 1989-06-08
HUT52497A (en) 1990-07-28
HU205105B (en) 1992-03-30
NO892616D0 (no) 1989-06-23
ZA887927B (en) 1990-06-27
WO1989003828A1 (en) 1989-05-05
IL88086A (en) 1997-01-10
ATE100805T1 (de) 1994-02-15
DK591588A (da) 1989-04-27
MY103436A (en) 1993-06-30
FI893048A0 (fi) 1989-06-21
IE63284B1 (en) 1995-04-05
NZ226689A (en) 1990-03-27
EP0314362A3 (en) 1989-10-18
KR890006616A (ko) 1989-06-14
NO892616L (no) 1989-06-23
KR900006741B1 (ko) 1990-09-20
DE3887443T2 (de) 1994-05-11
EP0314362B1 (de) 1994-01-26
EP0314362A2 (de) 1989-05-03
AU602431B2 (en) 1990-10-11
DK591588D0 (da) 1988-10-25
IL88086A0 (en) 1989-06-30
AU2432588A (en) 1988-10-25
ES2061680T3 (es) 1994-12-16
PT88837B (pt) 1993-01-29
IE883217L (en) 1989-04-26
FI893048A (fi) 1989-06-21
US5039683A (en) 1991-08-13

Similar Documents

Publication Publication Date Title
ATE100805T1 (de) Azetidinylchinoloncarbonsaeure und ester.
ES8604516A1 (es) Un derivado de dihidropiridina
DE3685248D1 (de) 7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel.
FR2725206B1 (fr) Nouvelles imidazolidines substituees par un heterocycle, leur procede et des intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
ES8602753A1 (es) Un procedimiento para la obtencion de agentes antibacteria- nos a base de acidos 7-amino-1-ciclopropil-6,8-difluor-1, 4-dihidro-4-oxo-3-quinolincarboxilicos
ATE159950T1 (de) N-alkyl-2-substituierte atp-analoge
LU88579I2 (fr) ATOVAQUONE et ses sels pharmaceutiquement acceptables (WELLVONE R)
HUT44523A (en) Process for producing new aromatic carboxamide derivatives and pharmaceutical compositions containing them as active components
DK705888A (da) Pyridazinonderivater
HUP9903584A2 (hu) Kinolinszármazékok NK3 antagonistákként alkalmazható sói
FR2346014A1 (fr) Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2047882A1 (en) Analgesic antiinflammatory 4-(2-alkoxy - phenylamino-quinolines and intermediates
FR2258840A1 (en) (4-Phenylpiperazino) alkyl esters - with analgesic activity for human and veterinary use
FR2116302A1 (en) 8-aminotheophyllines - with coronary - vasodilator bronchodilator diuretic, spasmolytic, antiinflammatory and analgesic activity
FR2244514A1 (en) 1,2-Dihydroquinoline derivs - useful as anti-inflammatories
NO963374D0 (no) Substituerte 4H-pyraner
FR2193822A1 (en) Trifluoromethoxy quinoline derivs - useful as inters in org. syntheses
FR2228779A1 (en) (4-Phenylpiperazino) alkyl esters - with analgesic activity for human and veterinary use
ES8604556A1 (es) Procedimiento para preparar derivados de flaveno y tioflave-no
FR2361893A2 (fr) Nouvelles oximes derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2226163A2 (en) 2-Amino-5-methyl-4-phenyl-1-pyrrolines - with antidepressant and antiarrhythmic activity
FR2361894A2 (fr) Nouvelles oximes derivees de l'acide 7-aminothiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
ES8609254A1 (es) Un procedimiento para preparar un derivado de piridinodicar-boxilato
ES8801125A1 (es) Procedimiento para la obtencion de medicamentos antiasmaticos que comprenden 5-sulfonil-1,4-dihidropiridinas como principio activo.
IT1104703B (it) Derivati di 2,3-difenil-cromone loro procedimento di preparazione e loro applicazione terapeutica

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee