ID27833A - METODA UNTUK MENGOBATI ATEROSKLEROSIS DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA - Google Patents

METODA UNTUK MENGOBATI ATEROSKLEROSIS DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA

Info

Publication number
ID27833A
ID27833A IDW20010626A ID20010626A ID27833A ID 27833 A ID27833 A ID 27833A ID W20010626 A IDW20010626 A ID W20010626A ID 20010626 A ID20010626 A ID 20010626A ID 27833 A ID27833 A ID 27833A
Authority
ID
Indonesia
Prior art keywords
aterosclelerosis
inhibitors
combinations
treatment
methods
Prior art date
Application number
IDW20010626A
Other languages
English (en)
Indonesian (id)
Inventor
Jeffry A Robl
Rex A Parker
Scott A Biller
Haris Jamil
Bruce L Jacobson
Krishna Kudukula
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22280975&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID27833(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ID27833A publication Critical patent/ID27833A/id

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/4211,3-Oxazoles, e.g. pemoline, trimethadione
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50Pyridazines; Hydrogenated pyridazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Electrical Discharge Machining, Electrochemical Machining, And Combined Machining (AREA)
  • Steroid Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IDW20010626A 1998-09-17 1999-09-13 METODA UNTUK MENGOBATI ATEROSKLEROSIS DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA ID27833A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10067798P 1998-09-17 1998-09-17

Publications (1)

Publication Number Publication Date
ID27833A true ID27833A (id) 2001-04-26

Family

ID=22280975

Family Applications (2)

Application Number Title Priority Date Filing Date
IDW20010626A ID27833A (id) 1998-09-17 1999-09-13 METODA UNTUK MENGOBATI ATEROSKLEROSIS DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA
IDW20010624A ID28450A (id) 1998-09-17 1999-09-13 METODA UNTUK MENGOBATI DIABETES DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA

Family Applications After (1)

Application Number Title Priority Date Filing Date
IDW20010624A ID28450A (id) 1998-09-17 1999-09-13 METODA UNTUK MENGOBATI DIABETES DENGAN MENGGUNAKAN INHIBITOR aP2 DAN KOMBINASINYA

Country Status (30)

Country Link
US (1) US20020035064A1 (cs)
EP (2) EP1113801A4 (cs)
JP (2) JP2002524518A (cs)
KR (2) KR20010075150A (cs)
CN (2) CN1317970A (cs)
AT (1) ATE406898T1 (cs)
AU (2) AU754488B2 (cs)
BG (2) BG105431A (cs)
BR (2) BR9913833A (cs)
CA (2) CA2344300A1 (cs)
CO (2) CO5130025A1 (cs)
CZ (2) CZ2001965A3 (cs)
DE (1) DE69939481D1 (cs)
EE (2) EE200100155A (cs)
ES (1) ES2311306T3 (cs)
GE (2) GEP20033044B (cs)
HU (2) HUP0104240A2 (cs)
ID (2) ID27833A (cs)
IL (2) IL141786A0 (cs)
LT (2) LT4870B (cs)
LV (2) LV12687B (cs)
NO (2) NO20011352L (cs)
NZ (2) NZ510209A (cs)
PE (2) PE20001056A1 (cs)
PL (2) PL346661A1 (cs)
SK (1) SK3202001A3 (cs)
TR (2) TR200100774T2 (cs)
UY (2) UY25714A1 (cs)
WO (2) WO2000015230A1 (cs)
ZA (2) ZA200207433B (cs)

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JP6223376B2 (ja) 2014-03-24 2017-11-01 花王株式会社 Gip上昇抑制剤の評価又は選択方法
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CA3066733A1 (en) 2017-06-09 2018-12-13 President And Fellows Of Harvard College Method to identify compounds useful to treat dysregulated lipogenesis, diabetes, and related disorders
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Also Published As

Publication number Publication date
US20020035064A1 (en) 2002-03-21
PE20001047A1 (es) 2000-12-24
CN1319012A (zh) 2001-10-24
DE69939481D1 (de) 2008-10-16
WO2000015230A1 (en) 2000-03-23
LT2001023A (en) 2001-08-27
KR20010079842A (ko) 2001-08-22
LV12687B (lv) 2001-10-20
BG105431A (en) 2001-12-29
PE20001056A1 (es) 2000-12-24
AU755563B2 (en) 2002-12-12
UY25713A1 (es) 2001-08-27
NO20011351L (no) 2001-05-11
JP2002524517A (ja) 2002-08-06
SK3202001A3 (en) 2002-04-04
CA2344309A1 (en) 2000-03-23
NZ510207A (en) 2003-08-29
EP1113801A1 (en) 2001-07-11
IL141785A0 (en) 2002-03-10
BR9913833A (pt) 2001-05-29
GEP20033045B (en) 2003-08-25
UY25714A1 (es) 2001-08-27
ID28450A (id) 2001-05-24
EP1121129A1 (en) 2001-08-08
PL346660A1 (en) 2002-02-25
CO5130025A1 (es) 2002-02-27
IL141786A0 (en) 2002-03-10
WO2000015229A1 (en) 2000-03-23
EP1121129B1 (en) 2008-09-03
LV12686A (en) 2001-07-20
EE200100155A (et) 2002-08-15
NO20011352D0 (no) 2001-03-16
ATE406898T1 (de) 2008-09-15
ES2311306T3 (es) 2009-02-01
CZ2001964A3 (cs) 2002-01-16
LT4871B (lt) 2001-12-27
LV12686B (lv) 2001-10-20
EE200100154A (et) 2002-12-16
ZA200207433B (en) 2003-10-27
AU754488B2 (en) 2002-11-14
EP1121129A4 (en) 2002-10-16
PL346661A1 (en) 2002-02-25
CN1317970A (zh) 2001-10-17
EE04356B1 (et) 2004-10-15
AU6387799A (en) 2000-04-03
ZA200207430B (en) 2003-09-16
BR9913831A (pt) 2001-05-29
CA2344300A1 (en) 2000-03-23
TR200100774T2 (tr) 2001-12-21
GEP20033044B (en) 2003-08-25
CZ2001965A3 (cs) 2002-02-13
LT4870B (lt) 2001-12-27
BG105432A (en) 2001-12-29
EP1113801A4 (en) 2002-10-02
NO20011351D0 (no) 2001-03-16
HUP0104108A2 (hu) 2002-03-28
TR200100773T2 (tr) 2001-07-23
NZ510209A (en) 2003-07-25
JP2002524518A (ja) 2002-08-06
CO5130026A1 (es) 2002-02-27
HUP0104240A2 (hu) 2002-03-28
KR20010075150A (ko) 2001-08-09
AU6143799A (en) 2000-04-03
LT2001022A (en) 2001-08-27
NO20011352L (no) 2001-05-11
LV12687A (en) 2001-07-20

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