IL236006A0 - Macrocyclic inhibitors of flavoviride viruses - Google Patents
Macrocyclic inhibitors of flavoviride virusesInfo
- Publication number
- IL236006A0 IL236006A0 IL236006A IL23600614A IL236006A0 IL 236006 A0 IL236006 A0 IL 236006A0 IL 236006 A IL236006 A IL 236006A IL 23600614 A IL23600614 A IL 23600614A IL 236006 A0 IL236006 A0 IL 236006A0
- Authority
- IL
- Israel
- Prior art keywords
- flaviviridae viruses
- macrocyclic inhibitors
- macrocyclic
- inhibitors
- flaviviridae
- Prior art date
Links
- 241000710781 Flaviviridae Species 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/504—Pyridazines; Hydrogenated pyridazines forming part of bridged ring systems
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- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7068—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid
- A61K31/7072—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines having oxo groups directly attached to the pyrimidine ring, e.g. cytidine, cytidylic acid having two oxo groups directly attached to the pyrimidine ring, e.g. uridine, uridylic acid, thymidine, zidovudine
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Oncology (AREA)
- Zoology (AREA)
- Microbiology (AREA)
- Mycology (AREA)
- Biotechnology (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201261657553P | 2012-06-08 | 2012-06-08 | |
PCT/US2013/044809 WO2013185090A1 (en) | 2012-06-08 | 2013-06-07 | Macrocyclic inhibitors of flaviviridae viruses |
Publications (1)
Publication Number | Publication Date |
---|---|
IL236006A0 true IL236006A0 (en) | 2015-01-29 |
Family
ID=48670106
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL236006A IL236006A0 (en) | 2012-06-08 | 2014-11-30 | Macrocyclic inhibitors of flavoviride viruses |
Country Status (21)
Country | Link |
---|---|
US (3) | US9090653B2 (enEXAMPLES) |
EP (1) | EP2859009B1 (enEXAMPLES) |
JP (1) | JP6209600B2 (enEXAMPLES) |
KR (1) | KR20150040266A (enEXAMPLES) |
CN (1) | CN104662033B (enEXAMPLES) |
AU (1) | AU2013271413B2 (enEXAMPLES) |
BR (1) | BR112014030649A2 (enEXAMPLES) |
CA (1) | CA2875718A1 (enEXAMPLES) |
EA (1) | EA201492205A1 (enEXAMPLES) |
ES (1) | ES2656087T3 (enEXAMPLES) |
HK (1) | HK1210483A1 (enEXAMPLES) |
IL (1) | IL236006A0 (enEXAMPLES) |
IN (1) | IN2014MN02658A (enEXAMPLES) |
MX (1) | MX2014014768A (enEXAMPLES) |
NO (1) | NO2887898T3 (enEXAMPLES) |
NZ (2) | NZ703066A (enEXAMPLES) |
PL (1) | PL2859009T3 (enEXAMPLES) |
PT (1) | PT2859009T (enEXAMPLES) |
SG (1) | SG11201408045UA (enEXAMPLES) |
SI (1) | SI2859009T1 (enEXAMPLES) |
WO (1) | WO2013185090A1 (enEXAMPLES) |
Families Citing this family (68)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR091279A1 (es) | 2012-06-08 | 2015-01-21 | Gilead Sciences Inc | Inhibidores macrociclicos de virus flaviviridae |
BR112014030630A2 (pt) | 2012-06-08 | 2017-06-27 | Gilead Sciences Inc | inibidores macrocíclicos de vírus flaviviridae |
US9090653B2 (en) | 2012-06-08 | 2015-07-28 | Gilead Sciences, Inc. | Macrocyclic inhibitors of flaviviridae viruses |
RU2683648C2 (ru) * | 2014-12-24 | 2019-04-01 | ЭлДжи КЕМ, ЛТД. | Биарильное производное в качестве агониста gpr120 |
BR112017013858A2 (pt) | 2014-12-26 | 2018-02-27 | Univ Emory | n4-hidroxicitidina e derivados e usos antivirais relacionados aos mesmos |
HUE050029T2 (hu) | 2015-03-04 | 2020-11-30 | Gilead Sciences Inc | 4,6-Diamino-pirido[3,2-d]pirimidin-származékok és alkalmazásuk toll-szerû receptorok modulátoraként |
CA2995004A1 (en) | 2015-08-26 | 2017-03-02 | Gilead Sciences, Inc. | Deuterated toll-like receptor modulators |
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