IL208838A0 - Purine pi3k inhibitor compounds and methods of use - Google Patents

Purine pi3k inhibitor compounds and methods of use

Info

Publication number
IL208838A0
IL208838A0 IL208838A IL20883810A IL208838A0 IL 208838 A0 IL208838 A0 IL 208838A0 IL 208838 A IL208838 A IL 208838A IL 20883810 A IL20883810 A IL 20883810A IL 208838 A0 IL208838 A0 IL 208838A0
Authority
IL
Israel
Prior art keywords
purine
methods
inhibitor compounds
pi3k inhibitor
pi3k
Prior art date
Application number
IL208838A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche, Genentech Inc filed Critical Hoffmann La Roche
Publication of IL208838A0 publication Critical patent/IL208838A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/26Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32Nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL208838A 2008-05-30 2010-10-20 Purine pi3k inhibitor compounds and methods of use IL208838A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5755908P 2008-05-30 2008-05-30
PCT/US2009/045603 WO2009146406A1 (en) 2008-05-30 2009-05-29 Purine pi3k inhibitor compounds and methods of use

Publications (1)

Publication Number Publication Date
IL208838A0 true IL208838A0 (en) 2011-01-31

Family

ID=41017038

Family Applications (1)

Application Number Title Priority Date Filing Date
IL208838A IL208838A0 (en) 2008-05-30 2010-10-20 Purine pi3k inhibitor compounds and methods of use

Country Status (14)

Country Link
US (2) US8158624B2 (OSRAM)
EP (1) EP2279188B1 (OSRAM)
JP (1) JP2011521968A (OSRAM)
KR (1) KR20110042153A (OSRAM)
CN (1) CN102105474B (OSRAM)
AU (1) AU2009251291B2 (OSRAM)
BR (1) BRPI0909614A2 (OSRAM)
CA (1) CA2721851A1 (OSRAM)
ES (1) ES2533788T3 (OSRAM)
IL (1) IL208838A0 (OSRAM)
MX (1) MX2010012583A (OSRAM)
RU (1) RU2509081C2 (OSRAM)
WO (1) WO2009146406A1 (OSRAM)
ZA (1) ZA201007524B (OSRAM)

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CN103804380B (zh) * 2014-01-24 2016-05-18 温州医科大学 以IKK-β为靶点的2-氨基-8-取代鸟嘌呤衍生物、应用及其制备方法
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CN110036109A (zh) 2016-12-02 2019-07-19 第一三共株式会社 新颖的内-β-N-乙酰基氨基葡糖苷酶
SG11202103118PA (en) * 2018-09-27 2021-04-29 Shanghai Yingli Pharmaceutical Co Ltd Crystal form of morpholino quinazoline compound, preparation method therefor and use thereof
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CN111875606B (zh) * 2020-07-20 2023-04-07 武汉工程大学 一种基于虚拟对接获得的嘌呤类化合物及其制备方法和应用
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Also Published As

Publication number Publication date
ZA201007524B (en) 2012-01-25
ES2533788T3 (es) 2015-04-14
CN102105474A (zh) 2011-06-22
BRPI0909614A2 (pt) 2015-09-22
US20120135988A1 (en) 2012-05-31
US8445487B2 (en) 2013-05-21
CN102105474B (zh) 2014-01-08
AU2009251291B2 (en) 2013-05-02
AU2009251291A1 (en) 2009-12-03
WO2009146406A1 (en) 2009-12-03
RU2010154428A (ru) 2012-07-10
CA2721851A1 (en) 2009-12-03
KR20110042153A (ko) 2011-04-25
EP2279188A1 (en) 2011-02-02
MX2010012583A (es) 2011-02-24
RU2509081C2 (ru) 2014-03-10
US8158624B2 (en) 2012-04-17
JP2011521968A (ja) 2011-07-28
US20090318411A1 (en) 2009-12-24
EP2279188B1 (en) 2015-01-28

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