IL141785A0 - A pharmaceutical composition containing an ap2 inhibitor - Google Patents

A pharmaceutical composition containing an ap2 inhibitor

Info

Publication number
IL141785A0
IL141785A0 IL14178599A IL14178599A IL141785A0 IL 141785 A0 IL141785 A0 IL 141785A0 IL 14178599 A IL14178599 A IL 14178599A IL 14178599 A IL14178599 A IL 14178599A IL 141785 A0 IL141785 A0 IL 141785A0
Authority
IL
Israel
Prior art keywords
inhibitor
pharmaceutical composition
composition containing
pravastatin
employing
Prior art date
Application number
IL14178599A
Other languages
English (en)
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22280975&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL141785(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of IL141785A0 publication Critical patent/IL141785A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL14178599A 1998-09-17 1999-09-13 A pharmaceutical composition containing an ap2 inhibitor IL141785A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10067798P 1998-09-17 1998-09-17
PCT/US1999/021069 WO2000015230A1 (en) 1998-09-17 1999-09-13 METHOD FOR TREATING ATHEROSCLEROSIS EMPLOYING AN aP2 INHIBITOR AND COMBINATION

Publications (1)

Publication Number Publication Date
IL141785A0 true IL141785A0 (en) 2002-03-10

Family

ID=22280975

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14178599A IL141785A0 (en) 1998-09-17 1999-09-13 A pharmaceutical composition containing an ap2 inhibitor
IL14178699A IL141786A0 (en) 1998-09-17 1999-09-13 A pharmaceutical composition for treating diabetes containing an ap2 inhibitor

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL14178699A IL141786A0 (en) 1998-09-17 1999-09-13 A pharmaceutical composition for treating diabetes containing an ap2 inhibitor

Country Status (30)

Country Link
US (1) US20020035064A1 (cs)
EP (2) EP1113801A4 (cs)
JP (2) JP2002524518A (cs)
KR (2) KR20010075150A (cs)
CN (2) CN1319012A (cs)
AT (1) ATE406898T1 (cs)
AU (2) AU754488B2 (cs)
BG (2) BG105432A (cs)
BR (2) BR9913833A (cs)
CA (2) CA2344300A1 (cs)
CO (2) CO5130025A1 (cs)
CZ (2) CZ2001965A3 (cs)
DE (1) DE69939481D1 (cs)
EE (2) EE200100155A (cs)
ES (1) ES2311306T3 (cs)
GE (2) GEP20033044B (cs)
HU (2) HUP0104240A2 (cs)
ID (2) ID27833A (cs)
IL (2) IL141785A0 (cs)
LT (2) LT4870B (cs)
LV (2) LV12686B (cs)
NO (2) NO20011351L (cs)
NZ (2) NZ510209A (cs)
PE (2) PE20001056A1 (cs)
PL (2) PL346660A1 (cs)
SK (1) SK3202001A3 (cs)
TR (2) TR200100773T2 (cs)
UY (2) UY25714A1 (cs)
WO (2) WO2000015230A1 (cs)
ZA (2) ZA200207433B (cs)

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AU2005201289B2 (en) * 1999-02-12 2008-04-17 President And Fellows Of Harvard College Inhibiting formation of atherosclerotic lesions
US6548529B1 (en) 1999-04-05 2003-04-15 Bristol-Myers Squibb Company Heterocyclic containing biphenyl aP2 inhibitors and method
US6586438B2 (en) 1999-11-03 2003-07-01 Bristol-Myers Squibb Co. Antidiabetic formulation and method
CA2396596A1 (en) 2000-01-28 2001-08-02 Bristol-Myers Squibb Company Tetrahydropyrimidone inhibitors of fatty acid binding protein and method
AU2002237664A1 (en) * 2000-11-20 2002-05-27 Bristol-Myers Squibb Company Pyridone derivatives as AP2 inhibitors
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WO2003006023A1 (en) 2001-07-13 2003-01-23 Bristol-Myers Squibb Company Pyrazinone inhibitors of fatty acid binding protein and method
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EP1443919A4 (en) 2001-11-16 2006-03-22 Bristol Myers Squibb Co DOUBLE INHIBITORS OF THE FATTY ACID BINDING PROTEIN OF THE ADIPOCYTES AND THE FATTY ACID BINDING PROTEIN OF KERATINOCYTES
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CA3184282A1 (en) 2020-06-27 2021-12-30 Emre Koyuncu Composition of compounds that modulate cell metabolism and methods of use
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Also Published As

Publication number Publication date
BG105431A (en) 2001-12-29
IL141786A0 (en) 2002-03-10
AU755563B2 (en) 2002-12-12
CO5130026A1 (es) 2002-02-27
CN1319012A (zh) 2001-10-24
DE69939481D1 (de) 2008-10-16
LT2001023A (en) 2001-08-27
CO5130025A1 (es) 2002-02-27
NO20011351D0 (no) 2001-03-16
EP1113801A1 (en) 2001-07-11
ES2311306T3 (es) 2009-02-01
TR200100774T2 (tr) 2001-12-21
HUP0104240A2 (hu) 2002-03-28
EE200100154A (et) 2002-12-16
ATE406898T1 (de) 2008-09-15
BR9913833A (pt) 2001-05-29
PL346661A1 (en) 2002-02-25
LV12687B (lv) 2001-10-20
JP2002524517A (ja) 2002-08-06
CZ2001965A3 (cs) 2002-02-13
NO20011352L (no) 2001-05-11
PL346660A1 (en) 2002-02-25
NZ510207A (en) 2003-08-29
EE04356B1 (et) 2004-10-15
CN1317970A (zh) 2001-10-17
AU6143799A (en) 2000-04-03
CA2344309A1 (en) 2000-03-23
EE200100155A (et) 2002-08-15
CA2344300A1 (en) 2000-03-23
BG105432A (en) 2001-12-29
NO20011352D0 (no) 2001-03-16
NZ510209A (en) 2003-07-25
CZ2001964A3 (cs) 2002-01-16
KR20010079842A (ko) 2001-08-22
KR20010075150A (ko) 2001-08-09
GEP20033044B (en) 2003-08-25
HUP0104108A2 (hu) 2002-03-28
EP1121129B1 (en) 2008-09-03
AU6387799A (en) 2000-04-03
LT4870B (lt) 2001-12-27
ID27833A (id) 2001-04-26
EP1113801A4 (en) 2002-10-02
EP1121129A4 (en) 2002-10-16
LT2001022A (en) 2001-08-27
PE20001056A1 (es) 2000-12-24
GEP20033045B (en) 2003-08-25
UY25713A1 (es) 2001-08-27
AU754488B2 (en) 2002-11-14
ZA200207430B (en) 2003-09-16
US20020035064A1 (en) 2002-03-21
LV12686A (en) 2001-07-20
NO20011351L (no) 2001-05-11
PE20001047A1 (es) 2000-12-24
EP1121129A1 (en) 2001-08-08
LV12687A (en) 2001-07-20
JP2002524518A (ja) 2002-08-06
BR9913831A (pt) 2001-05-29
WO2000015229A1 (en) 2000-03-23
TR200100773T2 (tr) 2001-07-23
ZA200207433B (en) 2003-10-27
SK3202001A3 (en) 2002-04-04
LT4871B (lt) 2001-12-27
LV12686B (lv) 2001-10-20
ID28450A (id) 2001-05-24
UY25714A1 (es) 2001-08-27
WO2000015230A1 (en) 2000-03-23

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