IL195851A0 - Modulators of metabolism and the treatment of disorders related thereto - Google Patents

Modulators of metabolism and the treatment of disorders related thereto

Info

Publication number
IL195851A0
IL195851A0 IL195851A IL19585108A IL195851A0 IL 195851 A0 IL195851 A0 IL 195851A0 IL 195851 A IL195851 A IL 195851A IL 19585108 A IL19585108 A IL 19585108A IL 195851 A0 IL195851 A0 IL 195851A0
Authority
IL
Israel
Prior art keywords
modulators
metabolism
treatment
disorders related
disorders
Prior art date
Application number
IL195851A
Other languages
English (en)
Original Assignee
Arena Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arena Pharm Inc filed Critical Arena Pharm Inc
Publication of IL195851A0 publication Critical patent/IL195851A0/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL195851A 2006-07-06 2008-12-10 Modulators of metabolism and the treatment of disorders related thereto IL195851A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81927806P 2006-07-06 2006-07-06
PCT/US2007/015670 WO2008005569A2 (en) 2006-07-06 2007-07-05 Modulators of metabolism and the treatment of disorders related thereto

Publications (1)

Publication Number Publication Date
IL195851A0 true IL195851A0 (en) 2009-09-01

Family

ID=38895258

Family Applications (1)

Application Number Title Priority Date Filing Date
IL195851A IL195851A0 (en) 2006-07-06 2008-12-10 Modulators of metabolism and the treatment of disorders related thereto

Country Status (30)

Country Link
US (1) US20090286816A1 (enExample)
EP (1) EP2051976B1 (enExample)
JP (1) JP2009542699A (enExample)
KR (1) KR20090029781A (enExample)
CN (1) CN101484441A (enExample)
AR (1) AR061968A1 (enExample)
AT (1) ATE469145T1 (enExample)
AU (1) AU2007269571A1 (enExample)
BR (1) BRPI0713998A2 (enExample)
CA (1) CA2656623A1 (enExample)
CL (1) CL2007001971A1 (enExample)
CO (1) CO6160319A2 (enExample)
CR (1) CR10537A (enExample)
DE (1) DE602007006815D1 (enExample)
DK (1) DK2051976T3 (enExample)
EA (1) EA200970088A1 (enExample)
EC (1) ECSP099037A (enExample)
ES (1) ES2344965T3 (enExample)
GT (1) GT200800306A (enExample)
IL (1) IL195851A0 (enExample)
MA (1) MA30602B1 (enExample)
MX (1) MX2008016253A (enExample)
NO (1) NO20090591L (enExample)
PE (1) PE20080519A1 (enExample)
SV (1) SV2009003146A (enExample)
TN (1) TNSN08533A1 (enExample)
TW (1) TW200811147A (enExample)
UY (1) UY30467A1 (enExample)
WO (1) WO2008005569A2 (enExample)
ZA (1) ZA200900055B (enExample)

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US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
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TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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JP5941916B2 (ja) 2010-09-22 2016-06-29 アリーナ ファーマシューティカルズ, インコーポレイテッド Gpr119レセプターのモジュレーターおよびそれに関連する障害の処置
AR083878A1 (es) 2010-11-15 2013-03-27 Boehringer Ingelheim Int Terapia antidiabetica vasoprotectora y cardioprotectora, linagliptina, metodo de tratamiento
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EP2718279B1 (en) 2011-06-09 2016-08-10 Rhizen Pharmaceuticals SA Novel compounds as modulators of gpr-119
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Also Published As

Publication number Publication date
GT200800306A (es) 2009-04-20
DK2051976T3 (da) 2010-09-20
KR20090029781A (ko) 2009-03-23
MX2008016253A (es) 2009-02-25
CA2656623A1 (en) 2008-01-10
ES2344965T3 (es) 2010-09-10
TW200811147A (en) 2008-03-01
CR10537A (es) 2009-01-27
MA30602B1 (fr) 2009-07-01
CL2007001971A1 (es) 2008-01-25
AR061968A1 (es) 2008-08-10
UY30467A1 (es) 2008-02-29
EA200970088A1 (ru) 2009-06-30
ZA200900055B (en) 2009-12-30
ECSP099037A (es) 2009-02-27
EP2051976B1 (en) 2010-05-26
HK1128921A1 (en) 2009-11-13
SV2009003146A (es) 2009-11-04
AU2007269571A1 (en) 2008-01-10
TNSN08533A1 (en) 2010-04-14
BRPI0713998A2 (pt) 2012-11-20
CN101484441A (zh) 2009-07-15
WO2008005569A3 (en) 2008-04-10
JP2009542699A (ja) 2009-12-03
EP2051976A2 (en) 2009-04-29
ATE469145T1 (de) 2010-06-15
CO6160319A2 (es) 2010-05-20
WO2008005569A2 (en) 2008-01-10
DE602007006815D1 (de) 2010-07-08
US20090286816A1 (en) 2009-11-19
NO20090591L (no) 2009-02-06
PE20080519A1 (es) 2008-05-16

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