IL154272A0 - The use of benzylideneaminoguanidines and hydroxyguanidines as melanocortin receptor ligands - Google Patents

The use of benzylideneaminoguanidines and hydroxyguanidines as melanocortin receptor ligands

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Publication number
IL154272A0
IL154272A0 IL15427201A IL15427201A IL154272A0 IL 154272 A0 IL154272 A0 IL 154272A0 IL 15427201 A IL15427201 A IL 15427201A IL 15427201 A IL15427201 A IL 15427201A IL 154272 A0 IL154272 A0 IL 154272A0
Authority
IL
Israel
Prior art keywords
benzylideneaminoguanidines
hydroxyguanidines
receptor ligands
melanocortin receptor
melanocortin
Prior art date
Application number
IL15427201A
Other languages
English (en)
Original Assignee
Melacure Therapeutics Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Melacure Therapeutics Ab filed Critical Melacure Therapeutics Ab
Publication of IL154272A0 publication Critical patent/IL154272A0/xx

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    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C281/00Derivatives of carbonic acid containing functional groups covered by groups C07C269/00 - C07C279/00 in which at least one nitrogen atom of these functional groups is further bound to another nitrogen atom not being part of a nitro or nitroso group
    • C07C281/16Compounds containing any of the groups, e.g. aminoguanidine
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    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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IL15427201A 2000-08-07 2001-08-07 The use of benzylideneaminoguanidines and hydroxyguanidines as melanocortin receptor ligands IL154272A0 (en)

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GB0019357A GB0019357D0 (en) 2000-08-07 2000-08-07 Novel phenyl guanidines
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US7060711B2 (en) 2001-10-25 2006-06-13 Biofrontera Bioscience Gmbh Derivatives of 4-(thio- or selenoxanthene-9-ylidene)-piperidine or acridine and its use as a selective 5-HT2B receptor antagonist
GB0622826D0 (en) * 2006-11-15 2006-12-27 Acurepharma Ab Novel amides acting on the adenosine receptors
GB0624987D0 (en) * 2006-12-14 2007-01-24 Acure Pharma Ab Novel aminoguanidines as melanocortin receptor ligands

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JP5654190B2 (ja) 2015-01-14
GB0019357D0 (en) 2000-09-27
KR20030022371A (ko) 2003-03-15
IL154272A (en) 2010-12-30
MXPA03001072A (es) 2004-03-10
JP5683396B2 (ja) 2015-03-11
US9227927B2 (en) 2016-01-05
US20120178820A1 (en) 2012-07-12
AU2001276522A1 (en) 2002-02-18
US20040024060A1 (en) 2004-02-05
BR0113053A (pt) 2003-07-08
US8410174B2 (en) 2013-04-02
US8148429B2 (en) 2012-04-03
US20070231267A1 (en) 2007-10-04
CA2417098A1 (fr) 2002-02-14
US20070088085A1 (en) 2007-04-19
WO2002011715A2 (fr) 2002-02-14
KR100929363B1 (ko) 2009-12-02
EP1313461A2 (fr) 2003-05-28
JP2004505912A (ja) 2004-02-26
ZA200300829B (en) 2004-02-25
US8309609B2 (en) 2012-11-13
JP2011246471A (ja) 2011-12-08
US20130295009A1 (en) 2013-11-07
US20110015437A1 (en) 2011-01-20

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