IL122345A0 - Benzamide derivatives their use as vasopressin antagonists processes for the preparation thereof and pharmaceutical compositions containing the same - Google Patents

Benzamide derivatives their use as vasopressin antagonists processes for the preparation thereof and pharmaceutical compositions containing the same

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Publication number
IL122345A0
IL122345A0 IL12234596A IL12234596A IL122345A0 IL 122345 A0 IL122345 A0 IL 122345A0 IL 12234596 A IL12234596 A IL 12234596A IL 12234596 A IL12234596 A IL 12234596A IL 122345 A0 IL122345 A0 IL 122345A0
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processes
preparation
pharmaceutical compositions
same
compositions containing
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IL12234596A
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Fujisawa Pharmaceutical Co
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    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
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    • C07C237/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
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    • A61K31/16—Amides, e.g. hydroxamic acids
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    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/205—Radicals derived from carbonic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
    • C07D295/215—Radicals derived from nitrogen analogues of carbonic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/28—Nitrogen atoms
    • C07D295/32—Nitrogen atoms acylated with carboxylic or carbonic acids, or their nitrogen or sulfur analogues

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IL12234596A 1995-06-09 1996-06-06 Benzamide derivatives their use as vasopressin antagonists processes for the preparation thereof and pharmaceutical compositions containing the same IL122345A0 (en)

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GBGB9511694.3A GB9511694D0 (en) 1995-06-09 1995-06-09 Benzamide derivatives
PCT/JP1996/001533 WO1996041795A1 (fr) 1995-06-09 1996-06-06 Derives de type benzamide et leur utilisation comme antagonistes de la vasopressine

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JP (2) JP4042160B2 (fr)
KR (1) KR19990022448A (fr)
CN (1) CN1192729A (fr)
AR (1) AR003005A1 (fr)
AT (1) ATE205185T1 (fr)
AU (1) AU5911096A (fr)
CA (1) CA2223869A1 (fr)
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EA (1) EA199800051A1 (fr)
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GB (1) GB9511694D0 (fr)
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TR (1) TR199600488A2 (fr)
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AR003005A1 (es) 1998-05-27
GB9511694D0 (en) 1995-08-02
GR3036881T3 (en) 2002-01-31
HUP9802694A3 (en) 1999-03-29
EA199800051A1 (ru) 1998-08-27
CN1192729A (zh) 1998-09-09
ES2159738T3 (es) 2001-10-16
HUP9802694A1 (hu) 1999-02-01
US6054457A (en) 2000-04-25
JP2008074855A (ja) 2008-04-03
DE69615025T2 (de) 2002-03-21
ZA964895B (en) 1996-12-12
JP4042160B2 (ja) 2008-02-06
PT832061E (pt) 2002-02-28
TR199600488A2 (tr) 1997-05-21
JPH11508244A (ja) 1999-07-21
CA2223869A1 (fr) 1996-12-27
EP0832061A1 (fr) 1998-04-01
MX9709951A (es) 1998-03-29
DK0832061T3 (da) 2001-11-19
DE69615025D1 (de) 2001-10-11
EP0832061B1 (fr) 2001-09-05
KR19990022448A (ko) 1999-03-25
ATE205185T1 (de) 2001-09-15
AU5911096A (en) 1997-01-09
WO1996041795A1 (fr) 1996-12-27

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