IL149473A0 - Heterocyclic dihydropyrimidine derivatives and pharmaceutical compositions containing the same - Google Patents

Heterocyclic dihydropyrimidine derivatives and pharmaceutical compositions containing the same

Info

Publication number
IL149473A0
IL149473A0 IL14947300A IL14947300A IL149473A0 IL 149473 A0 IL149473 A0 IL 149473A0 IL 14947300 A IL14947300 A IL 14947300A IL 14947300 A IL14947300 A IL 14947300A IL 149473 A0 IL149473 A0 IL 149473A0
Authority
IL
Israel
Prior art keywords
same
pharmaceutical compositions
compositions containing
dihydropyrimidine derivatives
heterocyclic
Prior art date
Application number
IL14947300A
Other languages
English (en)
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of IL149473A0 publication Critical patent/IL149473A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Hospice & Palliative Care (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
IL14947300A 1999-12-06 2000-12-04 Heterocyclic dihydropyrimidine derivatives and pharmaceutical compositions containing the same IL149473A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16909199P 1999-12-06 1999-12-06
US23603700P 2000-09-28 2000-09-28
PCT/US2000/032785 WO2001040231A1 (en) 1999-12-06 2000-12-04 Heterocyclic dihydropyrimidines as potassium channel inhibitors

Publications (1)

Publication Number Publication Date
IL149473A0 true IL149473A0 (en) 2002-11-10

Family

ID=26864749

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14947300A IL149473A0 (en) 1999-12-06 2000-12-04 Heterocyclic dihydropyrimidine derivatives and pharmaceutical compositions containing the same
IL149473A IL149473A (en) 1999-12-06 2002-05-05 History of tricyclic dihydropyrimidine and pharmaceutical preparations containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL149473A IL149473A (en) 1999-12-06 2002-05-05 History of tricyclic dihydropyrimidine and pharmaceutical preparations containing them

Country Status (25)

Country Link
US (3) US6706720B2 (xx)
EP (1) EP1237891B1 (xx)
JP (1) JP2004507442A (xx)
KR (1) KR20020060255A (xx)
CN (1) CN1407985A (xx)
AR (1) AR029457A1 (xx)
AT (1) ATE526329T1 (xx)
AU (1) AU781862B2 (xx)
BR (1) BR0016166A (xx)
CA (1) CA2393809C (xx)
CO (1) CO5570109A1 (xx)
CZ (1) CZ20021949A3 (xx)
HK (1) HK1048808A1 (xx)
HU (1) HUP0301834A3 (xx)
IL (2) IL149473A0 (xx)
MX (1) MXPA02005533A (xx)
MY (1) MY125533A (xx)
NO (1) NO323588B1 (xx)
NZ (1) NZ518663A (xx)
PE (1) PE20011029A1 (xx)
PL (1) PL364926A1 (xx)
RU (1) RU2296766C2 (xx)
TW (1) TWI291465B (xx)
UY (1) UY26472A1 (xx)
WO (1) WO2001040231A1 (xx)

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GB9901691D0 (en) 1999-01-26 1999-03-17 Cerebrus Ltd Chemical compounds
MY125533A (en) * 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
SK18412002A3 (sk) * 2000-06-30 2003-06-03 Wyeth Použitie substituovaných triazolopyrimidínových derivátov a farmaceutický prostriedok s ich obsahom
DE60135780D1 (de) * 2000-12-25 2008-10-23 Daiichi Sankyo Co Ltd Aspirin enthaltende medizinische zusammensetzungen
TWI243164B (en) 2001-02-13 2005-11-11 Aventis Pharma Gmbh Acylated indanyl amines and their use as pharmaceuticals
EP1956020A3 (en) * 2001-05-05 2008-08-20 Smithkline Beecham Plc 1-[2-(heterocyclyl-aminomethyl)-piperidin-1-YL]-1-(2-methyl-5-phenyl-heterocyclyl)-methanone derivatives and related compounds as orexin-1 antagonists for the treatment of obesity
EP1435955A2 (en) * 2001-05-05 2004-07-14 SmithKline Beecham P.L.C. N-aroyl cyclic amine derivatives as orexin receptor antagonists
US7139344B2 (en) * 2001-05-16 2006-11-21 Lexmark International, Inc. Method and apparatus for effecting synchronous pulse generation for use in variable speed serial communications
ES2266549T3 (es) * 2001-06-28 2007-03-01 Smithkline Beecham Plc Derivados de n-aroil-amina ciclicos como antagonistas del receptor de orexina.
GB0115862D0 (en) * 2001-06-28 2001-08-22 Smithkline Beecham Plc Compounds
CH1427415H1 (de) 2001-09-21 2023-12-21 Bristol Myers Squibb Holdings Ireland Lactamhaltige verbindungen und ihre derivate als faktor-xa-hemmer
US6833371B2 (en) * 2001-11-01 2004-12-21 Icagen, Inc. Pyrazolopyrimidines
US7435824B2 (en) 2002-04-19 2008-10-14 Bristol-Myers Squibb Company Prodrugs of potassium channel inhibitors
JP4602076B2 (ja) * 2002-06-04 2010-12-22 ネオジェネシス ファーマシューティカルズ インコーポレイテッド 抗ウイルス剤としてのピラゾロ［１，５ａ］ピリミジン化合物
US7169771B2 (en) 2003-02-06 2007-01-30 Bristol-Myers Squibb Company Thiazolyl-based compounds useful as kinase inhibitors
US6846836B2 (en) 2003-04-18 2005-01-25 Bristol-Myers Squibb Company N-substituted phenylurea inhibitors of mitochondrial F1F0 ATP hydrolase
RU2342365C2 (ru) 2003-05-01 2008-12-27 Бристол-Маерс Сквибб Компани Арилзамещенные пиразоламиды в качестве ингибиторов киназ
GB0315950D0 (en) 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
US20050187278A1 (en) * 2003-08-28 2005-08-25 Pharmacia Corporation Treatment or prevention of vascular disorders with Cox-2 inhibitors in combination with cyclic AMP-specific phosphodiesterase inhibitors
EP1677791A4 (en) * 2003-10-31 2007-08-15 Takeda Pharmaceutical NITROGENIC CONDENSED HETEROCYCLIC COMPOUNDS
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
EP1750862B1 (en) * 2004-06-04 2011-01-05 Teva Pharmaceutical Industries Ltd. Pharmaceutical composition containing irbesartan
GB0412986D0 (en) 2004-06-10 2004-07-14 Xention Discovery Ltd Compounds
US7253167B2 (en) * 2004-06-30 2007-08-07 Bristol-Myers Squibb Company Tricyclic-heteroaryl compounds useful as kinase inhibitors
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HUP0301834A2 (hu) 2003-09-29
AU781862B2 (en) 2005-06-16
NZ518663A (en) 2004-11-26
RU2002118622A (ru) 2004-01-10
MY125533A (en) 2006-08-30
BR0016166A (pt) 2003-06-24
US20070099899A1 (en) 2007-05-03
EP1237891A1 (en) 2002-09-11
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US6706720B2 (en) 2004-03-16
US20030022890A1 (en) 2003-01-30
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AR029457A1 (es) 2003-07-02
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IL149473A (en) 2009-05-04
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